2025
82. 
S. Zhong,+ S. Gan,+ X. Zhang,+ L. Song,* L. Shi*
Structurally Constrained Cyclic (Diacyloxyiodo)arenes as an Enabling Platform for Hypervalent iodine(III) Chemistry
81. 
P. Gong, L. Wang, C. Tian, S. Hao, L. Shi*
Pd-Catalyzed C(sp2)-P Cross-Coupling of Aryl Thianthrenium Salts
Chem. Eur. J. 2025, 31(38), e202501060.
80.
L. Wang,+ J. Yin,+ S. Gan, X. Yang, S. Hao, L. Shi*
Non-Covalent-Interaction-Dictated Product Selectivity in Intermolecular and Intramolecular Controllable Oxidation of Aromatic Amines Using 2,2’-Diperoxyphenic Acid
Adv. Synth. Catal. 2025, 367(14), e9598.
79. 
C. Tian, L. Shi*
Photoinduced Ring-Opening Functionalization of α-Imino-Oxy Acids and Alkanols Enabled by Phthalate-Derived Proton-Coupled Electron Transfer Mediator
Chin. J. Chem. 2025, 43(16), 1988-1996.
78.
C. Wei, K. Fu, Z. Yu, Z. Zhan, D. Chang, L. Shi*
Photochemical Generation and Cycloadditions of Strained Cycloallkynes
J. Am. Chem. Soc. 2025, 147(17), 14299-14307.
77. 
H. Gao, X. Yang, L. Shi*
Asymmetric Oxidative Rearrangement of Indoles Enabled by Dual Catalysis with in situ Generated Acyl Hypoiodite and Chiral Phosphoric Acid
Org. Chem. Front. 2025, 12(13), 3848-3855.
76. 
Z. Yu,+ Z. Zhan,+ K. Fu, L. Shi*
Intramoleculear and intermolecular benzannulation of arylethanone derivatives enabled by visible light-induced catalytic generation of tether-tunable distonic radical anions
Org. Chem. Front. 2025, 12(12), 3568-3578.
75. 
S. Zhong, Z. Yu, Y. Zhu, L. Shi*
Catalytic Fluorination of α-Branched Ketones with Nucleophilic Fluorine
Org. Lett. 2025, 27(13), 3452-3458.
74. 
C. Wei, D. Chang, N. Feng, Z. Zhan, L. Shi*
A Unified Approach to Lactonization/Lactamization by Leveraging Tether-Tunable Distonic Radical Anions
Org. Lett. 2025, 27(11), 2582-2586.
73. 
C. Tian, L. Shi*
Photochemical generation of heteroatom (N, Si, B) or carbon radicals leveraging preinstalled carboxylic acids
Org. Chem. Front. 2025, 12(8), 2838-2859.
2024
72. 
T. Yuan, L. Shi*
Recent advances in carbon atom addition for ring-expanding single-atom skeletal editing
Org. Chem. Front. 2024, 11(24), 7318-7332.
71. 
K. Fu, L. Shi*
Enabling Site-Selective C–H Functionalization of Aliphatic Alcohols and Amines with exo-Directing Groups by Tether-Tunable Design of PdII/PdIV Catalysis
ACS Catal. 2024, 14(22), 17077-17083.
70. 
C. Tian, L. Shi*
Photoinduced cross-coupling of aryl halides enabled by n-tetrabutylphosphonium phthalate
Org. Chem. Front. 2024, 11(23), 6718-6727.
69. 
K. Fu,+ X. Yang,+ Z. Yu, L. Song*, L. Shi*
Revealing the Nature of Covalently Tethered Distonic Radical Anions in the Generation of Heteroatom-Centered Radicals: Evidence for the Polarity-Matching PCET Pathway
Chem. Sci. 2024, 15(31), 12398-12409.
68. 
T. Yuan, K. Fu, L. Shi*
Palladium(II)-Catalyzed Intramolecular C–H Amination to Carbazole: the Crucial Role of Cyclic Diacyl Peroxides
Org. Chem. Front. 2024, 11(16), 4529-4538.
