当前位置: X-MOL 学术Tetrahedron › 论文详情
Our official English website, www.x-mol.net, welcomes your feedback! (Note: you will need to create a separate account there.)
Selective transformations of 2-(p-toluenesulfonyl)-N-tosylhydrazones to substituted 1,2,3-thiadiazoles
Tetrahedron ( IF 2.1 ) Pub Date : 2020-11-26 , DOI: 10.1016/j.tet.2020.131803
Yijiao Feng , Jing He , Weiwei Li , Zhen Yang , Yueting Wei , Ping Liu , Jixing Zhao , Chengzhi Gu , Wenli Wang

Selective transformations of 2-(p-toluenesulfonyl)-N-tosylhydrazones with different sulfur sources have been established. A series of 4-aryl-1,2,3-thiadiazoles and novel 4-aryl-5-tosyl-1,2,3-thiadiazoles were selectively constructed by the adjustment of reaction conditions. These protocols feature short reaction time, good compatibility of functional group, easily available materials, and good selectivity.



中文翻译:

2-(甲苯磺酰基)-N-甲苯磺酰hydr选择性转化为取代的1,2,3-噻二唑

已经建立了具有不同硫源的2-(甲苯磺酰基)-N-甲苯磺酰hydr的选择性转化。通过调节反应条件,选择性地构建了一系列的4-芳基-1,2,3-噻二唑和新型的4-芳基-5-甲苯基-1,2,3-噻二唑。这些协议的特点是反应时间短,官能团的相容性好,易于获得的材料和选择性好。

更新日期:2020-12-17
down
wechat
bug