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Microwave-Assisted One-Pot Telescoped Synthesis of 2-Amino-1,3-thiazoles, Selenazoles, Imidazo[1,2-a]pyridines, and Other Heterocycles from Alcohols J. Org. Chem. (IF 3.6) Pub Date : 2024-03-18 Pablo Macías-Benítez, Alfonso Sierra-Padilla, Francisco M. Guerra, F. Javier Moreno-Dorado
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Construction of Phosphorothiolated 2-Pyrrolidinones via Photoredox/Copper-Catalyzed Cascade Radical Cyclization/Phosphorothiolation J. Org. Chem. (IF 3.6) Pub Date : 2024-03-18 Pengbo Zhang, Wenwu Li, Shuai Yang, Weilong Qu, Longyu Wang, Jinming Lin, Xia Gao
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Furan Dearomatization: A Route to Diverse Fluoroalkyl/Aryl Triazoles J. Org. Chem. (IF 3.6) Pub Date : 2024-03-18 Guanghai Cheng, Penggang Zhao, Hang Su, Abdul Wahab, Ziwei Gao, Jing Gou, Binxun Yu
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Construction of Seven-Membered Oxacycles Using a Rh(I)-Catalyzed Cascade C–C Formation/Cleavage of Cyclobutenol Derivatives J. Org. Chem. (IF 3.6) Pub Date : 2024-03-18 Jin Su Ham, Mina Son, Christina G. Na, Bohyun Park, Mu-Hyun Baik, Richmond Sarpong
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Acid-Mediated Domino Cyclization of ortho-Formyl Cinnamate Esters: Synthesis of Substituted Indene/Indane Esters and Indeno[a]indenones J. Org. Chem. (IF 3.6) Pub Date : 2024-03-18 Chander Shekhar, Gedu Satyanarayana
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Cycloaddition of Phenyltriazolinedione with Carbazole-Alkynes and Yne-Carbamates to Access Diazacyclobutenes J. Org. Chem. (IF 3.6) Pub Date : 2024-03-17 Brock A. Miller, Chandima J. Narangoda, Samuel Kwain, William T. Bridges, Monireh Noori, Erin E. Solomon, Alexis A. Bragg, Alex T. Sung, Yusuke Iwai, Lauren Ulisse, William H. Schmidt, Colin D. McMillen, Brian N. Dominy, Daniel C. Whitehead
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Visible Light-Induced 1,2-Diphenyldisulfane-Mediated Defluoroborylation of Polyfluoroarenes J. Org. Chem. (IF 3.6) Pub Date : 2024-03-16 Qiao-Jing Pan, Yu-Qi Miao, Hou-Ji Cao, Zhenxing Liu, Xuenian Chen
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Isomeric Benzenediol-Linked Organophosphonates as a Handy Reusable Emitting Platform: Diversity in Polyamine Vapor Detection J. Org. Chem. (IF 3.6) Pub Date : 2024-03-15 Akshita Jain, Pandiyan Sivasakthi, Pralok K. Samanta, Manab Chakravarty
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Pseudodiproline (Pro–Cyp) Oligomers Fold into Helical Polyproline Type secondary structures J. Org. Chem. (IF 3.6) Pub Date : 2024-03-15 Jean-Baptiste Garsi, Pedro M. Aguiar, Gilles Berger, Thierry Maris, Stephen Hanessian
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Asymmetric Synthesis of CIDD-0072424 via an Enantioselective Nitro-Mannich Reaction: A Central Nervous System Penetrant, Selective Small Molecule Inhibitor of Protein Kinase C Epsilon J. Org. Chem. (IF 3.6) Pub Date : 2024-03-15 Harmannus De Kraker, Hua-Yu Leo Wang, Hadi D. Arman, Rachel N. Renteria, Caleb N. Fleischer, Robert O. Messing, Stanton F. McHardy
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HFIP-Mediated Multicomponent Reactions: Synthesis of Pyrazole-Linked Thiazole Derivatives J. Org. Chem. (IF 3.6) Pub Date : 2024-03-14 Riddhiman Banerjee, Danish Ali, Nurabul Mondal, Lokman H. Choudhury
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Rapid Synthesis of 3-Methyleneisoindolin-1-ones via Metal-Free Tandem Reactions of Ester-Functionalized Aziridines J. Org. Chem. (IF 3.6) Pub Date : 2024-03-14 Siyang Xing, Changkun Jin, Panpan Zhang, Jingmeng Yang, Yuxia Liang, Xinglian Ao, Wenyi Pi, Kui Wang, Bolin Zhu
