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61)SH2 Decarboxylative Monofluoromethylation of Aliphatic Carboxylic Acids Enabled by Nickel/Photoredox Dual Catalysis

 Angew Chem Int Ed  2025, 64(32)e202507632,DOI: doi.org/10.1002/anie.202507632.

Ting-Yu Fang, Meng-Ye Jiang, Meng-Meng Zheng, Jun-An Ma, and Fa-Guang Zhang*

Dedicated to the 130th anniversary of Tianjin University

Highlighted by Mark Lautens in Synfacts 2025, 21(08), 790. 


60)DBU-Triggered One-Pot Domino Transformation of Trifluoromethyl Ketones and Dicyanoalkenes into gem-Difluoroalkenyl γ-Lactams. 

 Adv. Syn. Catal. 2025367(17)e70090DOI: doi.org/10.1002/adsc.70090

Jian Wang, Cheng-Feng Gao, Houwen Zhou, Feng Li,* Jing Nie,*  Jun-An Ma, and  Fa-Guang Zhang*


59)Transition-Metal-Free Three-Component Chalcogen-Trifluoromethylation of Alkenes Enabled by a Catalytic Electron Donor-Acceptor Complex. 

 Chin J Chem  202543, 2642—2648 (Back Cover),   https://doi.org/10.1002/cjoc.70157. 

Hao-Yan Wu, Xiaodong Tang, Ran Guo,  Fa-Guang Zhang*, and Jun-An Ma *  


58)Transition metal/photocatalyst-free skeletal editing of indene with iodonium difluorodiazo reagent to access 2- (difluoromethyl)naphthalene. 

 Chem Commun 2025, 61(48), 8667-8670. DOI: 10.1039/d5cc01777g

Zong-Rui Yuan, Meng-Qi Sun, Wei-Chen Chen, Zhi-Qi Zhang, Jun-An Ma,* and Fa-Guang Zhang*

Highlighted in ChemComm Pioneering Investigators 2025 Collection(https://pubs.rsc.org/en/content/articlelanding/2025/cc/d5cc90272j).  


57)Photoinduced [3 + 2] Radical Cyclization of α‑Diazodifluoroethyl Sulfonium Salt with Hydrazones 

J. Org. Chem. 2025,  90(20), 6834-6843. DOI: 10.1021/acs.joc.5c00675

Ming-Yue He, Hao-Yan Wu, Xiaodong Tang, Jun-An Ma, and Fa-Guang Zhang*



56)17.2.1.10 1,2,3-Triazines (Update 2025), 17.2.2.4 1,2,4-Triazines (Update 2025)

Science of Synthesis 2025DOI: 10.1055/sos-SD-117-00732, DOI: 10.1055/sos-SD-117-00712. 

Fa-Guang Zhang* and Jun-An Ma*


55)Fe-Catalyzed Stereospecific Intramolecular Friedel–Crafts-type Reaction of Fluoroalkyl Cyclopropyl Carbinols via Non-classical Carbocation. 

 Adv. Syn. Catal. 2025367(10), e202500242DOI: 10.1002/adsc.202500242

Hong-Song Shi, Jun-An Ma,* Ilan Marek,* and Fa-Guang Zhang* 


54)Chemoenzymatic Synthesis of Fluorinated Mycocyclosin Enabled by the Engineered Cytochrome P450-Catalyzed Biaryl Coupling Reaction. 

 J. Am. Chem. Soc. 2024146, 19962-19973, DOI: 10.1021/jacs.4c03499

Shuo-Han Li,† Xue Zhang,† Ze-Long Mei, Yongjun Liu,* Jun-An Ma,* and Fa-Guang Zhang* 


53)Enzymatic Stereodivergent Access to Fluorinated β‑Lactam Pharmacophores via Triple-Parameter Engineered Ketoreductases. 

 ACS Catal. 202414, 6358−6368, DOI: 10.1021/acscatal.4c00945

Ze-Long Mei,† Cong-Cong Li,† Xu Han,† Yu-Chen Tian, Shuo-Han Li, Weidong Liu, Ge Qu, Manfred T. Reetz, Zhoutong Sun,* Jun-An Ma,* and Fa-Guang Zhang* 

Highlighted by Andrew Sutherland in Nat. Prod. Rep. 2024,41, 868-872


52)Catalytic photoactivation of a triarylamine electron donor-acceptor complex for difunctionalization of alkenes

Cell Reports Physical Science 2024, 5, 102135, DOI: 10.1016/j.xcrp.2024.102135

 Hao-Yan Wu†, Xiaodong Tang†,*,  Ran Guo, Hwee Ting Ang, Jing Nie, Jie Wu, Jun-An Ma*, Fa-Guang Zhang* 


51)The Smallest Monofluorodiazoethane Reagent and Its [3 + 2] Cycloaddition Reactions. 