67.
C. Wei, Z. Yu, L. Shi*
Two Catalytic Protocols for the Synthesis of CF2-Containing Quinazolinones via Domino Reaction
Adv. Synth. Catal. 2024, 366(14), 3181-3187.
66. 
X. Yang, H. Gao, J. Yan, J. Zhou*, L. Shi*
Intramolecular Chaperone-Assisted Dual-Anchoring Activation (ICDA): A Suitable Preorganization for Electrophilic Halocyclization
Chem. Sci. 2024, 15(16), 6130-6140.
2023
65. 
J.-J. Yin, Y.-P. Wang, J. Xue, F.-F. Zhou, X.-Q. Shan, R. Zhu, K. Fang, L. Shi*, S.-Y. Zhang, S.-H. Hou*, W.-J. Xia, Y.-Q. Tu*
Total Synthesis of Polycyclic Diterpenes Phomopsene, Methyl Phomopsenonate, and iso-Phomopsene via Reorganization of C–C Single Bonds
J. Am. Chem. Soc. 2023, 145(39), 21170-21175.
64.
S. Gan, S. Zhong, L. Wang, L. Shi*
Synthesis and Application of Organic Hypervalent Bromine Reagents
有机高价溴试剂的合成及其应用研究
Acta Chim. Sinica 2023, 81(8), 1030-1042.
63.
Z. Zhan,+ J. Yan,+ Z. Yu, L. Shi*
Recent Advances in Asymmetric Catalysis Associated with B(C6F5)3
2022
62.
X.-H. Yang, H.-W. Gao, J. Yan and L. Shi*
Recent Progress in Radical-Mediated Si-H Functionalization of Silanes: An Effective Strategy for Synthesis of Organosilanes Containing C-Si Bond
自由基介导的硅烷Si-H 键官能团化研究进展:一种合成含C-Si键有机硅化合物的有效策略
Chin. J. Org. Chem. 2022, 44, 106023/cjoc202207047.
61. 
Z. Yu and L. Shi*
Synthetic routes to bicyclo[1.1.1]pentylamines: booming toolkits for drug design
Org. Chem. Front. 2022, 9(13), 3591-3597.
60. 
S. Gan, J. Yin, Z. Yu, L. Song* and L. Shi*
A one-pot and two-stage Baeyer-Villiger reaction using 2,2'-diperoxyphenic acid under biomolecule-compatible conditions
Green. Chem. 2022, 24(5), 2232-2239.
59.
R. L.-Y. Bao, L. Shi* and K. Fu
Highly enantioselective construction of CF3-bearing all-carbon quaternary stereocenters: Chiral spiro-fused bisoxazoline ligands with 1,1'-binaphthyl sidearm for asymmetric Michael-type Friedel-Crafts reaction
Chin. Chem. Lett. 2022, 33(5), 2415-2419.
2021
58.
X. Yang, D. Chang, R. Zhao and L. Shi*
Recent Advances and Uses of (Me4N)XCF3(X = S, Se) in theSynthesis of Trifluoromethylthiolated andTrifluoromethylselenolated Compounds
Asian J. Org. Chem., 2021, 10(1), 61-73.
2020
57.
R. Zhao, K. Fu, Y. Fang, J. Zhou* and L. Shi*
Site-Specific C(sp3)−H Aminations of Imidates and Amidines Enabled by Covalently Tethered Distonic Radical Anions
Angew. Chem. Int. Ed., 2020, 59(46), 20682–20690.
56.
D. Zhu, S. Gan, R. L.-Y. Bao and L. Shi*
Copper-catalyzed cross-coupling of vinyliodonium salts and diboron reagents to generate alkenyl boronic esters
Org. Biomol. Chem., 2020, 18(29), 5567-5570.
55.
R. Zhao and L. Shi*
Reactions between Diazo Compounds and Hypervalent Iodine(III) Reagents
Angew. Chem. Int. Ed., 2020, 59(30), 12282–12292.
