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Construction of Switch Modules for CAR-T Cell Treatment Using a Site-Specific Conjugation System Bioconjugate Chem. (IF 4.7) Pub Date : 2024-04-25 Tuersunayi Abudureheman, Hang Zhou, Li-Ting Yang, Xiu-Song Huang, Jun-Jie Jing, Cai-Wen Duan, Kai-Ming Chen
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Light-Activated Nanodiamond-Based Drug Delivery Systems for Spatiotemporal Release of Antisense Oligonucleotides Bioconjugate Chem. (IF 4.7) Pub Date : 2024-04-24 Hoi Man Leung, Ling Sum Liu, Yuzhen Cai, Xinru Li, Yizhi Huang, Hoi Ching Chu, Y Rebecca Chin, Pik Kwan Lo
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Moving Beyond Isothiocyanates: A Look at the Stability of Conjugation Links Toward Radiolysis in 89Zr-Labeled Immunoconjugates Bioconjugate Chem. (IF 4.7) Pub Date : 2024-04-24 Romane Vizier, Pierre Adumeau, Mathieu Moreau, Victor Goncalves, Franck Denat
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Broadening the Utility of Farnesyltransferase-Catalyzed Protein Labeling Using Norbornene–Tetrazine Click Chemistry Bioconjugate Chem. (IF 4.7) Pub Date : 2024-04-23 Shelby A. Auger, Sneha Venkatachalapathy, Kiall Francis G. Suazo, Yiao Wang, Alexander W. Sarkis, Kaitlyn Bernhagen, Katarzyna Justyna, Jonas V. Schaefer, James W. Wollack, Andreas Plückthun, Ling Li, Mark D. Distefano
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Polyphenol-Assisted Biomineralization of Metal–Organic Framework Nanoparticles for Precision Delivery of Therapeutic Proteins to Cancer Cells Bioconjugate Chem. (IF 4.7) Pub Date : 2024-04-22 Tianli Luo, Qizhen Zheng, Ji Liu, Rui Yao, Ming Wang
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18F-Radiolabeling and Evaluation of an AMD3465 Derivative for PET Imaging of CXCR4 in a Mouse Breast Tumor Model Bioconjugate Chem. (IF 4.7) Pub Date : 2024-04-18 Huiqiang Li, Xiaochen Li, Lingyi Sun, Yanjie He, Li Wang, Yongju Gao, Dexing Zeng, Xinchang Pang, Junling Xu
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Dual Drug Delivery for Augmenting Bacterial Wound Complications via Tailored Ultradeformable Carriers Bioconjugate Chem. (IF 4.7) Pub Date : 2024-04-16 Kanika Arora, Bharti Dhruw, Sherilraj PM, Prasoon Madhukar, Shyam Sundar, Shyam Lal Mudavath
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Revival of Bioengineered Proteins as Carriers for Nucleic Acids Bioconjugate Chem. (IF 4.7) Pub Date : 2024-04-15 David Scherer, Michael Burger, Jean-Christophe Leroux
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Legumain-Triggered Macrocyclization of Radiofluorinated Tracer for Enhanced PET Imaging Bioconjugate Chem. (IF 4.7) Pub Date : 2024-04-10 Xiaoqing Gao, Qianhui Wang, Xiaofeng Yang, Jing Fang, Huirong Li, Hongjie Xi, Jianguo Lin, Ling Qiu
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Design and Biological Evaluation of the Long-Acting C5-Inhibited Ornithodoros moubata Complement Inhibitor (OmCI) Modified with Fatty Acid Bioconjugate Chem. (IF 4.7) Pub Date : 2024-04-09 Wenwen Shangguan, Xiaowan Li, Yandan Wang, Zongqing Huang, Yuanzhen Dong, Meiqing Feng, Jun Feng
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Adapting Ferritin, a Naturally Occurring Protein Cage, to Modulate Intrinsic Agonism of OX40 Bioconjugate Chem. (IF 4.7) Pub Date : 2024-04-09 Whitney Shatz-Binder, Caleigh M. Azumaya, Brandon Leonard, Ivan Vuong, Jawahar Sudhamsu, Alexis Rohou, Peter Liu, Wendy Sandoval, Karenna Bol, Saeed Izadi, Patrick G. Holder, Craig Blanchette, Remo Perozzo, Robert F. Kelley, Yogeshvar Kalia
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Noninvasive Analysis of Peptidoglycan from Living Animals Bioconjugate Chem. (IF 4.7) Pub Date : 2024-04-09 Karl L. Ocius, Sree H. Kolli, Saadman S. Ahmad, Jules M. Dressler, Mahendra D. Chordia, Brandon L. Jutras, Melanie R. Rutkowski, Marcos M. Pires
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Long-Acting Poly(ADP-ribose) Polymerase Inhibitor Prodrug for Humans Bioconjugate Chem. (IF 4.7) Pub Date : 2024-04-09 Christopher W. Carreras, Shaun D. Fontaine, Ralph R. Reid, Gary W. Ashley, Daniel V. Santi
