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15Hao Wei, Yujie Zhang, Sanlin Jin, Ying Yu, Ning Chen, Jiaxi Xu and Zhanhui Yang. PyBox–La(OTf)3-Catalyzed Enantioselective Diels–Alder Cycloadditions of 2-Alkenoylpyridines with Cyclopentadiene. Molecules 2024, 29(13), 2978; https://doi.org/10.3390/molecules29132978


14. Duo Fu, Jiaxi Xu. Synthesis of Sulfo(xo)nium Diacylmethylides. Eur. J. Org. Chem. 2024, e202400390.

 


13. Fu, Yuqing; Leng, Yijia; Bai, Haotong; Xu, Jiaxi;* Chen, Ning.* Regioselective oxidative cleavage of conjugated dienes to access α,β-unsaturated nitriles. Org. Chem. Front. 2024, 11, 3263–3269.



12.  Cunzhi Chen, Kang Lv, Youwei Chen, Hongguang Du, Jiaxi Xu, Tao Liu, and Zhanhui Yang. Catalytic Enantioselective (3+2) Annulations of Nucleophilic Thioacyl Rh(I)-Carbenes with Achmatowicz Rearrangement Products. ACS Catal. 2024, 14, 8949-8957.



11.  Yang Chen, Jingyu Zhang, Hongguang Du, Renshi Luo, Jiaxi Xu, Zhanhui Yang. Iridium-catalyzed reductive γ-lactonization of ortho-acylbenzoic acids in water: sustainable access to phthalides. Org. Chem. Front. 2024, 11, 2220-2230.



10.  Yujie Zhang, Shukui Shi, and Zhanhui Yang. Thiourea-Mediated Stereospecific Deoxygenation of Cyanoepoxides to Access Highly Diastereopure Alkenyl Nitriles. J. Org. Chem. 2024, 89, 2748-2758.



9. Chengzhuo Wang, Ning Chen, Zhanhui Yang, Jiaxi Xu. Y(OTf)3-Salazin-Catalyzed Asymmetric Aldol Condensation. Molecules, 2024, 29, 1963.

 

8. Wenlai Xie, Chengzhuo Wang, Jiaxi Xu. Reaction of 1,3,5-Triazinanes with Phosphoryl Diazomethanes: Access to 5-Phosphoryl-1,2,3,4-tetrahydropyrimidines. Org. Lett. 2024, 26, 3391-3396.

 

7. Yinqiao Wang, Yixiang Chen, Jiaxi Xu. π‑Stacking-Controlled Dearomatic Sulfur-Shifted Ene Reaction of Ketenes and Polycyclic Arylthiiranes: Access to Areno[d]‑ε-thiolactones. J. Org. Chem. 2024, 89, 4749-4759.



 

6. Duo Fu, Jiaxi Xu. Tf2O/2-Chloropyridine-Triggered Synthesis of Benzo[b]thiophene 1,1-Dioxides from Sulfonium α-Acyl Sulfonylmethylides. J. Org. Chem. 2024, 89, 3072-3083.


5. Hao Wei, Cunzhi Chen, Aijun Gao, Zhanhui Yang. Rh(I)-catalyzed enantioselective (3 + 2) transannulations of 1,2,3-thiadiazoles with P-chiral monodentate phosphines. Phosphorus, Sulfur, and Silicon and the Related Elements 2024, 199 (2), 157-161.


4.  Meng Han , Pingfan Li*.Sulfur-Mediated ipso-Cyclization of 4-(p-Methoxyaryl)alk-1-ynes Leading to 3-Thiospiro[4.5]deca-1,6,9-trien-8-ones. Synlett, 2024, DOI: 10.1055/a-2216-4882



3.  Zhang, Zhiqin.; Wang, Jianwei; Yu, Chengfeng Tan, Jiajing; Du, Hongguang;* Chen, Ning.* Visible-Light-Induced Acylative Pyridylation of Styrenes. Org. Lett. 2024, 26, 4727 – 4732.



2.  Zhang, Kun; Liu, Shiqi; Wang, Leyi.; Liu, Xiangrui; Xu, Jiaxi;* Chen, Ning.* Annuloselectivity of Dibenzoxazepines and Arynes in the Presence of CO2: [2+2] vs [2+2+2] Annulation. ChemistrySelect 2024, 9, e202304458.



1. Jiaxi Xu. Recent Advances in π-Stacking Interaction-Controlled Asymmetric Synthesis. Molecules. 2024, 29, 1454.


2024 Beginning

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22. Jiaxi Xu. Synthesis of 1,2-oxaphosphinane 2-oxides and 1,2-oxaphosphinine 2-oxides: δ-phosphonolactones and δ-phosphinolactones. New J. Chem. 2023, 47, 5441-5469.


21.Jiaxi Xu. Syntheses of 1,2-Oxaphospholane 2-Oxides and 1,2-Oxaphosphole 2-Oxides. ChemistrySelect, 2023, 8, e202300217


20.Jiaxi Xu, Simin Sun. Difluorocarbene in Cycloadditions and Annulations for the Synthesis of gem-Difluorocarbocycles and gem-Difluoroheterocycles. Eur. J. Org. Chem. 2024, 27, e202301031.