 CCS Chemistry 2024, 6, 28252834, DOI: 10.31635/ccschem.024.202403849

 Xiaodong Tang†, Ming-Yue He†, Ran Guo, Hao-Nan Liu, Jing Nie, Ilan Marek, Jun-An Ma, Fa-Guang Zhang* 


50)Allylation,  Alkenylation and Alkynylation of Monofluoromethyl Ketyl Radical Enabled by Photoredox Halogen-Atom-Transfer 

ChemCatChem 202416, e202401622DOI: 10.1002/cctc.202401622

Meng-Qi Sun,† Shi-Jing Zhai, Jing Nie,* Ying Cheng, Xiaojuan Deng, Guosheng Ding, Dominique Cahard, Jun-An Ma, and Fa-Guang Zhang*


49)Nickel-catalysed enantioselective cross-electrophile coupling reaction with the retention of ß-fluorine atom

Org. Chem. Front. 202411, 6459–6469 DOI: 10.1039/d4qo01555j

Xin-Yi Shi,Xueyuan Yan, Xiaodong Tang, Shi-Jing Zhai, Genping Huang, Jun-An Ma, and Fa-Guang Zhang*


48)Regioselective Synthesis of Multisubstituted Fluoropyrazoles via Silver-Catalyzed One-Pot Cyclization Reaction of Diazo Reagents with Fluoronitroalkenes. 

Adv. Synth. Catal. 20243663516-3521, DOI: 10.1002/adsc.202400385

Rong Wang, Jing Nie,* Xiaojuan Deng, Guosheng Ding,  Fa-Guang Zhang,* and Jun-An Ma* 


47)Copper-Catalyzed Regio- and Enantioselective Hydroboration of Difluoroalkyl-Substituted Internal Alkenes. 

Adv. Sci. 2023, 10, 2304194, DOI: 10.1002/advs.202304194

Tao-Qian Zhao, Hui Xu, Yu-Chen Tian, Xiaodong Tang, Yandeng Dang, Shaozhong Ge,* Jun-An Ma,* and Fa-Guang Zhang* 

Dedicated to Professor Ilan Marek on the occasion of his 60th birthday


46)Programmable synthesis of difluorinated hydrocarbons from alkenes through a photocatalytic linchpin strategy. 

Chem. Sci. 2023, 14, 11546–11553, DOI: 10.1039/d3sc03951j

Zhi-Qi Zhang, Cheng-Qiang Wang, Long-Ji Li, Jared L. Piper, Zhi-Hui Peng,* Jun-An Ma,* Fa-Guang Zhang,* and Jie Wu*


45)Tetrazole Diversification of Amino Acids and Peptides via Silver-Catalyzed Intermolecular Cycloaddition with Aryldiazonium Salts. 

Angew. Chem. Int. Ed. 2023, 62(37), e202304740 (Hot Paper, Front Cover), DOI: 10.1002/anie.202304740

Xuan-Yu Liu, Yi-Lin Yang, Yanfeng Dang, Ilan Marek,* Fa-Guang Zhang,* and Jun-An Ma* 

Highlighted by Hisashi Yamamoto in Synfacts 2023, 19(09), 0945. 


44) Dirhodium(II)-catalyzed enantioselective cyclopropenation of internal alkynes with trifluoromethyl carbene. 

Chem. Catal. 2023, 3, 10637, DOI: 10.1016/j.checat.2023.100637

Xiu-Qing Cui, Meng-Meng Zheng, Xiaodong Tang, Zhi-Qi Zhang, Ilan Marek*, Jun-An Ma*, and Fa-Guang Zhang*

Highlighted by Dominique Cahard in Chem Catal 2023, 3, 100665. 


43) Highly Enantio- and Diastereoselective Hydrogenation of Cyclic Tetra-Substituted β-Enamido Phosphorus Derivatives. 