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In Vivo Toxicology of Metabolizable Atomically Precise Au25 Clusters at Ultrahigh Doses Bioconjugate Chem. (IF 4.7) Pub Date : 2024-04-01 Miaoyu Wang, Fangzhen Tian, Qi Xin, Huizhen Ma, Ling Liu, Shuyu Yang, Si Sun, Nan Song, KeXin Tan, Zhenhua Li, Lijie Zhang, Qi Wang, Liefeng Feng, Hao Wang, Zhidong Wang, Xiao-Dong Zhang
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A Genetically Encoded Photocaged Cysteine for Facile Site-Specific Introduction of Conjugation-Ready Thiol Residues in Antibodies Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-28 Arianna O. Osgood, Soumya Jyoti Singha Roy, David Koo, Renpeng Gu, Abhishek Chatterjee
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Drug–Polymer Nanodroplet Formation and Morphology Drive Solubility Enhancement of GDC-0810 Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-28 Kaylee E. Barr, Monica L. Ohnsorg, Lucy Liberman, Louis G. Corcoran, Apoorva Sarode, Karthik Nagapudi, Christina R. Feder, Frank S. Bates, Theresa M. Reineke
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Correction to “Modular Click Assembly DNA-Encoded Glycoconjugate Libraries with on-DNA Functional Group Transformations” Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-25 Xing Ling, Sixiu Liu, Yixuan Yang, Qian Dong, Lisa A. Marcaurelle, Wei Huang, Yun Ding, Xuan Wang, Xiaojie Lu
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Hyper-Responsive Chemiluminescent Probe Reveals Distinct PYRase Activity in Pseudomonas aeruginosa Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-22 Rozan Tannous, Omri Shelef, Tal Kopp, Micha Fridman, Doron Shabat
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Metal-Free Click-Chemistry: A Powerful Tool for Fabricating Hydrogels for Biomedical Applications Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-22 Aysun Degirmenci, Rana Sanyal, Amitav Sanyal
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Bioreducible Amphiphilic Hyperbranched Polymer-Drug Conjugate for Intracellular Drug Delivery Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-21 Sukanya Bera, Raju Bej, Pintu Kanjilal, Satyaki Sinha, Suhrit Ghosh
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Acidity-Triggered “Sticky Spotlight”: CCK2R-Targeted TME-Sensitive NIR Fluorescent Probes for Tumor Imaging In Vivo Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-21 Ruiqi Sun, Yuxin Wang, Wenhui Shi, Hongfu Zhang, Jianhua Liu, Weina He
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Site-Specific Conjugation of Native Antibody: Transglutaminase-Mediated Modification of a Conserved Glutamine While Maintaining the Primary Sequence and Core Fc Glycan via Trimming with an Endoglycosidase Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-18 Amissi Sadiki, Shanshan Liu, Shefali R. Vaidya, Eric M. Kercher, Ryan T. Lang, James McIsaac, Bryan Q. Spring, Jared R. Auclair, Zhaohui Sunny Zhou
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Targeting Strategies for Site-Specific mRNA Delivery Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-16 Jiaxing Di, Pei Huang, Xiaoyuan Chen
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Bioorthogonal Radiolabeling of Azide-Modified Bacteria Using [18F]FB-sulfo-DBCO Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-14 Aryn A. Alanizi, Alexandre M. Sorlin, Matthew F. L. Parker, Marina López-Álvarez, Hecong Qin, Sang Hee Lee, Joseph Blecha, Oren S. Rosenberg, Joanne Engel, Michael A. Ohliger, Robert R. Flavell, David M. Wilson
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Passivating the Background of Living Microbes with a Zwitterionic Peptide for Therapies Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-08 Liang Fang, Simian Cai, Patrick McMullen, Yi-Chen Hsu, Michelle Yi Qin Chen, Shaoyi Jiang
