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成果及论文

52. Xin Yin, Azhar Anwar, Linbo Yan, Ranran Yu, Yang Luo, Liang Shi, Botao Li, Jiehao Chen, Gaoli Liang, Yongci Chen, Jie Tang, Jie Liang,  Yansheng Kan, Zhihao Zhang, Xiahuan, Zhou, Jizheng Ma, Chenbo Ji, Yanbo Wang, Qipeng Zhang, Jing Li, Liang Li, Xiaozhi Zhao, Feng Yin,  Liyuan Sheng, Dijun Chen*, Tao Zhang*, Chen-Yu Zhang*, Xi Chen*. Paternal Exercise Confers Endurance Capacity to Offspring Through Sperm MicroRNAs. Cell Metab. 2025, 37, 2167-2184.

        


51. Rui Wu, Saijian Shi, Yuanjie Huang, Feng Tian, Jiqin Hou, Xiangqing Kong, Longxiang Sheng, Tao Zhang*, Lijun Tang*, Wei Sun*.18F-DOPA Uptake Illustration Acts as An Indicator for Renal Sympathetic Activity. Front Physiol202516, 1569699.

50. Ken Lin, Qi Sun, Pengcheng Tang, Saizhou Wang, Mengjie Jiao, Tao Zhang*,  Hongjian Lu*. Late-Stage N-Atom Deletion of Multisubstituted 2-Azabicyclo[2.1.1]Hexanes. ACS Catalysis. 2025, 15, 5825-5834.


49. Chenchen Xu, Zhihao Zhang, Lizhu Wang, Xin Ji, Yue Yue, Xurui Liang, Yufei Han, Jiqin Hou, Tao Zhang*. Exploring the New Model of Medical Innovation and Entrepreneurship Talent Training Based on Biodesign in Eastern China. BMC Med Educ. 202525, 388.


48. Jianlun HuXiaofeng WangQi SunShuyang YangMin Feng*, Tao Zhang*Hao Hong*. A Polysaccharide Metal Phenolic Network Nanocomposite for Theranostic Applications in Inflammatory Bowel Disease. Adv. Funct. Mater. 2025, 35, 2416918.

 


47. Jingjing Shen, Kai Feng, Jing Yu, Yaxuan Zhao, Ruifang Chen, Hehua Xiong, Yiling Ruan, Zhengtao Xu, Tao Zhang*, Xiaolian  Sun*. Responsive and Traceless Assembly of Iron Nanoparticles and 131I labeled Radiopharmaceuticals for Ferroptosis Enhanced Radio-immunotherapy. Biomaterials2025313, 122795. 


46. Chang Hong Wei, Shipeng Dong, Zhiheng Xu, Muzi Li, Tao Zhang, Zhibin Xu, Si Lan, Shuao Wang, Liang Mao*. Controllable Multi-Exciton Zero-Dimensional Antimony-Based Metal Halides for White-light Emission and β-Ray Detection. Angew. Chem. Int. Ed2024, 63, e202412253. 




45. 周夏欢,施赛健,顾莹莹,李天女,唐立钧,张涛*. 放射性药物研发的一般流程与关键点分析.中华核医学与分子影像杂志,202444, 440-444.


44. German O Fonseca Cabrera, Xinrui Ma, Wilson Lin, Tao Zhang, Weiling Zhao, Liqin Pan, Xiaomei Li, Todd E Barnhart, Eduardo Aluicio-Sarduy, Huaifu Deng, Xuedan Wu, Kadalipura P Rakesh, Zibo Li, Jonathan W Engle, Zhanhong Wu*. Synthesis of 64Cu-, 55Co-, and 68Ga-Labeled Radiopharmaceuticals Targeting Neurotensin Receptor-1 for Theranostics: Adjusting In Vivo Distribution Using Multiamine Macrocycles. J. Nucl. Med., 202465, 1250-1256. 