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Ruthenium-Induced Decomposition of Hexamethylenetetramine as a Tool for the Acid-Free Sommelet Reaction in Aqueous Medium J. Org. Chem. (IF 3.6) Pub Date : 2024-03-14 Preeti Devi, Vikas Dasharath Ghule, Senthilkumar Muthaiah
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Reductive Coupling of P(O)–H Compounds and Aldehydes for the General Synthesis of Phosphines and Phosphine Oxides J. Org. Chem. (IF 3.6) Pub Date : 2024-03-14 Jie Wang, Jing Xiao, Zi-Long Tang, Dong-Hui Lan, Li-Biao Han
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Cu(I) Complexes Catalyzed the Dehydrogenation of N-Heterocycles J. Org. Chem. (IF 3.6) Pub Date : 2024-03-14 Yangyang Shen, Fei Chen, Zhihong Du, Hao Zhang, Jichang Liu, Ning Liu
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A Water-Soluble Cryptophane Decorated with Aromatic Amine Groups Shows High Affinity for Cesium and Thallium(I) J. Org. Chem. (IF 3.6) Pub Date : 2024-03-14 Rajaa Benchouaia, Martin Doll, Patrick Berthault, Kévin Chighine, Estelle Léonce, Thierry Brotin, Nicolas De Rycke
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Quantification of Hydrogen-Bond-Donating Ability of Biologically Relevant Compounds J. Org. Chem. (IF 3.6) Pub Date : 2024-03-14 Cameron B. Berlin, Eesha Sharma, Marisa C. Kozlowski
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Rapid, Homogenous, B-Alkyl Suzuki–Miyaura Cross-Coupling of Boronic Esters J. Org. Chem. (IF 3.6) Pub Date : 2024-03-14 Matthew J. Bock, Scott. E. Denmark
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Asymmetric Total Synthesis of Cryptorigidifoliol I J. Org. Chem. (IF 3.6) Pub Date : 2024-03-14 Rodney A. Fernandes, Dashrath Jangid
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Three-Component Reaction between 3-Acetylcoumarins, Amines, and Elemental Sulfur: A Designed Approach to 3-Amino-4H-thieno[3,2-c]coumarins J. Org. Chem. (IF 3.6) Pub Date : 2024-03-12 Behnaz Farajpour, Roujin Heydarzadeh, Faiq H. S. Hussain, Behrouz Notash, Peiman Mirzaei, Morteza Shiri
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Computational Exploration of 1,2-Carboamine Carbonylation Catalyzed by Nickel J. Org. Chem. (IF 3.6) Pub Date : 2024-03-12 Yi-Wen Gu, Man Chen, Wei Deng, Zheng-Yang Xu
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Synthesis of Chirally Enriched Pyrazolylpyrimidinone-Based Glycohybrids via Annulation of Glycals with 2-Hydrazineylpyrimidin-4(3H)-ones J. Org. Chem. (IF 3.6) Pub Date : 2024-03-12 Ghanshyam Tiwari, Vinay Kumar Mishra, Ashish Khanna, Rajdeep Tyagi, Ram Sagar
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Catalytic Light-Driven Strategy for Transforming Oximes to Carbonyls J. Org. Chem. (IF 3.6) Pub Date : 2024-03-13 Brandon White, Travis Dudding
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Cascade Electrochemical Aerobic Oxygenation of 2-Substituted Indoles and Electrochemical [5 + 3] Annulation with Amidines: Access to Eight-Membered Benzo[1,3,5]triazocin-6(5H)-ones J. Org. Chem. (IF 3.6) Pub Date : 2024-03-13 Weihui Zhuang, Fengyi Xiao, Yumei Chen, Xiaofeng Zhang, Qiufeng Huang
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Regioselective Deacetylation of Peracetylated Deoxy-C-glycopyranosides by Boron Trichloride (BCl3) J. Org. Chem. (IF 3.6) Pub Date : 2024-03-13 Shuangyuan Chen, Feifei Wei, Xinqiang Cheng, Ying Luo, Fancui Meng, Yuanwen Zhang, Wenqian Huang, Jun Lv, Hong Pan, Qingqing Wu, Guilong Zhao
