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N‐Arylated Sulfoximines as Cross‐Coupling Building Blocks
Advanced Synthesis & Catalysis ( IF 4.4 ) Pub Date : 2018-01-16 , DOI: 10.1002/adsc.201701394
Anne-Katrin Bachon 1 , Anne-Dorothee Steinkamp 1 , Carsten Bolm 1
Affiliation  

The application of borylated N‐aryl sulfoximines as newly designed synthetic building blocks in Suzuki‐type cross coupling reactions offers rapid access to a wide range of N‐biaryl derivatives with potential relevance for medicinal chemistry and crop protection in good to excellent yields (up to 98%).

中文翻译:

N-芳基磺胺嘧啶作为交叉偶联的构建基块

在Suzuki型交叉偶联反应中应用硼化的N-芳基亚砜亚胺作为新设计的合成构件,可以快速获得广泛的N-联芳基衍生物,对药物化学和作物保护具有潜在的相关性,且产量高至优异(可达98%)。
更新日期:2018-01-16
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