43. 张涛,施蒙,计欣,李天女,唐立钧,蒋建东*. 零期临床助力中国原创药研发新范式迭代.中国医药生物技术,2024, 19, 193-196.


42. Tao Zhang*, Xinrui Ma, Muyun Xu, Jinghua Cai, Jianhua Cai, Yanguang Cao, Zhihao Zhang, Xin Ji, Jian He, German Oscar Fonseca Cabrera, Xuedan Wu, Weiling Zhao, Zhanhong Wu, Jin Xie*, Zibo Li*. Chelator boosted tumor-retention and pharmacokinetic properties: development of 64Cu labeled radiopharmaceuticals targeting neurotensin receptor. Eur. J. Nucl. Med. Mol. Imaging202451, 3322-3333. 


41. Huihui Liu, Hehua Xiong, Changjun Li, Mengxia Xu, Yuyang Yun, Yiling Ruan, Lijun Tang, Tao Zhang*, Dan Su*, Xiaolian Sun*. 131I Induced In Vivo Proteolysis by Photoswitchable azoPROTAC Reinforces Internal Radiotherapy. Small., 2024, 20, e2310865. 


40. Xiaodan Jiao, Xiaoyang Li, Yan Du, Yiyang Cong, Shuyang Yang, Daiqin Chen, Tao Zhang*, Min Feng*, Hao Hong*. Positron Emission Tomography Guided Synergistic Treatment of Melanoma Using Multifunctional Zirconium-Hematoporphyrin Nanosonosensitizers. J. Control. Release., 2024, 370, 95-109. 


39. Xinmiao Zhang, Jingru Guo, Ziwei Zhou, Kai Feng, Huihui Liu, Yiling Ruan, Ruifang Chen, Zixuan Liu, Tao Zhang*, Lijun Tang*,  Xiaolian Sun*. Self-Illuminating In Situ Hydrogel with Immune-Adjuvant Amplify Cerenkov Radiation-Induced Photodynamic Therapy. Chem. Biomed. Imaging.,20232, 275-282.


38. Xin Ji, Xin Chen, Kexin Li, Zhihao Zhang, Lijun Tang, Tiannv Li, Feng Han, Hao Hong*,  Tao Zhang*. Molecular Eye: A System for Precise Diagnosis and Treatment of Major Clinical Diseases Based on Molecular Probe Technology. Chem. Biomed. Imaging.,2023,2, 168–184.


37. 李政,彭灿,李希臣,董国生,韩雨霏,张涛,唐立钧*.多靶点药物的研究策略及进展.中国新药杂志, 2024, 16, 1665-1675.


36. 彭灿,董国生,李希臣,李政,韩雨霏,张涛*. [18F]FDOPA放射标记合成工艺研究进展中国新药杂志202412, 1233-1242.


35. 李希臣,李政,彭灿,钱陈,韩雨霏,张涛*.MOFs在催化有机分子转化中的应用. 化学进展20243, 367-375.


34. 唐嘉逸,华娜,许晨晨,张涛*,韩雨霏*.靶向PARP-1 PET/CT成像在肿瘤精准诊疗中应用研究进展.中国药物化学杂志,2023, 12, 948-956.


33. Huihui Liu, Qing Wang, Jingru Guo, Kai Feng, Yiling Ruan, Zhihao Zhang, Xin Ji, Jigang Wang*, Tao Zhang*, Xiaolian Sun*. Prodrug-based Strategy with A Two-in-one Liposome for Cerenkov-induced Photodynamic Therapy and Chemotherapy. J. Control. Release., 2023, 364, 206-215.


32.Jingru Guo, Hehua Xiong, Huihui Liu, Tao Zhang*, Xiaolian Sun*. Radioiodine Based Biomedical Carriers for Cancer theranostics. Coordin Chem Rev., 2023497, 215430.


31.董国生, 陈欣, 李可欣, 张涛*. 放射性核素偶联药物的研究进展及临床应用.药学进展. 202347, 324-336.