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Salicylaldehyde-Cobalt(II)-Catalyzed C–H Alkoxylation of Indoles with Secondary Alcohols J. Org. Chem. (IF 3.6) Pub Date : 2024-03-12 Mao-Gui Huang, Yu-Yan Tan, Meng-Ting Ai, Xiao-Hong Chen, Hai-Bing Xu, Yue-Jin Liu
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A Mild and Modular Approach to the Total Synthesis of Desferrioxamine B J. Org. Chem. (IF 3.6) Pub Date : 2024-03-12 Todd E. Markham, Rachel Codd
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Unsymmetrical Benzothieno-Fused BODIPYs as Efficient NIR Heavy-Atom-Free Photosensitizers J. Org. Chem. (IF 3.6) Pub Date : 2024-03-12 Xiaofan Fu, Yingxiu Man, Changjiang Yu, Yingzhu Sun, Erhong Hao, Qinghua Wu, Anzhi Hu, Guangyao Li, Chang-Cheng Wang, Jiazhu Li
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Iridium-Catalyzed Asymmetric Hydrogenation of Heteroaromatics with Multiple N Atoms via Substrate Activation: An Entry to 4,5,6,7-Tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonitrile Core of a Potent BTK Inhibitor J. Org. Chem. (IF 3.6) Pub Date : 2024-03-11 Mu-Wang Chen, Hong-Wang Li, Ying-Qi Wang, Bo Wu, Zheng Liu, Xinzhong Lai, Joerg Deerberg, Yong-Gui Zhou
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Tetraethylammonium Salts as Solid, Easy to Handle Ethylene Precursors and Their Application in Mizoroki–Heck Coupling J. Org. Chem. (IF 3.6) Pub Date : 2024-03-11 Eleni Papaplioura, Maëva Mercier, Michael E. Muratore, Tobias Biberger, Soufyan Jerhaoui, Michael Schnürch
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Regioselective Fluorohydrin Synthesis from Allylsilanes and Evidence for a Silicon–Fluorine Gauche Effect J. Org. Chem. (IF 3.6) Pub Date : 2024-03-08 Alexie W. Clover, Adam P. Jones, Robert F. Berger, Werner Kaminsky, Gregory. W. O’Neil
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Stereodivergent Synthesis of Alkaloid (±)-223A and (±)-6-epi-223A via Rh-Catalyzed Hydroformylation Double Cyclization J. Org. Chem. (IF 3.6) Pub Date : 2024-03-08 Wen-Wei Huang, Jui-Teng Cheng, Wei-Ting Hsiao, Wen-Hua Chiou
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Photoinduced Alkylsulfonylation and Cyanoalkylsulfonylation of Morita–Baylis–Hillman Adducts via Multicomponent Insertion of Sulfur Dioxide J. Org. Chem. (IF 3.6) Pub Date : 2024-03-08 Zhi-Jie Song, Yu Bao, Yun-Jia Sun, Shenghu Yan, Yue Zhang, Guigen Li, Jia-Yin Wang
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Synthesis and Characterization of a [1,2,6]Diazaphosphonine Oxide: An Example of a Photoswitchable Phosphorus-Containing Cyclic Azobenzene J. Org. Chem. (IF 3.6) Pub Date : 2024-03-07 Nawel Goual, Stéphane Maisonneuve, Pascal Retailleau, Juan Xie, Angela Marinetti, Arnaud Voituriez
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Anhydrous and Stereoretentive Fluoride-Enhanced Suzuki–Miyaura Coupling of Immunomodulatory Imide Drug Derivatives J. Org. Chem. (IF 3.6) Pub Date : 2024-03-07 William F. Tracy, Geraint H. M. Davies, Lauren N. Grant, Jacob M. Ganley, Jesus Moreno, Emily C. Cherney, Huw M. L. Davies
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Synthesis and Chemoinformatic Analysis of Fluorinated Piperidines as 3D Fragments for Fragment-Based Drug Discovery J. Org. Chem. (IF 3.6) Pub Date : 2024-03-07 Myriam Le Roch, Jacques Renault, Gilles Argouarch, Elena Lenci, Andrea Trabocchi, Thierry Roisnel, Nicolas Gouault, Claudia Lalli