Angew. Chem., Int. Ed. 2023, 62(28), e202305315DOI: 10.1002/anie.202305315

Jun-Hao Zhang, Hui Xu, Xiaodong Tang, Yanfeng Dang*, Fa-Guang Zhang*, and Jun-An Ma*


42) Synthesis of di/trifluoromethyl cyclopropane-dicarbonitriles via [2+1] annulation of fluoro-based diazoethanes with (alkylidene)malononitriles. 

Chem. Commun. 2023, 59, 11664-11667, DOI: 10.1039/d3cc03897a

Cheng-Feng Gao, Yue-Ji Chen, Jing Nie, Fa-Guang Zhang,* Chi Wai Cheung,* and  Jun-An Ma* 


41) Electron Donor−Acceptor Complex Enabled Radical Cyclization of α‑Diazodifluoroethyl Sulfonium Salt with Unactivated Alkynes. 

Org. Lett. 2023, 25(50), 9041−9046, DOI: 10.1021/acs.orglett.3c03790

 Ming-Yue He, Xiaodong Tang,‡,* Hao-Yan Wu, Jing Nie, Jun-An Ma,* and Fa-Guang Zhang,* 


40)  Photoinduced Defluorinative Branch-Selective Olefination of Multifluoro (Hetero)arenes. 

Org. Lett. 2023, 25(5), 883–888, DOI: 10.1021/acs.orglett.3c00115

Ye Yuan, Muliang Zhang, Xiaodong Tang, Jared L. Piper, Zhi-Hui Peng, Jun-An Ma*, Jie Wu*, and Fa-Guang Zhang*,


39) Silver-catalysed [3 + 2] annulation reaction of aryldiazonium salts with allenes enabled by boronate direction. 

Org. Chem. Front. 2023, 10(1), 74–82, DOI: 10.1039/d2qo01585d

Xing Peng, Meng-Meng Zheng, Pei Qin, Xiao-Song Xue,* Fa-Guang Zhang,* and Jun-An Ma*, 


38) Difluoromethylation of Unactivated Alkenes Using Freon-22 through Tertiary Amine-Borane-Triggered Halogen Atom Transfer. 

J. Am. Chem. Soc. 2022, 144(31), 14288−14296, DOI: 10.1021/jacs.2c05356

Zhi-Qi Zhang, Yue-Qian Sang, Cheng-Qiang Wang, Peng Dai, Xiao-Song Xue, Jared L. Piper, Zhi-Hui Peng, Jun-An Ma,* Fa-Guang Zhang,* and Jie Wu*

Highlighted by Benjamin List in Synfacts 2022, 18(10), 1134 . 


37) Dual Incorporation of Trifluoromethyl and Cyano Groups into Pyrazole Pharmcophores via Silver-Catalyzed Cycloaddition Reaction of Trifluorodiazoethane

CCS Chem. 2022, 4(12), 3693–3704,  DOI: 10.31635/ccschem.022.202201923

Cheng-Feng Gao, Yin Zhou, Hai Ma, Yue Zhang, Jing Nie, Fa-Guang Zhang,* and Jun-An Ma* 


36)  Metal-free regioselective construction of 2-aryl-2H-tetrazol-5-yl difluoromethylene phosphonates

Chin. Chem. Lett. 2022, 33(2), 863–866, DOI: 10.1016/j.cclet.2021.08.007

Shi-Jing Zhai, Dominique Cahard, Fa-Guang Zhang,* and Jun-An Ma* 


35) Quadruple Functionalized Pyrazole Pharmacophores via One-pot Regioselective [3 + 2] Cycloaddition of Fluorinated Nitrile Imines and Dicyanoalkenes. 

Chem. Asian J. 2022, 17, e202200436, DOI: 10.1002/asia.202200436

Yin Zhou, Cheng-Feng Gao, Hai Ma, Jing Nie,* Jun-An Ma*, and Fa-Guang Zhang*


34)Enantioselective Construction of Amino Carboxylic-Phosphonic Acid Derivatives Enabled by Chiral Amino Thiourea-Catalyzed Decarboxylative Mannich Reaction.

Adv. Synth. Catal. 2022, 364(11), 1908−1912 (Very Important Publication), DOI: 10.1002/adsc.202200306

Xue-Qi Wang, Fang-Fang Feng, Jing Nie, Fa-Guang Zhang,* and Jun-An Ma* 


33)Triazines: Syntheses and Inverse Electron-demand Diels−Alder Reactions. 