30.张志豪, 朱晨亿, 丛容, 张涛*. 放射性金属核素及其核医学应用. 国际医学放射学杂志. 2023, 46, 333-339; 347.


29. Xunqing Dong, Mingzhou Shang, Shuguang Chen, Tao Zhang, Hitesh B Jalani, Hongjian Lu*. Carbonyl-Assisted Iridium-Catalyzed C-H Amination Using 2,2,2-Trichloroethoxycarbonyl Azide. J. Org. Chem., 202287, 13990-14004.

 


28. Anne M Talkington, Morgan D McSweeney, Timothy Wessler, Marielle K Rath, Zibo Li, Tao Zhang, Hong Yuan, Jonathan E Frank, M Gregory Forest, Yanguang Cao, Samuel K Lai*. A PBPK Model Recapitulates Early Kinetics of Anti-PEG Antibody-mediated Clearance of PEG-Liposomes. J. Control. Release.2022, 343, 518-527.


27. Tao Zhang, Jinghua Cai, Muyun Xu, Xinrui Ma, Hui Wang, Mengzhe Wang, Zhaoguo Han, Jason Wang, Eric Smith, Zibo Li*, Zhanhong Wu*. Development of 18F-Labeled Vinyl Sulfone-PSMAi Conjugates as New PET Agents for Prostate Cancer Imaging. Mol. Pharmaceutics, 2022, 19, 720-727. (T. Zhang,  J. Cai and M. Xu contributed equally)


26. Wei Chen, Hui Wang, Nicholas E. S. Tay, Vincent A. Pistritto, Kang-Po Li, Tao Zhang, Zhanhong Wu, David A. Nicewicz,* Zibo Li*. Arene Radiofluorination Enabled by Photoredox-mediated Halide Interconversion. Nat. Chem.2022, 14, 216-223.


25. Benjamin L Cline, Wen Jiang, Chaebin Lee, Zhengwei Cao, Xueyuan Yang, Shuyue Zhan, Harrison Chong, Tao Zhang, Zhaoguo Han, Xuedan Wu, Li Yao, Hui Wang, Weizhong Zhang,* Zibo Li,* Jin Xie*. Potassium Iodide Nanoparticles Enhance Radiotherapy against Breast Cancer by Exploiting the Sodium-Iodide Symporter. ACS Nano202115, 17401-17411.


24. Xiaofen Ma, Chaehin Lee, Tao Zhang, Jinghua Cai, Hui Wang, Fangchao Jiang, Zhanhong Wu, Jin Xie,* Guihua Jiang,* Zibo Li*. Image-guided Selection of Gd@C-dots as Sensitizers to Improve Radiotherapy of Non-small Cell lung Cancer. J. Nanobiotechnol., 2021, 19, 284. (X. Ma,  C. Lee and T. Zhang contributed equally)


23. Anne M Talkington, Morgan D McSweeney, Tao Zhang, Zibo Li, Andrew C Nyborg, Brian LaMoreaux, Eric W Livingston, Jonathan E Frank, Hong Yuan, Samuel K Lai.* High MW Polyethylene Glycol Prolongs Circulation of Pegloticase in Mice with Anti-PEG Antibodies. J. Control. Release., 2021, 338, 804-812.

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22. Xinyi Zhang, Li Wang, Wenhui Fu, Yue Feng, Chengrun Zeng, Liu Zhou, Tao Zhang, Tingting Xu, Jianpeng Cao, Zibo Li,*  Yue Chen*. 18F-PEG1-Vinyl Sulfone-Labeled Red Blood Cells as Positron Emission Tomography Agent to Image Intra-Abdominal Bleeding. Front. Med., 2021, 8, 646862.