54.
R. L.-Y. Bao+, J. Yin+, L. Shi* and L. Zheng
Rh(I)-Catalyzed enantioselective and scalable [4 + 2] cycloaddition of 1,3-dienes with dialkyl acetylenedicarboxylates
Org. Biomol. Chem., 2020, 18(15), 2956-2961.
2019
53. 
L. Shi*, R. L.‐Y. Bao, L. Zheng and R. Zhao
B(C6F5)3‐Catalyzed Reduction of Cyclic N‐Sulfonyl Ketimines
Eur. J. Org. Chem., 2019, 2019(38), 6550–6556.
52.
Y. Fang, R. Zhao, Y. Yao, Y. Liu, D. Chang, M. Yao and L. Shi*
Trichloroacetonitrile as an efficient activating agent for the ipso-hydroxylation of arylboronic acids to phenolic compounds
Org. Biomol. Chem., 2019, 17(32), 7558–7563.
2018
51.
R. Zhao and L. Shi*
A renaissance of ligand-to-metal charge transfer by cerium photocatalysis
Org. Chem. Front., 2018, 5(20), 3018-3021.
50.
D. Zhu and L. Shi*
Ni-catalyzed cross-coupling of aryl thioethers with alkyl Grignard reagents via C–S bond cleavage
Chem. Commun., 2018, 54(67), 9313-9316.
49.
C. Wei, R. Zhao, Z. Shen, D. Chang and L. Shi*
Two Catalytic Protocols for Achmatowicz Rearrangement by Using Cyclic Diacyl Peroxides as Oxidants
Org. Biomol. Chem., 2018, 16(31), 5566-5569.
48.
D. Chang, F. Gao and L. Shi*
Potassium tert-butoxide-mediated generation of arynes from o-bromoacetophenone derivatives
Tetrahedron, 2018, 74(20), 2428-2434.
47.
Y. Zhang, L. He and L. Shi*
Asymmetric hydrogenolysis of racemic 3-substitued-3-hydroxy-isoindolin-1-ones employing SPINOL-derived chiral phosphoric acid
Tetrahedron Lett., 2018, 59(16), 1592-1595.
46.
Y. Zhang, L. He and L. Shi*
Chiral Ion-pair Organocatalyst Promoted Efficient Enantioselective Reduction of α-Hydroxy Ketones
Adv. Synth. Catal., 2018, 360(10), 1926-1931.
45.
D. Chang, R. Zhao, C. Wei, Y. Yao, Y. Liu and L. Shi*
Sulfonamide-Directed Chemo- and Site-Selective Oxidative Halogenation/Amination Using Halogenating Reagents Generated in situ from Cyclic Diacyl Peroxides
J. Org. Chem., 2018, 83(6), 3305-3315.
44.
D. Zhu, Y. Yao, R. Zhao, Y. Liu and L. Shi*
Metal-Free Geminal Difunctionalization of Diazocarbonyl Compounds: A One-Pot Multicomponent Strategy for the Construction of α,β-Diamino Carbonyl Derivatives
Chem. Eur. J., 2018, 24(19), 4805-4809.
43.
F. Ding, Y. Jiang, K. Lin and L. Shi*
Tandem radical cyclization for the construction of 1-difluoroalkylated isoquinolines via Cu catalyzed and visible light-promoted pathways
Org. Biomol. Chem., 2018, 16(11), 1812-1815.
42.
F. Ding, Y. Fang, Y. Jiang, K. Lin and L. Shi*
Tandem Radical Cyclization for the Construction of Difluoro-Containing Oxindoles and Quinoline-2,4-diones
Chem. Asia. J., 2018, 13(6), 636-640.
41.
R. Zhao+, Y. Yao+, D. Zhu, D. Chang, Y. Liu and L. Shi*
Visible-Light-Enhanced Ring Opening of Cycloalkanols Enabled by Bronsted Base-Tethered Acyloxy Radical Induced Hydrogen Atom Transfer-Electron Transfer
Org. Lett., 2018, 20(4), 1228-1231.