Chem. Rev. 2021, 121(23), 14555–14593DOI: 10.1021/acs.chemrev.1c00611

Fa-Guang Zhang,*, Zhen Chen, Xiaodong Tang, and Jun-An Ma* 


32) Catalytic regioselective construction of phenylthio- and phenoxyldifluoroalkyl tetrazoles from difluorodiazoketones.

 Chem. Commun. 2021, 57(100), 13744–13747, DOI: 10.1039/d1cc05890h

Hong-Song Shi, Shuo-Han Li, Fa-Guang Zhang,* and Jun-An Ma* 


31) N‑Iodosuccinimide-Promoted [3 + 2] Annulation Reaction of Aryldiazonium Salts with Guanidines To Construct Aminotetrazoles.  

Org. Lett. 2021, 23, 8894−8898, DOI: 10.1021/acs.orglett.1c03395

Yi-Lin Yang, Shen Li, Fa-Guang Zhang,* and Jun-An Ma* 

Highlighted by Mark Reed in Synfacts 2022, 18(03), 0248. 


30Zinc-Enabled Annulation of Trifluorodiazoethane with 2H‑Azirines to Construct Trifluoromethyl Pyrazolines, Pyrazoles, and Pyridazines.

 Org. Lett. 2021, 23, 6062−6066,  DOI: 10.1021/acs.orglett.1c02139

 Yue-Ji Chen, Fa-Guang Zhang,* and Jun-An Ma* 


29) From Chemical Synthesis to Biosynthesis: New Trends toward Total Synthesis of Natural Products.

 Synthetic Biology Journal 2021, 2(5), 674-696 (Front Cover). 

Fa-Guang ZhangGe Qu, Zhou-Tong Sun,* and Jun-An Ma* 


28) Regioselective Decarboxylative Cycloaddition Route to Fully Substituted 3-CF3-Pyrazoles from Nitrilimines and Isoxazolidinediones” 

Adv. Synth. Catal. 2021, 363 (8), 2093–2097 (Very Important Publication), DOI: 10.1002/adsc.202100091

Yu-Chen Tian, Jun-Kuan Li, Fa-Guang Zhang,* and Jun-An Ma* 


27) Asymmetric Synthesis of Chiral Amino Carboxylic-Phosphonic Acid Derivatives

Adv. Synth. Catal. 2021, 363, 688−729, DOI: 10.1002/adsc.202001345

Hao-Qiang Cao, Jun-Kuan Li, Fa-Guang Zhang,* Dominique Cahard,* and Jun-An Ma* 


26) Remote Fluorination and Fluoroalkyl(thiol)ation Reactions

Chem.-Eur. J. 2020, 26, 15378–15396, DOI: 10.1002/chem.202003416

Fa-Guang Zhang,* Xue-Qi Wang, Yin Zhou, Hong-Song Shi, Zhe Feng, Jun-An Ma, and Ilan Marek* 


25) Aryl Diazonium Salt-Triggered Cyclization and Cycloaddition Reactions: Past, Present, and Future 

Chin. J. Chem. 2020, 38(10), 1132–1152,  DOI: 10.1002/cjoc.202000270

Fa-Guang Zhang, Zhen Chen, Chi Wai Cheung,* and Jun-An Ma* 


24)  Potassium Acetate-Catalyzed Double Decarboxylative Transannulation To Access Highly Functionalized Pyrroles.

Org. Lett. 2020, 22(24), 9585–9590, DOI: 10.1021/acs.orglett.0c03621

Jun-Kuan Li, Biying Zhou, Yu-Chen Tian, Chunman Jia, Xiao-Song Xue, Fa-Guang Zhang,* and Jun-An Ma*

 

23) Catalytic Enantioselective Synthesis of Difluoromethylated Tetrasubstituted Stereocenters in Isoindolones Enabled by a Multiple-Fluorine System.