19. Jiaxi Xu. Synthesis of medium and large phostams, phostones, and phostines. Beilstein J. Org. Chem. 2023, 19, 687–699.


18.       Jun Dong, Zhanhui Yang. Catalytic One-Pot Reductive Amination of Carboxylic Acids. ChemCatChem 2024, 16 (9), e202301427.




17.  Yang Chen, Meng-Yao Ma, Hongguang Du, Jiaxi Xu, Zhanhui Yang. Late-Stage Two-Step C11–H Arylation of Dibenzooxa/thiazepines. Synthesis 2023, 55 (14), 2195-2205.



16.  Lu Ouyang, Rui Miao, Zhanhui Yang, Renshi Luo. Iridium-catalyzed reductive amination of carboxylic acids. J. Catal. 2023, 418, 283-289.



15.Jiayi Wang, Dongning Sheng, Duo Fu, Jiaxi Xu. Convenient synthesis of N-sulfonyl α-hydroxyamides via DMSO oxidation of N-alk-1-ynylsulfonamides. J. Sulfur Chem. 2023, 44, 505-522.



 

14. Mengyao Zhang, Qiuyue Wu, Jiaxi Xu. Lewis Acid-Mediated Ring Contraction of 2,4-Diaryl-2,3-dihydro-1H-1,5-benzodiazepines: Access to 2-Aryl-1-styrylbenzimidazoles. Helv. Chim. Acta. 2023, 106, e202200143.



13. Yuliang Wei, Simin Sun, Jiaxi Xu. Direct and safe one-pot synthesis of functionalized dimethyl 1-aryl-1,9a-dihydropyrido[2,1-c][1,4]thiazine-1-phosphonates. Tetrahedron Lett. 2023, 120, 154444.

 

12. Simin Sun, Yuliang Wei, Jiaxi Xu. Difluorocarbene-Triggered [1+5] Annulation: Access to Functionalized 1,1-Difluoro-1,9a-dihydropyrido[2,1-c][1,4]thiazine Derivatives. Org. Lett. 2023, 25, 2868–2872.



11. Tong Pan , Pingfan Li.Sulfur-Mediated Formal Allylic C–H Cyclopropanation of α-Methylstyrenes. J. Org. Chem. 2023, 88, 7564 7570.



10. Guo Liu , Pingfan Li.Enantioselective Bromination of Silyl Enol Ethers with Chiral Pentacarboxycyclopentadienyl Bromide. Synlett. 2023 , 34 , 2447 2450.


9.  Chen, Yixin; (2021级本科生) Cheng, Shi, Su, Chongjie, Chen, Ning*, Xu, Jiaxi.* Theoretical mechanistic insights into the electrophilic addition of hydrogen halides to alkynes. Org. Biomol. Chem. 2023, 21, 7194-7208.


8.  Wang, Jing; Wang, Tingting; Du, Hongguang; Chen, Ning;*  Xu, Jiaxi; Yang, Zhanhui.* Accessing para-Alkylphenols via Iridium-Catalyzed Site-Specific Deoxygenation of Alcohols. J. Org. Chem. 2023, 88, 12572–12584.



7.  Liu, Shiqi; Zhang, Kun; Meng, Yutong; Xu, Jiaxi;* Chen, Ning* Aryne and CO2-based formal [2+2 +2] annulation to access tetrahydroisoquinoline-fused benzoxazinones. Org. Biomol. Chem. 2023, 21, 6892–6897.


6. Huo, Haonan; Cheng, Xingdi; Xu, Jiaxi; Lin, Jiaqi;* Chen, Ning; * Lu, Xueguang.* A fluorinated ionizable lipid improves the mRNA delivery efficiency of lipid nanoparticles. J. Mater. Chem. B. 2023, 11, 4171-4180. 



5. Chenxing Wang, Jiaxi Xu, Ning Chen. N1-Methylthiomethylation of (8-Aza)6-Chloropurine with DMSO through the Pummerer Rearrangement. ChemistrySelect. 2023, 8, e202203972.


4. Tingting Wang Rui Miao, Renshi Luo, Jiaxi Xu, and Zhanhui Yang. Furan-2-yl Anions as γ-Oxo/Hydroxyl Acyl Anion Equivalents Enabled by Iridium-Catalyzed Chemoselective Reduction.  Org. Lett. 2023, 25, 25, 4705–4710.


3. Duo Fu, Changmeng Xi, Jiaxi Xu. Demethyl oxidative halogenation of diacyl dimethylsulfonium methylides. Org. Biomol. Chem., 2023,21, 3991-3996.



2. Jiaxi Xu. Synthesis of medium and large phostams, phostones, and phostines. Beilstein J. Org. Chem. 2023, 19, 687–699. 


1. Luyong Li, Jie Hu, Yuqing Fu, Xiaolin Shi, Hongguang Du, Jiaxi Xu, Ning Chen.  Direct Regioselective C-H Cyanation of PurinesMolecules 2023, 28, 914.




2023年                Beginning!!


