Seventeen novel N-phenylbenzamide derivatives bearing a trifluoromethylpyrimidine moiety were synthesized via four-step reactions. Their antifungal and insecticidal properties were evaluated. Antifungal test results demonstrated that some of the synthesized compounds showed better in vitro bioactivities against Phomopsis sp., Botryosphaeria dothidea (B. dothidea), and Botrytis cinerea (B. cinerea) at 50 μg/mL than pyrimethanil. Unfortunately, the synthesized compounds revealed lower insecticidal activities against Spodoptera frugiperda (S. frugiperda) and Mythimna separata (M. separata) at 500 μg/mL than chlorantraniliprole.

中文翻译：

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含三氟甲基嘧啶部分的新型 N-苯基苯甲酰胺衍生物的合成及抗真菌和杀虫活性

通过四步反应合成了十七种带有三氟甲基嘧啶部分的新型N-苯基苯甲酰胺衍生物。评价了它们的抗真菌和杀虫特性。抗真菌试验结果表明，部分合成化合物在 50 μg /mL 浓度下对拟杆菌属、Botryosphaeria dothidea ( B. dothidea ) 和Botrytis cinerea ( B. cinerea ) 显示出 比嘧霉胺更好的体外生物活性。不幸的是，合成的化合物对草地贪夜蛾（S. frugiperda）和Mythimna separata 的杀虫活性较低（M. separata )比氯虫苯甲酰胺浓度为 500  μ g/mL。