One target, more options. The toolbox of high‐affinity ligands for clinically relevant proteins is continuously expanding. Covalent conjugates of these ligands with drugs, radiotracers and other bioactive agents are being studied for therapy and imaging. The pharmacokinetic properties, chemical accessibility and versatility are just a few examples of the positive features that could bring targeted small molecule conjugates to a leading role in future medicine.

中文翻译：

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有针对性的小分子共轭物：未来就在眼前。

一个目标，更多选择。用于临床相关蛋白的高亲和力配体的工具箱正在不断扩大。这些配体与药物，放射性示踪剂和其​​他生物活性剂的共价缀合物正在研究中，以用于治疗和成像。药代动力学特性，化学可及性和多功能性只是积极特征的几个例子，这些积极特征可以使靶向的小分子结合物在未来的医学中发挥主导作用。