Living microbial therapies have been proposed as a course of action for a variety of diseases. However, problematic interactions between the host immune system and the microbial organism present significant clinical concerns. Previously, we developed a genetically encoded superhydrophilic zwitterionic peptide, termed EKP, to mimic low-immunogenic zwitterionic materials, which have been used for the
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Development of an Engineered Single-Domain Antibody for Targeting MET in Non-Small Cell Lung Cancer Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-12 Natalie Y. Luo, Rachel L. Minne, Joseph P. Gallant, Gihan S. Gunaratne, Jayden L. West, Saahil Javeri, Austin J. Robertson, Eric W. Lake, Jonathan W. Engle, Jason C. Mixdorf, Eduardo Aluicio-Sarduy, Kwang P. Nickel, Reinier Hernandez, Randall J. Kimple, Andrew M. Baschnagel, Aaron M. LeBeau
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3-Acyl-4-Pyranone as a Lysine Residue-Selective Bioconjugation Reagent for Peptide and Protein Modification Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-07 Keyi Nong, Yi-Lu Zhao, Shandong Yi, Xuchun Zhang, Siyuan Wei, Zhu-Jun Yao
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Transthyretin-Penetratin: A Potent Fusion Protein Inhibitor against Alzheimer’s Amyloid-β Fibrillogenesis with High Blood Brain Barrier Crossing Capability Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-07 Ying Wang, Wei Liu, Yan Sun, Xiaoyan Dong
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Assessment of the Efficacy of the Combination of RNAi of lncRNA DANCR with Chemotherapy to Treat Triple Negative Breast Cancer Using Magnetic Resonance Molecular Imaging Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-06 Calin Nicolescu, Jiyoon Kim, Da Sun, Zheng-Rong Lu
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GalNAc- or Mannose-PEG-Functionalized Polyplexes Enable Effective Lectin-Mediated DNA Delivery Bioconjugate Chem. (IF 4.7) Pub Date : 2024-03-05 Ricarda C. Steffens, Paul Folda, Nikole L. Fendler, Miriam Höhn, Katharina Bücher-Schossau, Susanne Kempter, Nicole L. Snyder, Laura Hartmann, Ernst Wagner, Simone Berger
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Engineering the Propeptide of Microbial Transglutaminase Zymogen: Enabling Substrate-Dependent Activation for Bioconjugation Applications Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-29 Ryutaro Ariyoshi, Takashi Matsuzaki, Ryo Sato, Kosuke Minamihata, Kounosuke Hayashi, Taisei Koga, Kensei Orita, Riko Nishioka, Rie Wakabayashi, Masahiro Goto, Noriho Kamiya
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Amyloid β-Peptide Segment Conjugated Side-Chain Proline-Based Polymers as Potent Inhibitors in Lysozyme Amyloidosis Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-29 Kasturee Nayak, Pooja Ghosh, Soumen Barman, Babu Sudhamalla, Patrick Theato, Priyadarsi De
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Recent Progress in Site-Selective Modification of Peptides and Proteins Using Macrocycles Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-28 Ye-Cheng Wang, Si-Cong Bai, Wei-Lin Ye, Jing Jiang, Gao Li
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Radiolabeling Diaminosarcophagine with Cyclotron-Produced Cobalt-55 and [55Co]Co-NT-Sarcage as a Proof of Concept in a Murine Xenograft Model Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-27 Wilson Lin, German Oscar Fonseca Cabrera, Eduardo Aluicio-Sarduy, Todd E. Barnhart, Jason C. Mixdorf, Zibo Li, Zhanhong Wu, Jonathan W. Engle
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Interactions and Transport of a Bioconjugated Peptide Targeting the Mitomembrane Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-25 Son V. Nguyen, Lev Levintov, Roy P. Planalp, Harish Vashisth
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Synthetic and Computational Design Insights toward Mimicking Protein Binding of Phosphate Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-20 Whitney C. Fowler, Chuting Deng, O. Therese Teodoro, Juan J. de Pablo, Matthew V. Tirrell