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   21. Simin Sun, Yuliang Wei, Jiaxi Xu. Microwave-mediated stereocontrolled annulations of diazo(aryl)methyl(diaryl)phosphine oxides with pyridinium 1,4-zwitterionic thiolates. Chem. Common. 2022. DOI: 10.1039/d2cc05483c


  20. Xin Yuan, Zhicheng Fu, Yelong Lei, Jiaxi Xu. [4+2] Annulation of arylmethylphosphonochloridates with dibenzo[b,f][1,4]oxazepines: A practical approach to polycyclic benzo-δ-phosphonolactams. New. J. Chem. 2022. DOI: 10.1039/d2nj05558a


  19. Xin Yuan, Xuan Ke, Jiaxi Xu. [2 + 4] Annulation of Alkyl(phenyl)phosphinic Chlorides with Enones: Stereoselective Synthesis of δ-Phosphinolactones. Org. Lett. 2022. DOI: 10.1039/d2ob02078e


  18 . Duo Fu  and jiaxi Xu. Halide-Promoted Pyridinylation of α-Acylmethylides with 2-Halo-1-methylpyridinium Iodides as Reagents. Org. Biomol. Chem., 2022, Doi:  10.1039/d2ob02078e



 17Simin Sun, Yuliang Wei, and Jiaxi Xu. Visible-Light-Induced [1+5] Annulation of Phosphoryl Diazomethylarenes and Pyridinium 1,4-Zwitterionic Thiolates. Org. Lett. 2022, 24, 32, 6024–6030. Doi: 10.1021/acs.orglett.2c02321

                                                         


    16. Jiayi Wang, Duo Fu & Jiaxi Xu (2022) Microwave-assisted safe and efficient synthesis of α-ketothioesters from acetylenic sulfones and DMSO, Journal of Sulfur Chemistry, DOI: 10.1080/17415993.2022.2137414

      


15.  Tingting Wang, Changmeng Liu, Dong Xu, Jiaxi Xu, Zhanhui Yang. Iridium-Catalyzed and pH-Dependent Reductions of Nitroalkenes to Ketones. Molecules, 2022, 27(22), 7822; https://doi.org/10.3390/molecules27227822

               



14. Cunzhi Chen, Shuyan Fang, Mingwu Yu, Jiaxi Xu and Zhanhui Yang.Catalytic site-specific and regioselective (3 + 2) transannulations between 1,2,3-thiadiazoles and allenoates. Org. Chem. Front., 2022, Accepted Manuscript. DOI: 10.1039/D2QO01662A.

                                       



        13. Ziyang Dong, Meng-Yao Ma, Jiaxi Xu, Zhanhui Yang. Catalytic (3 + 2) umpolung annulations of α-thioacyl carbenes with aryl isothiocyanates. Chem. Common. 2022,58, 7980-7983.



12. Jiaxi Xu. Synthetic strategies for the preparation of γ-phostams: 1,2-azaphospholidine 2-oxides and 1,2-azaphospholine 2-oxides. Beilstein J. Org. Chem. 2022, 18, 889–915. https://doi.org/10.3762/bjoc.18.90

             




11. Jun Dong & Jiaxi Xu. Synthesis of 2,3-dihydro-1,4-benzoxathiine derivatives. Chemistry of Heterocyclic Compounds. 2022, 58, 271–278.


10. Guangyu Zhang, Simin Sun, Shili Hou and Jiaxi Xu. Diverse and chemoselective sigmatropic shift rearrangements of multisubstituted N,O-diarylhydroxylamines. Org. Biomol. Chem., 2022, 20, 5470–5480.


  9. Dongning Sheng and Jiaxi Xu. Theoretical mechanistic insights into the polar hydrohalogenation of olefins. Org. Biomol. Chem., 2022, 20, 4976–4985


8.  Simin Sun, Mengyao Zhang and Jiaxi Xu. Direct synthesis of highly strained bifunctionalized 2H-thiete 1,1-dioxides. Org. Chem. Front., 2022, 9, 3335–3341.


7. Jiaxi Xu. Synthesis of 1,2-Azaphosphinane 2-Oxides and 1,2-Azaphosphinine 2-Oxides: δ-Phosphonolactams and δ-Phosphinolactams. Asian J. Org. Chem. 2022, 11, e202200176.


6. Guangyu Zhang and Jiaxi Xu. A four-step cascade reaction involving O[1,3] sigmatropic shift and Smiles rearrangements as key steps. New J. Chem., 2022, 46, 9322–9330.


5.  Zhicheng Fu, Yelong Lei, Fang Sun and Jiaxi Xu. Electrophilic hydrophosphonylation of aldimines with alkylphosphonochloridates provides access to (E)-alk-1-enylphosphonamidates. Org. Chem. Front., 2022, 9, 2464–2470.


4.  Cunzhi Chen, Shuyan Fang, Ziyang Dong, Jiaxi Xu, and Zhanhui Yang. Catalytic Diastereospecific and Enantioselective (3 + 2) Transannulations of 1,2,3-Thiadiazoles with Strained Norbornene Derivatives. Org. Lett. 2022, 24, 11, 2110–2114.


3. Yelong Lei and Jiaxi Xu. Efficient synthesis of ethyl 2-(oxazolin-2-yl)alkanoates via ethoxycarbonylketene-induced electrophilic ring expansion of aziridines. Beilstein J. Org. Chem. 2022, 18, 70–76.