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At the Speed of Light: The Systematic Implementation of Photoredox Cross-Coupling Reactions for Medicinal Chemistry Research J. Org. Chem. (IF 3.6) Pub Date : 2024-03-05 Nathan J. Gesmundo, Alexander J. Rago, Jonathon M. Young, Sebastian Keess, Ying Wang
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Unraveling the Prominent Existence of Trace Metals in Photocatalysis: Exploring Iron Impurity Effects J. Org. Chem. (IF 3.6) Pub Date : 2024-03-07 Yahao Huang, Miao Wang, Wei Liu, Qiang Wu, Peng Hu
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Electrochemical Synthesis of Selenosulfonates from Diselenides and Sulfonyl Hydrazides J. Org. Chem. (IF 3.6) Pub Date : 2024-03-07 Jin-Feng Lv, Yang Deng, Xin-Yi Liang, Yu-Fang Tan, Yan-Hong He, Zhi Guan
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Organophotoredox Catalysis: Switchable Radical Generation from Alkyl Sodium Sulfinates for Sulfonylation and Alkylative Activation of C–C Bonds of Cyclopropenes J. Org. Chem. (IF 3.6) Pub Date : 2024-03-06 Palasetty Chandu, Sourabh Biswas, Koustav Pal, Devarajulu Sureshkumar
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Visible Light-Induced One-Pot Carbonylation of Alkyl Halides with Aryl Formates J. Org. Chem. (IF 3.6) Pub Date : 2024-03-06 Padon Chuentragool, Aurapat Ngamnithiporn, Prachnawadee Hongboon, Somsak Ruchirawat
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Heterogeneous Photocatalytic Ring Expansion of Cyclic Ketones for the Construction of Medium-Sized Lactams J. Org. Chem. (IF 3.6) Pub Date : 2024-03-06 Mengzhen Dang, Ruizhi Jia, Kai Tan, Danyang Hao, Wenjing Yang, Cong-Ying Zhou, Zhen Guo
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Organo-Photoredox Catalyzed gem-Difluoroallylation of Glycine and Glycine Residue in Peptides J. Org. Chem. (IF 3.6) Pub Date : 2024-03-06 Ruofan Lin, Yujie Shan, Yan Li, Xian Wei, Yue Zhang, Yuqian Lin, Yiman Gao, Weiwei Fang, Jing-Jing Zhang, Ting Wu, Lingchao Cai, Zhen Chen
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Electrochemical Multicomponent Cascade Reaction for the Synthesis of Selenazol-2-amines with Elemental Selenium J. Org. Chem. (IF 3.6) Pub Date : 2024-03-06 Hong-Tao Ji, Jun Jiang, Wei-Bao He, Yu-Han Lu, Yuan-Yuan Liu, Xiao Li, Wei-Min He
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Generation of Carbonyl Compounds from Oximes through Electrooxidative Deoximation J. Org. Chem. (IF 3.6) Pub Date : 2024-03-06 Yeliang Xue, Shaozhong Wang
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Synthesis of C3v-Symmetrical 1,3,5-Tris-Protected Calix[6]arene-Based Molecular Platforms J. Org. Chem. (IF 3.6) Pub Date : 2024-03-06 Martin Lepeintre, Julie Champciaux, Benoit Colasson, Ivan Jabin
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Preparation of a Key Intermediate En Route to the Anti-HIV Drug Lenacapavir J. Org. Chem. (IF 3.6) Pub Date : 2024-03-06 Juan C. Caravez, Yuting Hu, Erfan Oftadeh, Kirubel T. Mamo, Bruce H. Lipshutz
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A Disconnection for Rapid Access to Heterocyclic Benzylic Amines with Fully Substituted α-Carbons J. Org. Chem. (IF 3.6) Pub Date : 2024-03-05 Shouliang Yang, Fen Wang, Stephanie Scales, Michelle Tran-Dubé, Madeline Berry, Haiwei Xu, Feng Tang, Liangliang Xue, Zhongwei Ma, Bryan Li, Indrawan McAlpine
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Intramolecular Heteroatom and Styryl Diels–Alder Reactions, Asymmetric Cycloadditions of Chiral 3-Phenylallyl Maleic Esters J. Org. Chem. (IF 3.6) Pub Date : 2024-03-05 Peter Mpaata, Chandler R. Miller, Dickson K. Bonsrah, Alexander B. Camp, Karson M. Ballard, Liahona Angelie, Justin Kirkland, Jyothish Joy, William J. Hirschi, Stacey J. Smith, Daniel H. Ess, Merritt B. Andrus
