3‐Carboxy‐/3‐Aminobicyclo[1.1.1]pentane‐Derived Sulfonamides and Sulfonyl Fluorides – Advanced Bifunctional Reagents for Organic Synthesis and Drug Discovery,European Journal of Organic Chemistry

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3‐Carboxy‐/3‐Aminobicyclo[1.1.1]pentane‐Derived Sulfonamides and Sulfonyl Fluorides – Advanced Bifunctional Reagents for Organic Synthesis and Drug Discovery
European Journal of Organic Chemistry ( IF 2.5 ) Pub Date : 2020-04-17 , DOI: 10.1002/ejoc.202000303
Serhii O. Kokhan _{1,

2} , Yevheniia B. Valter ₂ , Andriy V. Tymtsunik _{2,

3} , Igor V. Komarov _{1,

2} , Oleksandr O. Grygorenko _{1,

2}

Affiliation

Synthesis of bifunctional bicyclo[1.1.1]pentane‐derived sulfonyl fluorides, sulfonamides, and sulfinates from the corresponding carboxylic acids is described, including an isosteric analogue of a classical sulfonamide antibiotic.