2.  Qiuyue Wu, Jiaxi Xu.Regio- and stereoselective synthesis of thiazoline derivatives via the thioketene-induced ring expansion of aziridines. Chem. Commun., 2022, 58, 2714–2717.


      1. Qiuyue Wu, Ning Chen, Jiaxi Xu. Chemoselectivity in the Transannulaction of 1,2,3-Thiadiazoles and Alk-2-enenitriles: Specific Synthesis of 3-(Alk-1-enyl)isothiazoles. ChemistrySelect 2022, 7, e202103943. Corrigendum: 10.1002/slct.202200522


  

2022年                Beginning!!


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DOI  

 

2021

       17.  Jun Dong, Duo Fu, Dongning Sheng, Jiayi Wang and Jiaxi Xu. Direct oxidation of N-ynylsulfonamides into N-sulfonyloxoacetamides with DMSO as a nucleophilic oxidant. RSC Adv., 2021, 11, 40243–40252.


      16.  Wenlai Xie, Simin Sun, Jiaxi Xu. Experimental Evidence on the Formation of Highly Strained 6,7-Dihydroazeto[2,1-b]oxazol-3-ium Derivatives as Reactive Intermediates. Helv. Chim. Acta. 2022,105, e2021001.

     15.  Xingyang Fu, Xinyao Li, and Jiaxi Xu. Synthesis of β-Phosphinolactams from Phosphenes and Imines. Org. Lett. 2021, 23, 22, 8733–8737.

    14. Ziyang Dong, Cunzhi Chen, Jing Wang, Jiaxi Xu and Zhanhui Yang. Dual roles of bisphosphines and epoxides: Rh-catalyzed highly chemoselective and diastereoselective (3 + 2) transannulations of 1,2,3-thiadiazoles with cyanoepoxides. Org. Chem. Front., 2021, 8, 6687–6698. 

   13. Tingting Wang, Yang Chen, Ning Chen, Jiaxi Xu and Zhanhui Yang. Iridium-catalyzed highly stereoselective deoxygenation of tertiary cycloalkanols: stereoelectronic insights and synthetic applications. Org. Biomol. Chem., 2021, 19, 9004–9011.


  12. Xingpeng Chen, Yelong Lei, Duo Fu and Jiaxi Xu. Microwave-accelerated and efficient synthesis of structurally diverse N-(2,2-diphenylvinyl)-β-oxoamides. Org. Biomol. Chem., 2021, 19, 7678–7689.


  11. Dong Xu, Yang Chen, Changmeng Liu, Jiaxi Xu and Zhanhui Yang. Iridium-catalyzed highly chemoselective and efficient reduction of nitroalkenes to nitroalkanes in water. Green Chem., 2021, 23, 6050–6058.


 10. Jiaxi Xu. Synthesis of sulfonopeptides. J Pep Sci. 2021; 27:e3331. https://doi.org/10.1002/psc.3331


  9. Jiaxi Xu. Synthetic strategies of phosphonodepsipeptides. Beilstein J. Org. Chem. 2021, 17, 461–484. https://doi.org/10.3762/bjoc.17.41


  8. Duo Fu, Jiayi Wang, Jiaxi Xu. Direct and Efficient Synthesis of Sulfonium Acyl Sulfonylmethylide Ylides from Acetylenic Sulfones and Dimethyl Sulfoxide. SynthesisDOI: 10.1055/a-1541-6271.


  7.  Wenhao Yuan, Wenlai Xie, Jiaxi Xu. Strong acid-catalyzed electrophilic ring expansion of oxetanes and sulfoxonium ylides. Mol. Catal. 2021, 510, 111687. Doi:10.1016/j.mcat.2021.111687.


 6. Zhang GuangyuXu Jiaxi. [3,3] Sigmatropic Shifts and Applications of Hydroxylamine Derivatives[J]. Chin. J. Org. Chem.2021. Doi: 10.6023/cjoc202103022.


  5. Xingpeng Chen, Zhengshuo Huang,  and Jiaxi Xu*. Catalyst-Free Electrophilic Ring Expansion of N-Unprotected Aziridines with α-Oxoketenes to Efficient Access 2-Alkylidene-1,3-Oxazolidines. Adv. Synth. Catal. 2021, 363, 1–12. 


   4. Shaoyu An, Dr. Zhong Zhang, Prof. Dr. Pingfan LiMetal-Free Synthesis of Selenodihydronaphthalenes by Selenoxide-Mediated Electrophilic Cyclization of Alkynes. Eur. J. Org. Chem. 2021, 3059 – 3070.


  3. Duo Fu, Dr. Jun Dong, Jiayi Wang, Prof. Jiaxi XuDirect 1,2-Oxosulfenylation of Acetylenic Sulfones with DMSO. Asian J. Org. Chem. 2021 DOI: 10.1002/ajoc.202100219. 


  2. Qiuyue Wu, Ziyang Dong, Jiaxi Xu* and  Zhanhui Yang* Sulfur-controlled and rhodium-catalyzed formal (3+3) transannulation of thioacyl carbenes with alk-2-enals and mechanistic insights. Org. Biomol. Chem., 2021,19, 3173-3180.


