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Chromones bearing amino acid residues: Easily accessible and potent inhibitors of the breast cancer resistance protein ABCG2 Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-05 Emile Roussel; Alexis Moréno; Nicolas Altounian; Christian Philouze; Basile Pérès; Aline Thomas; Olivier Renaudet; Pierre Falson; Ahcène Boumendjel
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New manganese(II), iron(II), cobalt(II), nickel(II) and copper(II) saccharinate complexes of 2,6-bis(2-benzimidazolyl)pyridine as potential anticancer agents Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-03 Ceyda Icsel; Veysel T. Yilmaz; Şeyma Aydinlik; Muhittin Aygun
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The design, synthesis and anti-tumor mechanism study of new androgen receptor degrader Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-10 Hang Xie; Jian-Jia Liang; Ya-Lei Wang; Tian-Xing Hu; Jin-Yi Wang; Rui-Hua Yang; Jun-Ke Yan; Qiu-Rong Zhang; Xia Xu; Hong-Min Liu; Yu Ke
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Structure-activity relationships of Wee1 inhibitors: A review Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-10 Xingkai Du; Jian Li; Xiaojiao Luo; Rong Li; Feng Li; Yiwen Zhang; Jianyou Shi; Jun He
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Natural and synthetic coumarins as antileishmanial agents: A review Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-09 Guilherme Arraché Gonçalves; Adriano Ronchi Spillere; Gustavo Machado das Neves; Luciano Porto Kagami; Gilsane Lino von Poser; Rômulo Faria Santos Canto; Vera Lucia Eifler-Lima
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Design, synthesis and biological evaluation of rasagiline-clorgyline hybrids as novel dual inhibitors of monoamine oxidase-B and amyloid-β aggregation against Alzheimer’s disease Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-30 Sai-Sai Xie; Jing Liu; Chunli Tang; Chengyun Pang; Qing Li; Yuelian Qin; Xiaojie Nong; Zhipeng Zhang; Jie Guo; Maojun Cheng; Weizhong Tang; Ningsheng Liang; Neng Jiang
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Synthesis, antiproliferative activity and SAR analysis of (−)-cleistenolide and analogues Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-06 Goran Benedeković; Mirjana Popsavin; Ivana Kovačević; Vesna Kojić; Marko Rodić; Velimir Popsavin
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8-Alkynyl-3-nitroimidazopyridines display potent antitrypanosomal activity against both T. b. brucei and cruzi Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-08 Cyril Fersing; Clotilde Boudot; Caroline Castera-Ducros; Emilie Pinault; Sébastien Hutter; Romain Paoli-Lombardo; Nicolas Primas; Julien Pedron; Line Seguy; Sandra Bourgeade-Delmas; Alix Sournia-Saquet; Jean-Luc Stigliani; Jean-Yves Brossas; Luc Paris; Alexis Valentin; Susan Wyllie; Alan H. Fairlamb; Élisa Boutet-Robinet; Patrice Vanelle
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Natural and nature-inspired stilbenoids as antiviral agents Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-04 Luce M. Mattio; Giorgia Catinella; Andrea Pinto; Sabrina Dallavalle
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Anticancer fungal natural products: Mechanisms of action and biosynthesis Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-02 Siwen Yuan; Jannu Vinay Gopal; Shuya Ren; Litong Chen; Lan Liu; Zhizeng Gao
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Design, synthesis and anti-inflammatory activity of 3-amino acid derivatives of ocotillol-type sapogenins Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-26 Gangqiang Yang; Meng Gao; Yixiao Sun; Conghui Wang; Xiaojuan Fang; Hongyan Gao; Wenshuang Diao; Hui Yu
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Design, synthesis, and bioevaluation of pyrazolo[1,5-a]pyrimidine derivatives as tubulin polymerization inhibitors targeting the colchicine binding site with potent anticancer activities Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-27 Gang Li; Yuxi Wang; Ling Li; Yichang Ren; Xin Deng; Jin Liu; Wei Wang; Meihua Luo; Shuwen Liu; Jianjun Chen
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F10, a new camptothecin derivative, was identified as a new orally–bioavailable, potent antitumor agent Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-05 Shu Fan; Yong-Xiao Cao; Guang-Yan Li; Hao Lei; Mawusse K.I. Attiogbe; Jing-Chun Yao; Xue-Yan Yang; Yan-Jie Liu; Yuan-Yuan Hei; Hao Zhang; Lei Cao; Xiao-Yan Zhang; Shuai-Shuai Du; Gui-Min Zhang; San-Qi Zhang