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A Kinetically Controlled Bioconjugation Method for the Synthesis of Radioimmunoconjugates and the Development of a Domain Mapping MS-Workflow for Its Characterization Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-17 Marco A. Pometti, Giuseppe Di Natale, Giancarlo Geremia, Nileshgiri Gauswami, Gianni Garufi, Giuseppina Ricciardi, Marcella Sciortino, Fabrizio Scopelliti, Giorgio Russo, Massimo Ippolito
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pH-Responsive Amphiphilic Triblock Fluoropolymers as Assemble Oxygen Nanoshuttles for Enhancing PDT against Hypoxic Tumor Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-17 Jun-an Zhang, David Haddleton, Paul Wilson, Lin-hua Zhu, Chun-yan Dai, Lin-lu Zhao
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Cathepsin B Processing Is Required for the In Vivo Efficacy of Albumin–Drug Conjugates Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-12 Barbara Bernardim, João Conde, Tuuli Hakala, Julie B. Becher, Mary Canzano, Aldrin V. Vasco, Tuomas P. J. Knowles, Jason Cameron, Gonçalo J. L. Bernardes
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Bioorthogonal Labeling Enables In Situ Fluorescence Imaging of Expressed Gas Vesicle Nanostructures Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-12 Erik Schrunk, Przemysław Dutka, Robert C. Hurt, Di Wu, Mikhail G. Shapiro
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A Cysteine-Maleimide-Based Design for Hemostatic, Antibacterial, and Biodegradable Wound Dressing Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-11 Pei Zhu, Tianjie You, Ying Wang, Mingxue Ma, Sheng Ye, Si Liu
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Peptide-Conjugated MRI Probe Targeted to Netrin-1, a Novel Metastatic Breast Cancer Biomarker Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-10 Clémentine Moreau, Tea Lukačević, Agnès Pallier, Julien Sobilo, Samia Aci-Sèche, Norbert Garnier, Sandra Même, Éva Tóth, Sara Lacerda
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Micropreparative Gel Electrophoresis for Purification of Nanoscale Bioconjugates Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-06 Sayyed Hashem Sajjadi, Shang-Jung Wu, Yahya Rabbani, Vitalijs Zubkovs, Hossein Ahmadzadeh, Elaheh K. Goharshadi, Ardemis A. Boghossian
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A Spontaneous Assembling Lipopeptide Nanoconjugate Transporting the Anthracycline Drug N-Benzyladriamycin-14-valerate for Personalized Therapy of Ewing Sarcoma Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-06 Nirupama Sabnis, Sangram Raut, Bhavani Nagarajan, Ammar Kapic, Akpedje Serena Dossou, Leonard Lothstein, Rafal Fudala, Bruce A. Bunnell, Andras G. Lacko
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[18F]pFBC, a Covalent CLIP-Tag Radiotracer for Detection of Viral Reporter Gene Transfer in the Murine Brain Bioconjugate Chem. (IF 4.7) Pub Date : 2024-02-03 Gregory D. Bowden, Sophie Stotz, Gina Dunkel, Sabrina Haas, Elena Kimmerle, Martin Schaller, Bettina Weigelin, Kristina Herfert, Bernd J. Pichler, Andreas Maurer
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Hydrophobicity Tuning of Cationic Polyaspartamide Derivatives for Enhanced Antisense Oligonucleotide Delivery Bioconjugate Chem. (IF 4.7) Pub Date : 2024-01-30 Jongmin Yum, Fadlina Aulia, Keisuke Kamiya, Mao Hori, Nan Qiao, Beob Soo Kim, Mitsuru Naito, Satomi Ogura, Tetsuya Nagata, Takanori Yokota, Satoshi Uchida, Satoshi Obika, Hyun Jin Kim, Kanjiro Miyata
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Asymmetry of Dual-Display DNA-Encoded Chemical Libraries Bioconjugate Chem. (IF 4.7) Pub Date : 2024-01-24 Louise Plais, Louis Trachsel, Jörg Scheuermann
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Design, Synthesis, and In Vitro and In Vivo Evaluation of Cereblon Binding Bruton’s Tyrosine Kinase (BTK) Degrader CD79b Targeted Antibody–Drug Conjugates Bioconjugate Chem. (IF 4.7) Pub Date : 2024-01-24 Alan Zhang, Katherine Seiss, Laurent Laborde, Sebastian Palacio-Ramirez, Daniel Guthy, Mylene Lanter, Julien Lorber, Anna Vulpetti, Luca Arista, Thomas Zoller, Thomas Radimerski, Claudio Thoma, Christina Hebach, William R. Tschantz, Alexei Karpov, Gregory J. Hollingworth, Joseph A. D’Alessio, Stephane Ferretti, Matthew T. Burger