  1. Pingfan Li. Sulfur-Mediated Reactions through Sulfonium Salts and Ylides. Synlett.  2021, 32.  DOI: 10.1055/a-1409-0906.



2021年                Beginning!!


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     21“Methanesulfinylation of benzyl halides with dimethyl sulfoxide”. Duo Fu, Jun Dong, Hongguang Du and Jiaxi Xu*  . J. Org. Chem.  2019, Just Accepted Manuscript • DOI: 10.1021/acs.joc.9b03041.

      

       

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         20. BF3·OEt2-promoted tandem Meinwald rearrangement and nucleophilic substitution of oxiranecarbonitrilesChuangchuang Xu and Jiaxi Xu. Org. Biomol. Chem., 2019,  Accepted Manuscript. DOI: 10.1039/C9OB02428J.

     
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          19“BF3·OEt2-Catalyzed Synthesis of anti-β-(N-Arylamino)-α-hydroxynitriles by Regio- and Diastereospecific Ring Opening of 3-Aryloxirane-2-carbonitriles with Anilines”. Chuangchuang Xu, Yang Lu, Kaini Xu and Jiaxi XuSynthesis, 2019 DOI:10.1055/s-0039-1690243.

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            18. Transition metal-free access to 3,4-dihydro-1,2-oxaphosphinine-2-oxides from phosphonochloridates and chalcones through tandem Michael addition and nucleophilic substitution”. Zhicheng Fu, Simin Sun, Anjian Yang, Fang Sun and Jiaxi Xu*Chem. Commun. 2019,55, 13124-13127 .DOI: 10.1039/C9CC06352H.

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            17. “Regiospecific synthesis of polysubstituted furans with mono- to tricarboxylates from various sulfonium acylmethylides and acetylenic esters”. Jun Dong, Hongguang Du and Jiaxi XuRSC Adv., 2019, 9, 25034 . DOI: 10.1039/c9ra03563j.


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    16. "Synthesis of Functionalized Thietanes via Electrophili Carbenoid-Induced Ring Expansion of Thiiranes with Sulfonium Acylmethylides as Carbene Precursors”. Jun Dong, Hongguang Du, and Jiaxi Xu. J. Org. Chem. 2019, 84, 10724-10739.

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    15.“Safe, Metal-Free, and Direct Synthesis of Dialkyl Acylmethylidenehydrazine-1,1-dicarboxylates from Dimethylsulfoxonium Acylmethylides and DialkylAzodicarboxylates”. Bingnan Zhou, Jun Dong and Jiaxi XuAdvanced Synthesis & Catalysis2019DOI:10.1002/adsc.201900549.


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         14.“Intramolecular Carbene C-H Insertion Reactions of 2-Diazo-2-sulfamoylacetamides”. Chuqiang Que , Peipei Huang , Zhanhui Yang , Ning Chen and Jiaxi XuMolecules201924, 2628; DOI:10.3390/molecules24142628.


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    13.“Synthesis of N-alkylpyridin-4-ones and thiazolo[3,2-a]pyridin-5-ones through Pummerer-type reactions”. Jingjia Huang, Gang Hu, Shaoyu An, Dongding Chen, Minglei Li, and Pingfan LiJ. Org. Chem. Just Accepted Manuscript. DOI: 10.1021/acs.joc.9b01672 .


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    12.Sulfur Mediated Allylic C-H Arylation, Epoxidation and Aziridination”.Hang Luo, Gang Hu, Pingfan LiJ. Org. Chem. Just Accepted Manuscript. DOI: 10.1021/acs.joc.9b01438.   ( Featured Article).

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    11Fluorium-Initiated Dealkylative Cyanation of Thioethers to Thiocyanates”. Yang Chen, Hongyi Qi, Ning Chen, Demin Ren, Jiaxi Xu, and Zhanhui YangJ. Org. Chem., Just Accepted Manuscript . DOI: 10.1021/acs.joc.9b00965.

    原文 (扫描或长按二维码,识别后到原文页面)

         10Enantioselective Protonation of Silyl Enol Ethers Catalyzed by a
    Chiral Pentacarboxycyclopentadiene-Based Brønsted Acid
    ”. Jun Li, Shaoyu An,Chao Yuan, 
    Pingfan LiSynlett. 2019; 30(11): 1317-1320,  DOI: 10.1055/s-0037-1611849.

    原文 (扫描或长按二维码,识别后到原文页面)


    9. Microwave-Assisted CuCl-Catalyzed Three-Component Reactions
    of Alkynes, Aldehydes, and Amino Alcohols
    ”. Xiang LiNing ChenJiaxi XuSynthesis. 2019, 51, A–I,  DOI: 10.1055/s-0037-1611536.

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    8. Cobalt-Catalyzed Cycloisomerization of N,N-Diallylanilines”. Jun Liu, Zhanhui Yang,Minfang Zheng,Hongfei Wu, Ning Chen, Jiaxi XuSynthesis. 2019, 51, A–G,  DOI: 10.1055/s-0037-1611832.