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Design, synthesis, and evaluation of amphiphilic sofalcone derivatives as potent Gram-positive antibacterial agents Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-08 Shuimu Lin; Yongzhi Chen; Hongxia Li; Jiayong Liu; Shouping Liu
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Design, synthesis, and biological evaluation of aryl piperazines with potential as antidiabetic agents via the stimulation of glucose uptake and inhibition of NADH:ubiquinone oxidoreductase Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-27 R. Devine; M. Kelada; S. Leonard; D.S.D. Martin; J.M.D. Walsh; C.J. Breen; R.B. Driver; G.K. Kinsella; J.B.C. Findlay; J.C. Stephens
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Synthesis, bioevaluation and docking studies of some 2-phenyl-1H-benzimidazole derivatives as anthelminthic agents against the nematode Teladorsagia circumcincta Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-07 Nerea Escala; Elora Valderas-García; María Álvarez Bardón; Verónica Castilla Gómez de Agüero; Ricardo Escarcena; José Luis López-Pérez; Francisco A. Rojo-Vázquez; Arturo San Feliciano; Rafael Balaña-Fouce; María Martínez-Valladares; Esther del Olmo
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Chlorine substituents and linker topology as factors of 5-HT6R activity for novel highly active 1,3,5-triazine derivatives with procognitive properties in vivo Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-06 Sylwia Sudoł; Katarzyna Kucwaj-Brysz; Rafał Kurczab; Natalia Wilczyńska; Magdalena Jastrzębska-Więsek; Grzegorz Satała; Gniewomir Latacz; Monika Głuch-Lutwin; Barbara Mordyl; Ewa Żesławska; Wojciech Nitek; Anna Partyka; Kamila Buzun; Agata Doroz-Płonka; Anna Wesołowska; Anna Bielawska; Jadwiga Handzlik
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Rationally Engineered Prolyl Endopeptidases from Sphingomonas Capsulata with Improved Hydrolytic Activity towards Pathogenic Peptides of Celiac Diseases Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-06 Bin Xiao; Chun Zhang; Xiaotong Song; Miao Wu; Jianping Mao; Rong Yu; Yongxiang Zheng
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Design and synthesis of 1H-indazole-3-carboxamide derivatives as potent and selective PAK1 inhibitors with anti-tumour migration and invasion activities Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-06 Mingliang Zhang; Xiaobao Fang; Cong Wang; Chen Huang; Meng Wang; Lu Zhu; Zixu Wang; Yuhan Gao; Tianyi Zhang; Haichun Liu; Yanmin Zhang; Shuai Lu; Tao Lu; Yadong Chen; Hongmei Li
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Design, synthesis and antitumor activity of novel thiophene-pyrimidine derivatives as EGFR inhibitors overcoming T790M and L858R/T790M mutations Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-06 Zhen Xiao; Zhihui Zhou; Cilong Chu; Qian Zhang; Lingjia Zhou; Zunhua Yang; Xin Li; Liying Yu; Pengwu Zheng; Shan Xu; Wufu Zhu
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Synthesis and evaluation of Na+/K+-ATP-ase inhibiting and cytotoxic in vitro activities of oleandrigenin and its selected 17β-(butenolidyl)- and 17β-(3-furyl)- analogues Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-22 Karol Michalak; Lucie Rárová; Martin Kubala; Tereza Štenclová; Miroslav Strnad; Jerzy Wicha
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Recent progress in Keap1-Nrf2 Protein-protein Interaction Inhibitors Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-06 Yi Mou; Shuai Wen; Yu-Xiu Li; Xin-Xing Gao; Xin Zhang; Zheng-Yu Jiang
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A novel pipeline of 2-(benzenesulfonamide)-N-(4-hydroxyphenyl) acetamide analgesics that lack hepatotoxicity and retain antipyresis Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-30 Hernan A. Bazan; Surjyadipta Bhattacharjee; Carolina Burgos; Javier Recio; Valentina Abet; Amanda R. Pahng; Bokkyoo Jun; Jessica Heap; Alexander J. Ledet; William C. Gordon; Scott Edwards; Dennis Paul; Julio Alvarez-Builla; Nicolas G. Bazan
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Structure guided design and synthesis of furyl thiazolidinedione derivatives as inhibitors of GLUT 1 and GLUT 4, and evaluation of their anti-leukemic potential Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-02 Kalpana Tilekar; Neha Upadhyay; Jessica D. Hess; Lucasantiago Henze Macias; Piotr Mrowka; Renato J. Aguilera; Franz-Josef Meyer-Almes; Cristina V. Iancu; Jun-yong Choe; C.S. Ramaa
