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Iodine-Mediated Facile One-Pot Access to N-Aryl-2-benzoxazolamines
SynOpen ( IF 2.0 ) Pub Date : 2020-11-24 , DOI: 10.1055/s-0040-1705982 Shinji Tanimori , Haruna Nariki , Takuya Miyamura , Daiki Matsui , Motohiro Sonoda
中文翻译:
碘介导的一锅法获得N-芳基-2-苯并恶唑胺
更新日期:2020-11-25
SynOpen ( IF 2.0 ) Pub Date : 2020-11-24 , DOI: 10.1055/s-0040-1705982 Shinji Tanimori , Haruna Nariki , Takuya Miyamura , Daiki Matsui , Motohiro Sonoda
Facile, iodine-mediated access to N-aryl-2-benzoxazolamines has been achieved in a one-pot manner under mild reaction conditions. Reaction of 2-aminophenols and aryl isothiocyanates afforded N-aryl-2-benzoxazolamines in the presence of molecular iodine and pyridine in tetrahydrofuran at room temperature in moderate to excellent yields.
中文翻译:
碘介导的一锅法获得N-芳基-2-苯并恶唑胺
在温和的反应条件下,以单锅方式实现了碘介导的N-芳基-2-苯并恶唑胺的便捷连接。在室温下,在四氢呋喃中,在存在分子碘和吡啶的条件下,在氨基碘和吡啶存在下,N-芳基-2-苯并恶唑胺与2-氨基酚和芳基异硫氰酸酯反应,得到中等至极好的收率。