Abstract

Tandem reactions between β-iodoazides and propargyl alcohols under mild conditions are presented, providing a general and convenient method for the synthesis of 6,7-dihydro-4H-[1,2,3]triazolo[5,1-c][1,4]oxazines. The advantages of this method are its simple operation, high efficiency and high product yields (80–95%).

中文翻译：

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通过β-碘叠氮化物与炔丙醇的串联反应合成6,7-二氢-4H-[1,2,3]三唑并[5,1-c][1,4]恶嗪

摘要

介绍了β-碘叠氮化物和炔丙醇在温和条件下的串联反应，为合成6,7-二氢-4 H- [1,2,3]三唑并[5,1- c ][提供了一种通用方便的方法。1,4]恶嗪。该方法的优点是操作简单、效率高、产品收率高（80-95%）。