A highly selective synthesis of saturated aza-heterocycles from vicinal functionally substituted electron-deficient enoates and binucleophiles under classical and hyperbaric conditions is described. The assembly of the heterocyclic core proceeds through conjugate nucleophilic addition/cyclocondensation sequence.

中文翻译：

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β-官能取代的烯酸酯对饱和氮杂杂环的选择性组装

描述了在经典和高压条件下，由邻位功能取代的缺电子烯酸酯和双亲核试剂高度选择性合成饱和氮杂杂环的方法。杂环核的组装通过共轭亲核加成/环缩合序列进行。