Copper‐Mediated Tandem C(sp2)‐H Amination and Annulation of Arenes with 2‐Aminopyridines: Synthesis of Pyrido‐fused Quinazolinone Derivatives,Advanced Synthesis & Catalysis

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Copper‐Mediated Tandem C(sp2)‐H Amination and Annulation of Arenes with 2‐Aminopyridines: Synthesis of Pyrido‐fused Quinazolinone Derivatives
Advanced Synthesis & Catalysis ( IF 4.4 ) Pub Date : 2017-12-12 , DOI: 10.1002/adsc.201701286
Jidan Liu ₁ , Jinhui Zou ₁ , Jiawei Yao ₁ , Guoshu Chen ₁

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An efficient and convenient copper‐mediated tandem C(sp²)‐H amination and annulation of arenes with 2‐aminopyridines to provide 11H‐pyrido[2,1‐b]quinazolin‐11‐ones has been developed. A variety of benzamides and 2‐aminopyridines bearing different substituents are compatible with this transformation

中文翻译：

铜介导的串联C（sp2）-H氨基化和芳烃与2-氨基吡啶的环化反应：吡啶基稠合的喹唑啉酮衍生物的合成

开发了一种高效便捷的铜介导的串联C（sp ²）-H胺化和芳烃与2-氨基吡啶的环化反应，以提供11个H-吡啶并[ 2,1- b ]喹唑啉-11-酮的方法。各种带有不同取代基的苯甲酰胺和2-氨基吡啶与这种转化相容

更新日期：2017-12-12

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