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张永磊在JMC报道CDK6/PARP双靶点抑制剂
发布时间:2025-06-13

Yonglei Zhang, Fucheng Yin, Zhongwen Luo, Yiwei Zheng, Shunxin Guo, Sijie Wu, Yuhan Jiang, Long Zheng, Liangliang Ma, Meiting Zou, Xiaobing Wang, Lingyi Kong.

Design and Synthesis of PARP/CDK6 Dual Target Inhibitors and Modulation of Wnt/β-catenin Signaling Pathway for the Treatment of BRCA Wild-Type TNBC

Journal of Medicinal Chemistry, 2025, 68, 12, 13030–13056. DOI: 10.1021/acs.jmedchem.5c01058.


【JMC】新型PARP/CDK6双靶点抑制剂的设计合成及在BRCA野生型TNBC治疗中的作用机制