Graphene Derivatives (GDs) have captured the interest and imagination of pharmaceutical scientists. This review exclusively provides pharmacokinetics and pharmacodynamics information with a particular focus on biopharmaceuticals. GDs can be used as multipurpose pharmaceutical delivery systems due to their ultra-high surface area, flexibility, and fast mobility of charge carriers. Improved effects, targeted delivery to tissues, controlled release profiles, visualization of biodistribution and clearance, and overcoming drug resistance are examples of the benefits of GDs. This review focuses on the application of GDs for the delivery of biopharmaceuticals. Also, the pharmacokinetic properties and the advantage of using GDs in pharmaceutics will be reviewed to achieve a comprehensive understanding about the GDs in pharmaceutical sciences.

石墨烯衍生物（GDs）引起了药物科学家的兴趣和想象力。这篇综述专门提供了药代动力学和药效学信息，特别侧重于生物制药。GD由于具有超高的表面积，柔韧性和电荷载体的快速迁移性，因此可以用作多用途药物输送系统。改进的效果，对组织的靶向递送，控释曲线，生物分布和清除的可视化以及克服药物抗性是GD益处的示例。这篇综述着重于GDs在生物制药中的应用。此外，将审查药代动力学特性以及在药物学中使用GD的优势，以全面了解药物科学中的GD。