A metal-free iodine/TBHP-mediated oxidative CN bond formation for the one-pot synthesis of N-fused 1,2,4-triazoles and related heterocycles via cyclization has been developed. This reaction which is amenable to scale-up affords the corresponding products with good to excellent yields and tolerates a wide range of functional groups.

中文翻译：

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通过I ₂ / TBHP介导的氧化性C N键形成一锅合成N稠合的1,2,4-三唑和相关杂环

已经开发了无金属的碘/ TBHP介导的氧化C N键形成，用于通过环化一锅合成N稠合的1,2,4-三唑和相关杂环。该适合扩大规模的反应提供了具有良好至优异收率的相应产物，并容许宽范围的官能团。