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Visible Light Mediated Organophotoredox Catalyzed Synthesis of Tetraketones Using Tertiary Amines as Alkyl Synthons J. Org. Chem. (IF 3.6) Pub Date : 2024-03-05 Shankhajit Mondal, Akanksha M. Pandey, Boopathy Gnanaprakasam
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Synthetic Utilization of 2H-Heptafluoropropane: Ionic 1,4-Addition to Electron-Deficient Carbon–Carbon Unsaturated Bonds J. Org. Chem. (IF 3.6) Pub Date : 2024-03-05 Yusuke Higashi, Kotono Shima, Mikiya Suzuki, Moe Fujishiro, Tsuyoshi Kawai, Tsumoru Morimoto
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Conformational Analysis Explores the Role of Electrostatic Nonclassical CF···HC Hydrogen Bonding Interactions in Selectively Halogenated Cyclohexanes J. Org. Chem. (IF 3.6) Pub Date : 2024-03-05 Mengfan He, Bruno A. Piscelli, Rodrigo A. Cormanich, David O’Hagan
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Photochemical C(sp3)–H Activation for Diversity-Oriented Synthesis of 3-Functionalized Oxindoles J. Org. Chem. (IF 3.6) Pub Date : 2024-03-05 Hao Hou, Wei Ou, Chenliang Su
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Minisci-Type Dehydrogenative Coupling of N-Heteroaromatic Rings with Inert C(sp3)–H Enabled by a Visible-Light-Catalyzed Intermolecular Hydrogen Atom Transfer Process J. Org. Chem. (IF 3.6) Pub Date : 2024-03-05 Jun-Feng Yang, Yun-Fei Liu, Lin-Lin Wei, Kai-Kai Qiao, Yan-Qiu Zhao, Lei Shi
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Total Synthesis and Determination of the Absolute Configuration of Berkeleylactone I J. Org. Chem. (IF 3.6) Pub Date : 2024-03-04 Sudip Mandal, Dora Mahananda, Dileep Paladugu, Barla Thirupathi
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Synthesis of Dihydroquinoxalinones from Biomass-Derived Keto Acids and o-Phenylenediamines J. Org. Chem. (IF 3.6) Pub Date : 2024-03-04 Wenfeng Zhao, Hu Li, Qingmei Ge, Hang Cong, Song Yang
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De Novo Access to BODIPY C-Glycosides as Linker-Free Nonsymmetrical BODIPY-Carbohydrate Conjugates J. Org. Chem. (IF 3.6) Pub Date : 2024-03-04 Clara Uriel, Dylan Grenier, Florian Herranz, Natalia Casado, Jorge Bañuelos, Esther Rebollar, Inmaculada Garcia-Moreno, Ana M. Gomez, J. Cristobal López
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Asymmetric Brominative Dearomatization of 2-Naphthols Using a Cinchona Alkaloid-Based Organocatalyst J. Org. Chem. (IF 3.6) Pub Date : 2024-03-04 Kouhei Omae, Yoshihiro Miyake, Mio Shimogaki
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Visible-Light-Promoted Selenylation/Cyclization of o-Alkynyl Benzylazides/o-Propargyl Arylazides: Synthesis of Seleno-Substituted Isoquinolines and Quinolines J. Org. Chem. (IF 3.6) Pub Date : 2024-03-04 Xi-Rui Gong, Shuang-Shuang Sun, Mei-Lin Ren, Qiao-Yan Wu, Yan-Yan Chen, Yan-Li Xu
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A Perspective on Being Black and in STEM J. Org. Chem. (IF 3.6) Pub Date : 2024-03-01 Aria Gonzalez
When I was a child, I checked out a book containing an exhaustive list of all of the types of scientists. As I flipped through page after page, the descriptions that caught my eye one after the other were related to health-based research. I remember telling my dad that when I grew up I would become a scientist and cure the common cold─because I hated getting sick. He humored me, saying if I managed