Multigram Synthesis of Heterabicyclo[n.1.0]alkan‐1‐yl Trifluoroborates,European Journal of Organic Chemistry

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Multigram Synthesis of Heterabicyclo[n.1.0]alkan‐1‐yl Trifluoroborates
European Journal of Organic Chemistry ( IF 2.5 ) Pub Date : 2020-08-17 , DOI: 10.1002/ejoc.202000977
Ihor Kleban _{1,

2} , Yevhen Krokhmaliuk _{1,

3} , Sofiia Reut _{1,

3} , Serhii Shuvakin _{1,

3} , Vyacheslav V. Pendyukh ₁ , Oleksandr I. Khyzhan ₁ , Dmytro S. Yarmoliuk ₁ , Andriy V. Tymtsunik _{1,

4} , Yuliya V. Rassukana _{2,

4} , Oleksandr O. Grygorenko _{1,

3}

Affiliation

Multigram synthesis of oxa‐ and azabicyclo[n.1.0]alkan‐1‐yl trifluoroborates relying on efficient 4–5‐step reaction sequences is described. The title compounds was obtained in up to 50 g scale in a single run (10–41 % overall yield).