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Rh(III)-Catalyzed N-Arylation of Alkyl Dioxazolones with Arylboronic Acids for the Synthesis of N-Aryl Amides
European Journal of Organic Chemistry ( IF 2.5 ) Pub Date : 2022-07-28 , DOI: 10.1002/ejoc.202200710 Jia-Lin Song 1 , Shao-Yong Chen 2 , Lin Xiao 2 , Xiao-Ling Xie 1 , Yi-Chuan Zheng 2 , Zhang Shang-Shi 3 , Bing Shu 1
European Journal of Organic Chemistry ( IF 2.5 ) Pub Date : 2022-07-28 , DOI: 10.1002/ejoc.202200710 Jia-Lin Song 1 , Shao-Yong Chen 2 , Lin Xiao 2 , Xiao-Ling Xie 1 , Yi-Chuan Zheng 2 , Zhang Shang-Shi 3 , Bing Shu 1
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SAn original and practical method for N-aryl amides preparation has been established through Rh(III)-catalyzed C(sp2)−N cross-coupling reactions of alkyl dioxazolones with arylboronic acids, heterocyclic boronic acid, and alkenyl boronic acid, featured with a broad substrate scope, good functional group compatibility, high yields, and suitability for late-stage modification of drug molecular structures.
中文翻译：
Rh(III)-催化烷基二恶唑酮与芳基硼酸的 N-芳基化合成 N-芳基酰胺
通过Rh(III)催化烷基二恶唑酮与芳基硼酸、杂环硼酸和烯基硼酸的C(sp 2 )-N交叉偶联反应，建立了一种独创且实用的制备N-芳基酰胺的方法。底物范围广，官能团相容性好，收率高，适合药物分子结构的后期修饰。
更新日期：2022-07-28
中文翻译：
Rh(III)-催化烷基二恶唑酮与芳基硼酸的 N-芳基化合成 N-芳基酰胺
通过Rh(III)催化烷基二恶唑酮与芳基硼酸、杂环硼酸和烯基硼酸的C(sp 2 )-N交叉偶联反应，建立了一种独创且实用的制备N-芳基酰胺的方法。底物范围广，官能团相容性好，收率高，适合药物分子结构的后期修饰。
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