21.Chuangqi Wang, He Zhang, Tao Zhang, Xiaoyu Zou, Hui Wang, Julia Rosenbenger, Raghu Vannam, Wliiliam S. Trout, Xinqiao Jia, * Zibo Li, * Joseph M. Fox *. Enabling In Vivo Photocatalytic Activation of Rapid Bioorthogonal Chemistry by Repurposing Silicon-Rhodamine Fluorophores as Cytocompatible Far-Red Photocatalysts. J. Am. Chem. Soc., 2021, 143, 10793-10803. (C. Wang and H. Zhang contributed equally)


20. Li Wang, Hui Wang, Kun Shen, Hyejin Park, Tao Zhang, Xuedan Wu, Mei Hu, Hong Yuan, Yue Chen, Zhanhong Wu,* Qiu Wang,* Zibo Li. Development of Novel 18F-PET Agents for Tumor Hypoxia Imaging. J. Med. Chem., 2021, 64, 5593-5602.



19. Tao Zhang, Jianhua Cai, Hui Wang, Mengzhe Wang, Zhanhong Wu, Xiaofen Ma,* Zibo Li*. RXH-Reactive 18F-Vinyl Sulfones as Versatile Agents for PET Probe Construction. Bioconjugate. Chem., 2020, 31, 2482-2487. (T. Zhang and J. Cai contributed equally)

 


18. Xunqing Dong, Panpan Ma, Tao Zhang, Hitesh Jalani, Guigen Li, Hongjian Lu*, Iridium-Catalyzed C-H Amination of Weinreb Amides: A Facile Pathway towards Anilines and Quinazolin-2,4-diones, J. Org. Chem., 2020, 85, 13096-13107. (X. Dong and P. Ma contributed equally)

 


17. Mengzhe Wang, Hui Wang, Crystal Q. Niu, Tao Zhang, Zhanhong Wu, Zibo Li*, Tetrazine-TCO Ligation: A Potential Simple Approach to Improve Tumor Uptake through Enhanced Blood Circulation, Bioconjugate. Chem., 2020, 31, 1795-1803.

 


16. Xiaofen Ma, Mengzhe Wang, Hui Wang, Tao Zhang, Zhanhong Wu, Mariia V. Sutton, Vladimir V. Popik, Guihua Jiang*, Zibo Li*, Development of Bispecific NT-PSMA Heterodimer for Prostate Cancer Imaging: A Potential Approach to Address Tumor Heterogeneity, Bioconjugate. Chem., 2019, 30, 1314-1322.

 


15. Tao Zhang, Xunqing Dong, Hitesh B Jalani, Jiaqi Zou, Guigen Li, Hongjian Lu*, Iridium-Catalyzed C-H Amination/Cyclization for Medium to Large N‑Heterocycle-Fused Dihydroquinazolinones, Org. Lett., 2019, 21, 3706-3710. (T. Zhang and X. Dong contributed equally)

 


14. Tao Zhang, Xuejiao Hu, Xunqing Dong, Guigen Li, Hongjian Lu*, Iridium-Catalyzed Unreactive C(sp3)-H Amination with 2,2,2-Trichloroethoxycarbonyl Azide, Org. Lett., 2018, 20, 6260-6264.

 


13. Meng Yu, Tao Zhang, Hitesh B Jalani, Xunqing Dong, Hongjian Lu*, Guigen Li, Iridium-Catalyzed Aryl C-H Sulfonamidation and Amide Formation Using a Bifunctional Nitrogen Source, Org. Lett., 2018, 20, 4828-4832. (M. Yu and T. Zhang contributed equally)

 


12. Tao Zhang, Zhen Wang, Xuejiao Hu, Meng Yu, Tianning Deng, Guigen Li, Hongjian Lu*, Cesium Carboxylate-Promoted Iridium Catalyzed C-H Amidation/Cyclization with 2,2,2-Trichloroethoxycarbonyl Azide, J. Org. Chem., 2016, 81, 4898-4905.

 


11. Tao Zhang, Xuejiao Hu, Zhen Wang, Tiantian Yang, Hao Sun, Guigen Li, Hongjian Lu*, Carboxylate-assisted Iridium-Catalyzed C-H Amination of Arenes with Biologically Relevant Alkyl Azides. Chem. - Eur. J., 2016, 22, 2920-2924.