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Hit-to-lead optimization of a latency-associated nuclear antigen inhibitor against Kaposi’s sarcoma-associated herpesvirus infections Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-28 Philine Kirsch; Saskia C. Stein; Aylin Berwanger; Julia Rinkes; Valentin Jakob; Thomas F. Schulz; Martin Empting
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Discovery of carboxyl-containing biaryl ureas as potent RORγt inverse agonists Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-05 Nannan Sun; Yafei Huang; Mingcheng Yu; Yunpeng Zhao; Ji-An Chen; Chenyu Zhu; Meiqi Song; Huimin Guo; Qiong Xie; Yonghui Wang
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Discovery of MGS0274, an ester prodrug of a metabotropic glutamate receptor 2/3 agonist with improved oral bioavailability Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-05 Hiroki Urabe; Naoki Miyakoshi; Norikazu Ohtake; Akiko Nozoe; Motoki Ochi; Misako Fukasawa; Kohnosuke Kinoshita; Jun-ichi Yamaguchi; Toshiyuki Marumo; Hirohiko Hikichi; Shigeyuki Chaki; Takashi Hashihayata
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Targeting topoisomerase II with trypthantrin derivatives: Discovery of 7-((2-(dimethylamino)ethyl)amino)indolo[2,1-b]quinazoline-6,12-dione as an antiproliferative agent and to treat cancer Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-04 Elena Catanzaro; Nibal Betari; Jose M. Arencibia; Serena Montanari; Claudia Sissi; Angela De Simone; Ivano Vassura; Alan Santini; Vincenza Andrisano; Vincenzo Tumiatti; Marco De Vivo; Dmitri V. Krysko; Marco B.L. Rocchi; Carmela Fimognari; Andrea Milelli
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Synthesis, structure and anticancer activity of new geldanamycin amine analogs containing C(17)- or C(20)- flexible and rigid arms as well as closed or open ansa-bridges Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-03 Natalia Skrzypczak; Krystian Pyta; Piotr Ruszkowski; Maria Gdaniec; Franz Bartl; Piotr Przybylski
The nucleophilic attack of amines at C(17) or C(17)/C(20) positions of geldanamycin’s (GDM) benzoquinone, via initial 1,4-Michael conjugate addition mechanism, yield new analogs with closed or open ansa-bridges (1-31), respectively. X-ray structures of analogs 22 and 24 reveals an unexpected arrangement of the ansa-bridge in solid (conformer B), that is located between those of conformers A, prevailing
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Design, synthesis and antimicrobial evaluation of novel glycosylated-fluoroquinolones derivatives Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-27 Aya A.M. Mohammed; Ghadeer A.R.Y. Suaifan; Mayadah B. Shehadeh; Patrick N. Okechukwu
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Design, synthesis and antitumour evaluation of pyrrolo[1,2-f]-phenanthridine and dibenzo[f,h]pyrrolo[1,2-b]isoquinoline derivatives Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-23 Anilkumar S. Patel; Vicky Jain; Vaikar Navakanth Rao; Yi-Wen Lin; Anamik Shah; Kuo-Chu Lai; Tsann-Long Su; Te-Chang Lee
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Synthesis of indole inhibitors of silent information regulator 1 (SIRT1), and their evaluation as cytotoxic agents Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-02 Hanna Laaroussi; Ying Ding; Teng Yuou; Patrick Deschamps; Michel Vidal; Peng Yu; Sylvain Broussy
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Bioisosterism-based design and enantiomeric profiling of chiral hydroxyl-substituted biphenyl-diarylpyrimidine nonnucleoside HIV-1 reverse transcriptase inhibitors Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-02 Xiaomei Chen; Li Ding; Yuan Tao; Christophe Pannecouque; Erik De Clercq; Chunlin Zhuang; Fen-Er Chen
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Development of a metabolically stable topoisomerase I poison as anticancer agent Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-07-02 Biswajit Kundu; Dipayan Sarkar; Srijita Paul Chowdhuri; Sourav Pal; Subhendu K. Das; Benu Brata Das; Arindam Talukdar