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    7. Rhodium-Catalyzed 1,1-Hydroacylation of Thioacyl Carbenes with Alkynyl Aldehydes and Subsequent Cyclization”. Bingnan Zhou, Qiuyue Wu, Ziyang Dong, Jiaxi Xu  and Zhanhui Yang. Org. Lett., 2019, Accepted Manuscript. DOI: 10.1021/acs.orglett.9b01003.



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        6. “Synthesis of α-Heterosubstituted Ketones through Sulfur Mediated Difunctionalization of Internal Alkynes”. Zhong Zhang, Yuzheng Luo, Hongguang Du, Jiaxi Xu and Pingfan LiChem. Sci.201910, 5156-5161. DOI: 10.1039/C9SC00568D



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     5. “Iridium-catalysed highly selective reduction–elimination of steroidal 4-en-3-ones to 3,5-dienes in water” Jide LiWeiping TangDemin RenJiaxi Xu* and Zhanhui Yang*. Green Chem., 2019, 21, 2088-2094. DOI: 10.1039/C9GC00654K



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      4. “Sulfur-Mediated Electrophilic Cyclizationof Aryl-Substituted Internal Alkynes”. Zhong Zhang , Pan He, Hongguang Du*, Jiaxi Xu* , and Pingfan LiJ. Org. Chem.2019, 84 (7), pp 4517–4524. DOI: 10.1021/acs.joc.9b00136.


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      3. “Nucleophilic Organic Base DABCO-Mediated Chemospecific Meinwald Rearrangement of Terminal Epoxides into Methyl Ketones”. Siqi Li, Yi Shi, Pingfan Li*, and Jiaxi Xu*. J. Org. Chem.2019, 84 (7), pp 4443–4450. DOI: 10.1021/acs.joc.8b03171.




    原文 (扫描或长按二维码,识别后到原文页面)


         343. "Efficient Direct Synthesis of Aziridine‐Containing Chiral Tridentate Ligands by the Iminium‐Mediated Self‐Ring Opening Reaction of Enantiopure Aziridines and Salicylaldehydes." Xingpeng ChenChao LinHongguang DuJiaxi Xu.  Adv. Synth. Catal2019, 361, 1647–1661. DOI: 10.1002/adsc.201801545.


    原文 (扫描或长按二维码,识别后到原文页面)


         342. A Tandem Sulfonylation andKnoevenagel Condensation for the Preparation of Sulfocoumarin-3-carboxylates. Ziyang Dong, Yang Chen, Zhiheng Yang, Zhanhui Yang*, Jiaxi Xu*. Synthesis2019, 51, 1809-1818. DOI: 10.1055/s-0037-1611703


    原文 (扫描或长按二维码,识别后到原文页面)



    2019年                Beginning!!


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    2007 - 2018 published over 150 SCI papers

     2007 北京化工大学

2007 (10篇, SCI 10篇) (SCI 共计143篇)
1.         Cai, Shuzong; Yin, Wei; Ma, Yuan; Liu, Han; Zhao, Yufen; Xu, Jiaxi*. Synthesis and mass spectrometry of 2-hydroxyethyl 1-aryl-1-(N-benzoxycarbonylamino)methylphosphonate monoesters. Phosphorus Sulfur Silicon Relat. Elem. 2007, 182(1), 2533.


2.         Li, Bonan; Wang, Yikai; Du, Da-Ming; Xu, Jiaxi*. Notable and obvious ketene substituent-dependent effect of temperature on the stereoselectivity in the Staudinger reaction. J. Org. Chem. 2007, 72(3), 990–997.


3.         Ma, Linge; Jiao, Peng; Zhang, Qihan; Du, Da-Ming; Xu, Jiaxi* Ligand and substrate pi-stacking interaction controlled enantioselectivity in the asymmetric aziridination. Tetrahedron: Asymmetry 2007, 18(7), 878884.
4.         许家喜. 微波与有机化学反应的选择性.化学进展 2007, 19(5), 700712.


5.         Li, Bonan; Cai, Shuzong; Du, Da-Ming; Xu, Jiaxi*. Synthesis of phosphinopeptides via the Mannich ligation. Org. Lett. 2007, 9(12), 22572260.


6.         Hu, Libo; Zhu, Hui; Du, Da-Ming; Xu, Jiaxi*. Efficient synthesis of taurine and structurally diverse substituted taurines from aziridines. J. Org. Chem. 2007, 72(12), 45434546.


7.         Hu, Libo; Wang, Yikai; Li, Bonan; Du, Da-Ming; Xu, Jiaxi*. Diastereoselectivity in the Staudinger reaction: A useful probe for investigation on nonthermal microwave effects. Tetrahedron 2007, 63(38), 93879392.


8.         李伯男, 梁勇, 焦雷, 胡立博, 杜大明, 许家喜*. 3-(噻吩-2-基)-b-内酰胺的合成及其立体化学. 化学学报, 2007, 65(16), 16491653.


9.         Liu, Han; Xu, Jiaxi; Du, Da-Ming*. Asymmetric Friedel-Crafts alkylation of methoxyfuran with nitroalkenes catalyzed by diphenylamine-tethered bis(oxazoline)-Zn(II) complexes. Org. Lett. 2007, 9(23), 4725–4728.