 


10. Tao Zhang, Zisong Qi, Xueyun Zhang, Lamei Wu, Xingwei Li*, Rh(III)-Catalyzed Hydroacylation Reactions between N-Sulfonyl 2-Aminobenzaldehydes and Olefins, Chem. - Eur. J., 2014, 20, 3283-3287. (Back Cover)

 


9. Zhiyou Li, Lamei Wu*, Tao Zhang, Zhengxi Huang, Guofu Qiu, Zhongqiang Zhou, Longfei Jin, N-2-Hydroxybenzaldehyde Acylhydrazone-Fe(III) complex: Synthesis, Crystal Structure and Its Efficient and Selective N-methylation. Dalton. Trans., 2014, 43, 7554-7560.

 


8. Tingting Yang, Tao Zhang, Shangdong Yang, Shanshan Chen, Xingwei Li*, Rhodium(III)-Catalyzed Coupling of N-Sulfonyl 2-Aminobenzaldehydes with Oxygenated Allylic Olefins through C-H Activation. Org. Biomol. Chem., 2014, 12, 4290-4294. (T. Yang and T. Zhang contributed equally)

 


7. Yimeng Zhang, Tao Zhang, Haoqiang Zhan and Xingwei Li*. Rh(III)-accelerated Synthesis of Quinoline Derivates Via Annulation of N-Sulfonyl 2-Aminobenzaldehydes with Olefins. Chin. J. Catal.2014, 35, 1840-1845. (Y. Zhang and T. Zhang contributed equally)

 


6. Tao ZhangLamei Wu*and Xingwei Li*. Rh(III)-Catalyzed Olefination of NSulfonyl Imines: Synthesis of Ortho-Olefinated Benzaldehydes. Org. Lett., 2013, 15, 6294-6297.

 


5. Xianran He, Min Zhong, Tao Zhang, Wen Wu, Zhongyuan Wu, Yuling Xiao,  Xianming Hu*, Synthesis and anticonvulsant activity of ethyl 1-(2-arylhydrazinecarboxamido)-2,2-dimethylcyclopropanecarboxylate derivatives. Eur. J. Med. Chem., 2012, 54, 542-548.

 


4. Xianran He, Min Zhong, Tao Zhang, Jin Yang, Zhongyuan Wu, Yuling Xiao, Hao Guo, Guofu Qiu, Xianming Hu*, Synthesis and anticonvulsant activity of 1-(8-(benzyloxy)quinolin-2-yl)-6-substituted-4,6-diazaspiro[2,4]heptane-5,7-diones. Eur. J. Med. Chem., 2012, 48, 338-346.

 


3. Hao Guo, Guolan Zhang, Tao Zhang, Xianran He, Zhongyuan Wu, Yuling Xiao, Yuanhu Pan, Guofu Qiu, Peng Liu, Xianming Hu*, Synthesis, characterization and biological evaluation of some 16β-azolyl-3β-amino-5α-androstane derivatives as potential anticancer agents. Eur. J. Med. Chem., 2011, 46, 3662-3674.

 


2. Jin Yang, Zhen Qu, Yuling Xiao, Guofu Qiu, Tao Zhang, Zhongyuan Wu, Xianran He, Xianming Hu*, Chemical composition and antioxidant activity of the essential oil of endemic Viola tianshanica. Natural. Product. Research., 2011, 25, 1635-1640.

 


1. Xianran He, Min Zhong, Tao Zhang, Wen Wu, Yuling Xiao, Jin Yang, Zhongyuan Wu, Yuanhu Pan, Guofu Qiu, Xianming Hu*, Synthesis and anticonvulsant activity of N-3-arylamide substituted 5,5-cyclopropanespirohydantoin derivatives. Eur. J. Med. Chem., 2010, 45, 5870-5877.