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Design, synthesis and biological evaluation of 4-aniline quinazoline derivatives conjugated with hydrogen sulfide (H2S) donors as potent EGFR inhibitors against L858R resistance mutation Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-27 You-Guang Zheng; Wu-Qi Zhang; Long Meng; Xiao-Qing Wu; Ling Zhang; Lin An; Cheng-Lin Li; Cai-Yun Gao; Liang Xu; Yi Liu
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Identification of dibucaine derivatives as novel potent enterovirus 2C helicase inhibitors: In vitro, in vivo, and combination therapy study Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-25 Qi Tang; Zhichao Xu; Mengyu Jin; Ting Shu; Yinuo Chen; Leilei Feng; Qiuhan Zhang; Ke Lan; Shuwen Wu; Hai-Bing Zhou
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Drug repurposing: Discovery of troxipide analogs as potent antitumor agents Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-26 Nan Lu; Jin-ling Huo; Shuai Wang; Xiao-Han Yuan; Hong-Min Liu
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Oligosaccharide-camptothecin conjugates as potential antineoplastic drugs: Design, synthesis and biological evaluation Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-30 Maolin Li; Wenchong Ye; Kaishuo Fu; Cui zhou; Yonghui Shi; Weiping Huang; Wenming Chen; Jiliang Hu; Zhilin Jiang; Wen Zhou
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Rational modification, synthesis and biological evaluation of 3,4-dihydroquinoxalin-2(1H)-one derivatives as potent and selective c-Jun N-terminal kinase 3 (JNK3) inhibitors Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-26 Xiaodong Dou; Huixia Huang; Lan Jiang; Guiwang Zhu; Hongwei Jin; Ning Jiao; Liangren Zhang; Zhenming Liu; Lihe Zhang
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The importance of indole and azaindole scaffold in the development of antitumor agents Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-28 Yu Han; Wei Dong; Qunqun Guo; Xiufen Li; Longjiang Huang
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Medicinal chemistry insights into novel CDC25 inhibitors Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-04-26 Yucen Tao; Xia Hao; Xiao Ding; Srinivasulu Cherukupalli; Yuning Song; Xinyong Liu; Peng Zhan
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Rosuvastatin based novel 3-substituted isocoumarins / 3-alkylidenephthalides: Ultrasound assisted synthesis and identification of new anticancer agents Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-14 Jetta Sandeep Kumar; B. Thirupataiah; Raghavender Medishetti; Aramita Ray; Shilpak Dilip Bele; Kazi Amirul Hossain; Gangireddy Sujeevan Reddy; Rebecca Kristina Edwin; Alex Joseph; Nitesh Kumar; Gautham G. Shenoy; C. Mallikarjuna Rao; Manojit Pal
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Structure–activity relationship and hypoglycemic activity of tricyclic matrines with advantage of treating diabetic nephropathy Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-24 Sheng Tang; Can Wang; Ying–Hong Li; Tian–Yu Niu; Yuan–Hui Zhang; Yu–Dong Pang; Yan–Xiang Wang; Wei–Jia Kong; Dan–Qing Song
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Design, synthesis and biological evaluation of novel potent STAT3 inhibitors based on BBI608 for cancer therapy Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-25 Kai-Rui Feng; Feng Wang; Xin-Wei Shi; Yun-Xuan Tan; Jia-Ying Zhao; Jian-Wei Zhang; Qing-Hua Li; Guo-Qiang Lin; Dingding Gao; Ping Tian
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Structure-based design, semi-synthesis and anti-inflammatory activity of tocotrienolic amides as 5-lipoxygenase inhibitors Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-27 Chau Phi Dinh; Alexia Ville; Konstantin Neukirch; Guillaume Viault; Veronika Temml; Andreas Koeberle; Oliver Werz; Daniela Schuster; Hermann Stuppner; Pascal Richomme; Jean-Jacques Helesbeux; Denis Séraphin
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Pyrido[2,3-b][1,5]benzoxazepin-5(6H)-one derivatives as CDK8 inhibitors Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-20 Sonia Martínez-González; Ana Belén García; M. Isabel Albarrán; Antonio Cebriá; Adrián Amezquita-Alves; Francisco Javier García-Campos; Jaime Martínez-Gago; Jorge Martínez-Torrecuadrada; Inés Muñoz; Carmen Blanco-Aparicio; Joaquín Pastor
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Design, Diversity-Oriented Synthesis and Biological Evaluation of Novel Heterocycle Derivatives as Non-nucleoside HBV Capsid Protein Inhibitors Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-26 Haiyong Jia; Ji Yu; Xianhong Du; Srinivasulu Cherukupalli; Peng Zhan; Xinyong Liu
