Abstract

Microwave-assisted one-pot quick synthesis to 1-monosubstituted 1,2,3-triazoles was achieved with good to excellent yields using the widely available arylboronic acids, sodium azide and 3-butyn-2-ols within 15 min. This method features high efficient and facile as organic azides, acetylene gas and harsh conditions were avoided.

Graphic abstract

Microwave-assisted one-pot quick synthesis to 1-monosubstituted 1,2,3-triazoles was achieved with good to excellent yields using the widely available arylboronic acids, sodium azide and 3-butyn-2-ols within 15 min.

中文翻译：

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微波辅助一锅快速从芳基硼酸，叠氮化钠和3-丁炔-2-醇合成1-单取代的1,2,3-三唑

摘要

使用广泛使用的芳基硼酸，叠氮化钠和3-butyn-2-ols，在15分钟内即可实现微波辅助一锅快速合成1-单取代的1,2,3-三唑，收率良好至优异。由于避免了有机叠氮化物，乙炔气和苛刻的条件，该方法具有高效简便的特点。

图形摘要

使用广泛使用的芳基硼酸，叠氮化钠和3-butyn-2-ols，在15分钟内即可实现微波辅助一锅快速合成1-单取代的1,2,3-三唑，收率良好至优异。