Org. Lett. 2020, 22(22), 9010–9015, DOI: 10.1021/acs.orglett.0c03406

Meng-Yu Rong, Jin-Shan Li, Yin Zhou, Fa-Guang Zhang,* and Jun-An Ma* 


22) Catalytic Direct Construction of Cyano-tetrazoles 

Org. Lett. 2020, 22(19), 7762–7767, DOI: 10.1021/acs.orglett.0c03025

 Ming-Yang Xiao, Meng-Meng Zheng, Xing Peng, Xiao-Song Xue, Fa-Guang Zhang,* and Jun-An Ma* 


21) Silver-Catalyzed [3 + 2] Cycloaddition Approach to Coumarin-Decorated Tetrazoles

ChemCatChem 2020, 12, 5623–5626, DOI: 10.1002/cctc.202001143

Xuan-Yu Liu, Shi-Jing Zhai, Fang-Fang Feng, Fa-Guang Zhang,* and Jun-An Ma* 


20) Cu-Catalysed Three-Component Reaction of Aryldiazonium Salts with Fluorinated Diazo Reagents and Nitriles: Access to Difluoro- and Trifluoromethylated N1-Aryl-1,2,4-triazoles 

Adv. Synth. Catal. 2020, 362, 4432–4437, DOI: 10.1002/adsc.202000776

Xing Peng, Fa-Guang Zhang,* and Jun-An Ma* 


19) Direct Enamido C(sp2)-H Diphosphorylation Enabled by PCET-triggered Double Radical Relay: Access to gem-Bisphosphonates

 Chem.-Eur. J. 2020, 26, 5515–5521, DOI: 10.1002/chem.202000517 

Hao-Qiang Cao, Hao-Nan Liu, Zhe-Yuan Liu, Bao-Kun Qiao, Fa-Guang Zhang,* and Jun-An Ma* 


18) Phosphorylation of Bulky C(sp2)−H Bond to Build Fully Substituted β‑Phosphonodehydroamino Acids

Org. Lett. 2020, 22(16), 6414–6419, DOI: 10.1021/acs.orglett.0c02229 

Hao-Qiang Cao, Hao-Nan Liu, Zhe-Yuan Liu, Baokun Qiao, Fa-Guang Zhang,* and Jun-An Ma* 


17)Catalytic Enantioselective Cyclopropenation of Internal Alkynes: Access to Difluoromethylated Three-Membered Carbocycles

Angew. Chem., Int. Ed. 201958(50), 18191–18196  (Hot Paper, Back Cover), DOI: 10.1002/anie.201911701

Zhi-Qi Zhang, Meng-Meng Zheng, Xiao-Song Xue, Ilan, Marek,* Fa-Guang Zhang,* and Jun-An Ma* 

Highlighted by 卿凤翎 院士 in Chin. J. Org. Chem. 2020, 40, 806~807. 

Highlighted by Paul Knochel in Synfacts 2020, 16(02), 0173. 


16) Silver-Catalyzed [3 + 3] Dipolar Cycloaddition of Trifluorodiazoethane and Glycine Imines: Access to Highly Functionalized Trifluoromethyl-Substituted Triazines and Pyridines

ACS Catal. 2019, 9, 4600−4608. (Impact factor 11.384), DOI: 10.1021/acscatal.9b00846

Zhen Chen, Nan Ren, Xiaoxiao Ma, Jing Nie, Fa-Guang Zhang,* and Jun-An Ma* 

Highlighted by Victor Snieckus in Synfacts 2019, 15(08), 0864. 


15) Catalytic Direct Regioselective Synthesis of Phosphonylated Tetrazoles from Aryl Diazonium Salts and Seyferth-Gilbert Reagent

Org. Lett. 2019, 21(24), 9884–9888,  DOI: 10.1021/acs.orglett.9b03800

Shi-Jing Zhai, Xing Peng, Fa-Guang Zhang,* and Jun-An Ma* 


14) Chemodivergent and Stereoselective Construction of gem-Difluoroallylic Amines from Masked Difluorodiazo Reagents 

Org. Lett. 2019, 21(20), 8244–8249, DOI: 10.1021/acs.orglett.9b02989

Jun-Liang Zeng, Yue Zhang, Meng-Meng Zheng, Zhi-Qi Zhang, Xiao-Song Xue, Fa-Guang Zhang,* and Jun-An Ma*


13) Construction of Difluoromethylated Tetrazoles via Silver-Catalyzed Regioselective [3 + 2] Cycloadditions of Aryl Diazonium Salts

Org. Lett. 2019, 21(12), 4808–4811, DOI: 10.1021/acs.orglett.9b01697

Xing Peng, Ming-Yang Xiao, Jun-Liang Zeng, Fa-Guang Zhang,* and Jun-An Ma* 


12Construction of Chiral β‑Trifluoromethyl Alcohols Enabled by Catalytic Enantioselective Aldol-Type Reaction of CF3CHN2