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N-tert-Butoxycarbonyl-N-(2-(tritylthio)ethoxy)glycine as a Building Block for Peptide Ubiquitination Bioconjugate Chem. (IF 4.7) Pub Date : 2024-01-18 Lingling Peng, Elizabeth Helgason, Rafael Miranda, Jeffrey Tom, Jennifer Zhang, Erin C. Dueber, Aimin Song
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An Albumin-Holliday Junction Biomolecular Modular Design for Programmable Multifunctionality and Prolonged Circulation Bioconjugate Chem. (IF 4.7) Pub Date : 2024-01-17 Anders Dinesen, Veronica L. Andersen, Marwa Elkhashab, Diego Pilati, Pernille Bech, Elisabeth Fuchs, Torbjørn R. Samuelsen, Alexander Winther, Yunpeng Cai, Anders Märcher, Archie Wall, Marjan Omer, Jesper S. Nielsen, Vijay Chudasama, James R. Baker, Kurt V. Gothelf, Jesper Wengel, Jørgen Kjems, Kenneth A. Howard
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Rational Approach to Improve Detergent Efficacy for Membrane Protein Stabilization Bioconjugate Chem. (IF 4.7) Pub Date : 2024-01-12 Soyoung Yoon, Hyoung Eun Bae, Parameswaran Hariharan, Andreas Nygaard, Baoliang Lan, Menebere Woubshete, Aiman Sadaf, Xiangyu Liu, Claus J. Loland, Bernadette Byrne, Lan Guan, Pil Seok Chae
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Palladium-Mediated S-Arylation of Cysteine Residues with 4-[18F]Fluoroiodobenzene ([18F]FIB) Bioconjugate Chem. (IF 4.7) Pub Date : 2024-01-12 Felix Francis, Melinda Wuest, Jenilee D. Woodfield, Frank Wuest
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Exploring the Sensitivity of Antibody–Drug Conjugate Efficacy to the Selection of Payload, Antibody, and Cell line Bioconjugate Chem. (IF 4.7) Pub Date : 2024-01-03 Mara Rao, Shruthi Murali, Danielle Amores, Feifan Yu, Andrew Tsourkas
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Contiguous Silver(I)-Mediated Base Pairs of Imidazophenanthroline and Canonical Nucleobases in DNA Duplexes: Formation of Classical Duplexes versus Homodimer Formation Bioconjugate Chem. (IF 4.7) Pub Date : 2023-12-29 Nils Lefringhausen, Catharina Erbacher, Matthias Elinkmann, Uwe Karst, Jens Müller
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Aqueous Activation of RNA 2′-OH for Conjugation with Amines and Thiols Bioconjugate Chem. (IF 4.7) Pub Date : 2023-12-27 Ryuta Shioi, Lu Xiao, Eric T. Kool
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DNA Nanostructures as Catalysts: Double Crossover Tile-Assisted 5′ to 5′ and 3′ to 3′ Chemical Ligation of Oligonucleotides Bioconjugate Chem. (IF 4.7) Pub Date : 2023-12-22 Andrea C. Bardales, Joseph R. Mills, Dmitry M. Kolpashchikov
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Dual-Function Antibody Conjugate-Enabled Photoimmunotherapy Complements Fluorescence and Photoacoustic Imaging of Head and Neck Cancer Spheroids Bioconjugate Chem. (IF 4.7) Pub Date : 2023-12-21 Mohammad A. Saad, Stacey Grimaldo-Garcia, Allison Sweeney, Srivalleesha Mallidi, Tayyaba Hasan
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Cleavage and Noncleavage Chemistry in Reactive Oxygen Species (ROS)-Responsive Materials for Smart Drug Delivery Bioconjugate Chem. (IF 4.7) Pub Date : 2023-12-20 Teng Chi, Ting Sang, Yanjing Wang, Zhou Ye
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Enhancing Protective Antibodies against Opioids through Antigen Display on Virus-like Particles Bioconjugate Chem. (IF 4.7) Pub Date : 2023-12-19 Fatemeh Shafieichaharberoud, Shuyao Lang, Connor Whalen, Cristina Rivera Quiles, Lillie Purcell, Cameron Talbot, Pengfei Wang, Elizabeth B. Norton, Michelle Mazei-Robison, Agnieszka Sulima, Arthur E. Jacobson, Kenner C. Rice, Gary R. Matyas, Xuefei Huang
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Design Parameters for a Mass Cytometry Detectable HaloTag Ligand Bioconjugate Chem. (IF 4.7) Pub Date : 2023-12-19 Nicole Potter, Simon Latour, Edmond C. N. Wong, Mitchell A. Winnik, Hartland W. Jackson, Alison P. McGuigan, Mark Nitz