10.     Wang, Xiao; Du, Juanjuan; Liu, Han; Du, Da-ming; Xu, Jiaxi*. Effect of the borane source on the enantioselectivity in the chiral oxazaborolidine-catalyzed asymmetric borane reduction of ketones. Heterat. Chem. 2007, 18(7), 740–746.


2008 (10篇, SCI 9篇) (SCI 共计152篇)
11.     Wang, Boyuan; Zhang, Wei; Zhang, Leilei; Du, Da-Ming; Liu, Gang; Xu, Jiaxi*. Versatile synthesis of free and N-benzyloxycarbonyl-protected 2,2-disubstituted taurines. Eur. J. Org. Chem. 2008, (2), 350–355.


12.     Zhang, Wei; Wang, Boyuan; Chen, Ning; Du, Da-Ming; Xu, Jiaxi*. Expeditious and practical synthesis of various substituted taurines from amino alcohols. Synthesis 2008, (2), 197–200.


13.     Guo, Qun-Sheng; Du, Da-Ming; Xu, Jiaxi. The development of double axially chiral phosphoric acids and their catalytic transfer hydrogenation of quinolines. Anew. Chem. Int. Ed. 2008, 47(4), 759762.


14.     Du, Juanjuan; Li, Zhiyi; Du, Da-Ming; Xu, Jiaxi*. Unexpected influence and its origin in rationally tuning the electronic effect of catalysts in the asymmetric borane reduction of ketones. J. Mol. Cat. A: Chem. 2008, 284(1-2), 4045.


15.     Zhu, Min; Hu, Libo; Chen, Ning; Du, Da-Ming; Xu, Jiaxi*. Synthesis of NH-aziridines from vicinal amino alcohols via the Wenker reaction: Scope and limitation. Lett. Org. Chem. 2008, 5(3), 212–217.


16.     Sadler, Kristen; Zhang, Ying; Xu, Jiaxi; Yu, Qitao; Tam, James P. Quaternary protein mimetics of gp41 elicit neutralizing antibodies against HIV fusion-active intermediate state. Biopolymers 2008, 90(3), 320329.


17.     Liu, Han; Lu, Shaofeng; Xu, Jiaxi; Du, Da-Ming. Asymmetric Friedel-Crafts alkylation of electron-rich N-heterocycles with nitroalkenes catalyzed by diphenylamine-tethered bis(oxazoline) and bis(thiazoline) ZnII Complexes. Chem. Asian J. 2008, 3(7), 11111121.