2017
40. 
F. Ding, Y. Zhang, R. Zhao, Y. Jiang, R. L.-Y. Bao, K. Lin and L. Shi*
B(C6F5)3-promoted hydrogenations of N-heterocycles with ammonia borane
Chem. Commun., 2017, 53(66), 9262-9264.
39.
Y. Zhang, Y. Yao, L. He, Y. Liu and L. Shi*
Rhodium(II)/Chiral Phosphoric Acid Co-Catalyzed Enantioselective O–H Bond Insertion of α-Diazoesters (as VIP)
Adv. Synth. Catal., 2017, 359(16), 2754-2761.
38.
R. Zhao, D. Chang and L. Shi*
Recent Advances in Cyclic Diacyl Peroxides: Reactivity and Selectivity Enhancement Brought by Cyclic Structure
Synthesis., 2017, 49(15), 3357-3365.
37.
F. Ding, Y. Jiang, S. Gan, R. L.-Y. Bao, K. Lin and L. Shi*
B(C6F5)3-Catalyzed Deoxygenation of Sulfoxides and Amine N-Oxides with Hydrosilanes
Eur. J. Org. Chem., 2017, 2017(24), 3427-3430.
36.
S. Gan, J. Yin, Y. Yao, Y. Liu, D. Chang, D. Zhu and L. Shi*
Metal- and additive-free oxygen-atom transfer reaction: an efficient and chemoselective oxidation of sulfides to sulfoxides with cyclic diacyl peroxides
Org. Biomol. Chem., 2017, 15(12), 2647-2654.
2016
35. 
D. Zhu, D. Chang, S. Gan and L. Shi*
Direct α-acyloxylation of organic sulfides with the hypervalent (diacyloxyiodo)benzene/tetra-n-butylammonium bromide (TBAB) reagent combination
RSC Adv., 2016, 6(33), 27983-27987.
2015
34.
D. Chang, D. Zhu and L. Shi*
[3+2] Cycloadditions of Azides with Arynes via Photolysis of Phthaloyl Peroxide Derivatives
J. Org. Chem., 2015, 80(11), 5928-5933.
33.
S. Kong, L. Zhang, X. Dai, L. Tao, C. Xie, L. Shi* and M. Wang*
DDQ-mediated Direct C(sp3)-H Cyanation of Benzyl Ethers and 1,3-Diarylpropenes under Solvent- and Metal-free Conditions
Adv. Synth. Catal., 2015, 357(11), 2453-2456.
32.
Y. Zhang, R. Zhao, R. L.-Y. Bao and L. Shi*
Highly Enantioselective SPINOL-Derived Phosphoric Acid Catalyzed Transfer Hydrogenation of Diverse C=N-Containing Heterocycles
Eur. J. Org. Chem., 2015, 2015(15), 3344-3351.
31.
D. Zhu, D. Chang and L. Shi*
Transition-metal-free cross-coupling of thioethers with aryl(cyano)iodonium triflates: a facile and efficient method for the one-pot synthesis of thiocyanates
Chem. Commun., 2015, 51(33), 7180-7183.
30.
R. L.-Y. Bao, R. Zhao and L. Shi*
Progress and developments in the turbo Grignard reagent i-PrMgCl·LiCl: a ten-year journey
Chem. Commun., 2015, 51(32), 6884-6900.
29.
D. Chang, D. Zhu, P. Zou and L. Shi*
Cleavage of C-N bonds in guanidine derivatives and its relevance to efficient C-N bonds formation
Tetrahedron, 2015, 71(11), 1684-1693.
2014
28. 
R. Zhao and L. Shi*
Promising Combination for Asymmetric Organocatalysis: Bronsted Acid-Assisted Chiral Phosphoric Acid Catalysis
ChemCatChem., 2014, 6(12), 3309-3311.