Photochemical Synthesis of 2-Azabicyclo[3.2.0]heptanes: Advanced Building Blocks for Drug Discovery. Synthesis of 2,3-Ethanoproline,The Journal of Organic Chemistry

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Photochemical Synthesis of 2-Azabicyclo[3.2.0]heptanes: Advanced Building Blocks for Drug Discovery. Synthesis of 2,3-Ethanoproline
The Journal of Organic Chemistry ( IF 3.3 ) Pub Date : 2018-01-16 00:00:00 , DOI: 10.1021/acs.joc.7b02910
Tetiana Druzhenko _{1,

2} , Yevhen Skalenko _{1,

2} , Maryna Samoilenko ₁ , Aleksandr Denisenko ₁ , Sergey Zozulya ₁ , Petro O. Borysko ₁ , Maria I. Sokolenko ₁ , Alexandr Tarasov ₁ , Pavel K. Mykhailiuk _{1,

3}

Affiliation

Intramolecular photochemical [2 + 2]-cyclization of acetophenone enamides gave 2-azabicyclo[3.2.0]heptanes, advanced building blocks for drug discovery. Synthesis of a conformationally restricted analogue of proline, 2,3-ethanoproline, was performed.

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