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Recent researches for dual Aurora target inhibitors in antitumor field Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-26 Maoyu Liu; Xueming Ju; Jing Zou; Jiangyou Shi; Guiqing Jia
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β-Lactams as promising anticancer agents: Molecular hybrids, structure activity relationships and potential targets Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-23 Dong-Jun Fu; Yun-Feng Zhang; An-Qi Chang; Jun Li
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Evaluation of N-Phenyl-2-aminothiazoles for Treatment of Multi-Drug Resistant and Intracellular Staphylococcus aureus Infections Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-25 Inas G. Shahin; Nader S. Abutaleb; Marwa Alhashimi; Asmaa E. Kassab; Khaled O. Mohamed; Azza T. Taher; Mohamed N. Seleem; Abdelrahman S. Mayhoub
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Discovery of simplified benzazole fragments derived from the marine benzosceptrin B as necroptosis inhibitors involving the receptor interacting protein Kinase-1 Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-25 Mohamed Benchekroun; Ludmila Ermolenko; Minh Quan Tran; Agathe Vagneux; Hristo Nedev; Claire Delehouzé; Mohamed Souab; Blandine Baratte; Béatrice Josselin; Bogdan I. Iorga; Sandrine Ruchaud; Stéphane Bach; Ali Al-Mourabit
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Synthesis, structure and anti-cancer activity of osmium complexes bearing π-bound arene substituents and phosphane Co-Ligands: A review Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-05-28 Tomiris Nabiyeva; Christoph Marschner; Burgert Blom
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Synthesis and biological evaluation of diaryl urea derivatives designed as potential anticarcinoma agents using de novo structure-based lead optimization approach Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-24 Fereshteh Azimian; Maryam Hamzeh-Mivehroud; Javid Shahbazi Mojarrad; Salar Hemmati; Siavoush Dastmalchi
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Discovery of highly potent and selective antiparasitic new oxadiazole and hydroxy-oxindole small molecule hybrids Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-05-16 Fábio S. Fernandes; Hugo Santos; Samia R. Lima; Caroline Conti; Manoel T. Rodrigues; Lucas A. Zeoly; Leonardo L.G. Ferreira; Renata Krogh; Adriano D. Andricopulo; Fernando Coelho
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The structure-based optimization of δ-sultone-fused pyrazoles as selective BuChE inhibitors. Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-12 Ziwen Zhang,Jingli Min,Mengdie Chen,Xia Jiang,Yingying Xu,Huali Qin,Wenjian Tang
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Development of small-molecule inhibitors of fatty acyl-AMP and fatty acyl-CoA ligases in Mycobacterium tuberculosis Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-13 Marzena Baran; Kimberly D. Grimes; Paul A. Sibbald; Peng Fu; Helena I.M. Boshoff; Daniel J. Wilson; Courtney C. Aldrich
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Targeting Fungal Virulence Factor by Small Molecules: Structure-based Discovery of Novel Secreted Aspartic Protease 2 (SAP2) Inhibitors Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-21 Chenglan Li; Yang Liu; Shancao Wu; Guiyan Han; Jie Tu; Guoqiang Dong; Na Liu; Chunquan Sheng
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Fight against novel coronavirus: A perspective of medicinal chemists. Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-12 Sk Abdul Amin,Tarun Jha
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Synthesis and biological evaluation of thiophenylbenzofuran derivatives as potential P-glycoprotein inhibitors. Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-06 Chin-Chuan Hung,Chien-Yu Chen,Yu-Chieh Wu,Chien-Fu Huang,Yu-Chun Huang,Ying-Chieh Chen,Chih-Shiang Chang
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Synthesis of adenine dinucleosides SAM analogs as specific inhibitors of SARS-CoV nsp14 RNA cap guanine-N7-methyltransferase. Eur. J. Med. Chem. (IF 5.572) Pub Date : 2020-06-12 Rostom Ahmed-Belkacem,Priscila Sutto-Ortiz,Mathis Guiraud,Bruno Canard,Jean-Jacques Vasseur,Etienne Decroly,Françoise Debart
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