当前位置: X-MOL 学术Synlett › 论文详情
Our official English website, www.x-mol.net, welcomes your feedback! (Note: you will need to create a separate account there.)
The First Example of Azole-Fused Cyclic Anhydride Reacting in the Castagnoli–Cushman Way
Synlett ( IF 1.7 ) Pub Date : 2018-02-27 , DOI: 10.1055/s-0036-1591908
Mikhail Krasavin 1 , Ella Moreau 1 , Dmitry Dar’in 1
Affiliation  

Pyrazole-fused cyclic anhydrides have been employed for the first time as the Castagnoli–Cushman reaction partners to produce hitherto unknown 4-oxo-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-7-carboxylates in remarkably convenient and speedy fashion. Attempts to realize the same chemistry with indole and benzimidazole analogues failed.

中文翻译:

唑稠环酸酐以 Castagnoli-Cushman 方式反应的第一个例子

吡唑稠合环酐首次被用作 Castagnoli-Cushman 反应伙伴,以显着地制备迄今为止未知的 4-oxo-4,5,6,7-四氢吡唑并[1,5-a]pyrazine-7-carboxylates方便快捷的时尚。用吲哚和苯并咪唑类似物实现相同化学反应的尝试失败了。
更新日期:2018-02-27
down
wechat
bug