Org. Lett. 2019, 21(11), 4280–4283, DOI: 10.1021/acs.orglett.9b01468

Meng-Yu Rong, Lijun Yang, Jing Nie, Fa-Guang Zhang,* and Jun-An Ma* 


11) Zinc-Mediated Mannich-Type Reaction of 2,2,2-Trifluorodiazoethane with Imines: Access to β‑CF3‑Amines

 Org. Lett. 2018, 20, 6994–6997, DOI: 10.1021/acs.orglett.8b02816

Ran Guo, Ning Lv, Fa-Guang Zhang,* and Jun-An Ma,* 


10) Direct Regioselective [3 + 2] Cycloaddition Reactions of Masked Difluorodiazoethane with Electron-Deficient Alkynes and Alkenes: Synthesis of Difluoromethyl-Substituted Pyrazoles

Org. Lett. 2018, 20(15), 4562–4565,  DOI: 10.1021/acs.orglett.8b01854

Jun-Liang Zeng, Zhen Chen, Fa-Guang Zhang,* and Jun-An Ma* 


9) Telescoping Reactions with Trifluorodiazoethane-Derived Aza-Wittig Reagents and Allenyl esters

Chem. Eur. J. 2018, 24(30), 7749–7754,  DOI: 10.1002/chem.201801171

Fa-Guang Zhang, Jun-Liang Zeng, Yi-Qiang Tian, Yan Zheng, Dominique Cahard, and Jun-An Ma* 


8) Phosphine-Relayed Aldehyde-Olefination and Aza-Wittig Reaction with 2,2,2-Trifluorodiazoethane

 Chin. J. Chem. 2018, 36, 723–730. 

 Fa-Guang Zhang,* Ning Lv, Yan Zheng, and Jun-An Ma*


7) One-Pot Cascade Transformations of Zinc Trifluorodiazoethylide and α,β-Unsaturated Enones: Access to Trifluoromethylated Polycyclic Pyrazolines

Org. Lett. 2017, 19(13), 3406–3409, DOI: 10.1021/acs.orglett.7b01362

Shuang Qin, Yan Zheng, Fa-Guang Zhang,* and Jun-An Ma* 


6) Brook Rearrangement as Trigger for Carbene Generation: Synthesis of Stereodefined and Fully Substituted Cyclobutenes

J. Am. Chem. Soc. 2017, 139, 8364−8370, DOI: 10.1021/jacs.7b04255

Fa-Guang Zhang and Ilan Marek


5) Brook Rearrangement as a Trigger for Ring-Opening of strained Carbocycles 

Angew. Chem., Int. Ed. 2016, 55, 714–718, DOI: 10.1002/anie.201510094

 Fa-Guang Zhang, Guillaume Eppe and Ilan Marek


4) Enantioselective Base-Free Electrophilic Amination of Benzofuran-2(3H)-ones: Catalysis by Binol-Derived P-Spiro Quaternary Phosphonium Salts

Angew. Chem., Int. Ed. 2011, 50, 58695872. 

Chuan-Le Zhu, Fa-Guang Zhang, Wei Meng, Jing Nie, Dominique Cahard, and Jun-An Ma

3) Regioselective Cycloaddition of Trifluorodiazoethane with Electron-Deficient Allenic Esters and Ketones: Access to CF3Substituted Pyrazolines and Pyrazoles

 Org. Lett. 2014, 16, 3122–3125. 

Fa-Guang Zhang, Yi Wei, Yu-Ping Yi, Jing Nie, and Jun-An Ma

2Enantioselective Diynylation of Cyclic N-Acyl Ketimines: Access to Chiral Trifluoromethylated Tertiary Carbinamines

 Adv. Synth. Catal. 2012, 354, 1422–1428.

 Fa-Guang Zhang, Hai Ma, Jing Nie, Yan Zheng, Qingzhi Gao and Jun-An Ma

1) Highly enantioselective organocatalytic Strecker reaction of cyclic N-acyl trifluoromethylketimines: synthesis of anti-HIV drug DPC 083. 

Chem. Commun. 2012, 48, 11552–11554. 

Fa-Guang Zhang, Xiao-Yan Zhu, Shen Li, Jing Nie and Jun-An Ma*