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Microwave-assisted one-pot quick synthesis of 1-monosubstituted 1,2,3-triazoles from arylboronic acids, sodium azide and 3-butyn-2-ols
Journal of Chemical Sciences ( IF 1.7 ) Pub Date : 2020-11-11 , DOI: 10.1007/s12039-020-01856-4
ZHONGLIN DU , FENRUI LI , LI LI , RAN LI

Abstract

Microwave-assisted one-pot quick synthesis to 1-monosubstituted 1,2,3-triazoles was achieved with good to excellent yields using the widely available arylboronic acids, sodium azide and 3-butyn-2-ols within 15 min. This method features high efficient and facile as organic azides, acetylene gas and harsh conditions were avoided.

Graphic abstract

Microwave-assisted one-pot quick synthesis to 1-monosubstituted 1,2,3-triazoles was achieved with good to excellent yields using the widely available arylboronic acids, sodium azide and 3-butyn-2-ols within 15 min.



中文翻译:

微波辅助一锅快速从芳基硼酸,叠氮化钠和3-丁炔-2-醇合成1-单取代的1,2,3-三唑

摘要

使用广泛使用的芳基硼酸,叠氮化钠和3-butyn-2-ols,在15分钟内即可实现微波辅助一锅快速合成1-单取代的1,2,3-三唑,收率良好至优异。由于避免了有机叠氮化物,乙炔气和苛刻的条件,该方法具有高效简便的特点。

图形摘要

使用广泛使用的芳基硼酸,叠氮化钠和3-butyn-2-ols,在15分钟内即可实现微波辅助一锅快速合成1-单取代的1,2,3-三唑,收率良好至优异。

更新日期:2020-11-12
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