18.     宋华付, 许家喜, 卢永军, 金春华, 陈云华. MeO-CBS不对称催化还原苯乙酮的量子化学计算. 计算机与应用化学 2008, 25(6), 707–710.
19.     Liu, Lei; Zhang, Leilei; Liu, Gang; Xu, Jiaxi.* Synthesis of spiro-fused polycyclic β-lactam derivatives. ARKIVOC 2008, (xvi), 318326.
20.     Du, Juanjuan; Li, Zhiyu; Du, Da-Ming; Xu, Jiaxi*. Improving enantioselectivity via rationally tuning electronic effect of catalysts in the organocatalytic asymmetric aldol reaction. ARKIVOC 2008, (xvii), 145156.
2009 (9篇, SCI 7篇) (SCI 共计159篇)
21.     Liang, Yong; Jiao, Lei; Zhang, Shiwei; Yu, Zhixiang*; Xu, Jiaxi.* New insights into the torquoselectivity of the Staudinger reaction. J. Am. Chem. Soc. 2009, 131(4), 15421549.
22.     Xu, Jiaxi. Stereoselectivity in the synthesis of 2-azetidinones from ketenes and imines via the Staudinger reaction. ARKIVOC 2009, (ix), 21–44.
23.     许家喜. 蛋白质的检测方法与乳制品中蛋白含量测定.大学化学 2009, 24(1), 66–69.
24.     Chen, Ning; Xu, Jiaxi.* HCOOH, an inexpensive, convenient, and practical 13C NMR solvent for strong polar amino acids and their derivatives. Lett. Org. Chem. 2009, 6(4), 349–353.
25.     Yu, Hao; Cao, Shengli; Zhang, Leilei; Liu, Gang; Xu, Jiaxi.* Synthesis of α-aliphatic and β-aromatic substituted taurines via the regioselective ammonia ring-opening of thiiranes. Synthesis 2009, (13), 2205–2209.
26.     Chen, Ning; Zhu, Min; Zhang, Wei; Du, Da-Ming; Xu, Jiaxi*. Synthesis of gem-disubstituted taurines by the regioselective ring-opening of 2,2-disubstituted aziridines with sodium bisulfite and sulfite. Amino Acids 2009, 37(2), 309–313.
27.     He, Fengdan; Meng, Fanhua; Song, Xiuqing; Hu, Wenxiang; Xu, Jiaxi. First and convergent synthesis of hybrid sulfonophosphinopeptides. Org. Lett. 2009, 11(17), 39223925.
28.     骊鑫耀, 许家喜. 二级卤代烷亲核取代反应立体选择性差别的解释. 大学化学 2009, 24(5), 66–68, 74.
29.     Chen, Ning; Jia, Weiyi; Xu, Jiaxi. A versatile synthesis of various substituted taurines from vicinal amino alcohols and aziridines. Eur. J. Org. Chem. 2009, (33), 5841–5846.
2010 (4篇, SCI 4篇) (SCI 共计163篇)
30.     Meng, Fanhua; Xu, Jiaxi. Direct synthesis of phosphinopeptides containing C-terminal a-aminoalkylphosphinic acids. Amino Acids 2010, 39(2), 533–538.
31.     Wang, Renchao; Xu, Jiaxi. Selective alkylation of aminophenols. ARKIVOC 2010, (ix), 293–299.
32.     Li, Xinyao; Chen, Ning; Xu, Jiaxi. An improved and mild Wenker synthesis of aziridines. Synthesis 2010, (20), 3423–3428.
33.     Xu, Jiaxi. Influence of the Electronic Effect of Catalysts on the Enantioselectivity: Applicability and Complexity. Curr. Org. Synth. 2010, 7(6), 650–676.
2011 (16篇, SCI 16篇) (SCI 共计175篇)
34.     周婵, 许家喜. 非对称环氧乙烷的区域选择性亲核开环反应. 化学进展 2011, 23(1), 174–189.
35.     Li, Xinyao; Xu, Jiaxi. Theoretical calculational investigation on the regioselectivity of the ring opening of thiiranes with ammonia and amines. Tetrahedron 2011, 67(9), 1681–1688.
36.     Qi, Hengzhen; Yang, Zhanhui; Xu, Jiaxi. Synthesis of 3-alkoxy/aryloxy-b-lactams with diazoacetate esters as ketene precursors under photoirradiation. Synthesis 2011, (5), 723–730.
37.     Qi, Hengzhen; Zhang, Jiantao; Xu, Jiaxi. Expeditious synthesis of 2,3,6-trisubstituted 2H-1,3-oxazin-4(3H)-ones via the tertiary amine-induced reaction of 2-diazo-3-oxoalkanals and imines under mild condition. Synthesis 2011, (6), 887894.
38.     Li, Xinyao; Xu, Jiaxi. Abundant intramolecular ring rearrangements of 1-(N-benzyloxycarbonylamino)arylmethylphosphonate phenyl monoesters under electrospray ionization conditions. Phosphorus Sulfur Silicon Relat. Elem. 2011, 186(3), 503510.
39.     Qi, Hengzhen; Li, Xinyao; Xu, Jiaxi. Stereoselective control in the Staudinger reactions involving monosubstituted ketenes with electron acceptor substituents: Experimental investigation and theoretical rationalization. Org. Biomol. Chem. 2011, 9(8), 27022714.
40.     Xu, Chuanxiang; Xu, Jiaxi. Versatile synthesis of a-substituted taurines from nitroolefins. Amino Acids 2011, 41(1), 195–203.
41.     Liu, Guocheng; Xu, Jiaxi; Park, Ki Chul; Chen, Ning; Zhang, Si; Ding, Zhongren; Wang, Feng; Du, Hongguang. Novel synthesis approach and antiplatelet-activity evaluation of 6-alkylamino-2,4-dialkyl(aryl)thiopyrimidines. Tetrahedron 2011, 67(29), 5156–5161.
42.     Yu, Hao; Deng, Xiaobing; Cao, Shengli; Xu, Jiaxi. Practical Corey-Chaykovsky epoxidation: Scope and limitation. Lett. Org. Chem. 2011, 8(7), 509–514.
43.     Deng, Xiaobing; Chen, Ning; Wang, Zhixin; Li, Xinyao; Hu, Hongyan; Xu, Jiaxi. A convenient synthesis of thiazolidin-2-ones from thiazolidine-2-thiones: Antibiotic activity and revisiting the mechanism. Phosphorus Sulfur Silicon Relat. Elem. 2011, 186(7), 15631571.
44.     Li, Xinyao; Xu, Jiaxi. Theoretical insights into the metal-free and formal [2+2+2] cycloaddition strategy via intramolecular cascade propargylic ene/Diels-Alder reactions with tautomerization. Org. Biomol. Chem. 2011, 9(17), 5997–6003.
45.     Chen, Ning; Huang, Zhongyan; Zhou, Chan; Xu, Jiaxi. Thorpe-Ingold effect in the reaction of vicinal amino primary alcohol hydrogen sulfates and carbon disulfide. Tetrahedron 2011, 67(41), 7971–7976.
46.     Liu, Jing; Hou, Shili; Xu, Jiaxi. Diverse reactions of sulfonyl chlorides and cyclic imines. Phosphorus Sulfur Silicon Relat. Elem. 2011, 186(12), 23772391.
47.     Wang, Zhixin; Chen, Ning; Xu, Jiaxi. Selectivities in the reaction of vicinal diimines and acyl chlorides. Tetrahedron 2011, 67(50), 9690–9699.
48.     Wang, Zhixin; Xu, Jiaxi. Stereospecific synthesis of cis- and trans-4-acyl-b-lactams from vicinal diketones and ketoaldehydes. Sci China Chem. 2011, 54(11), 1711–1717.
49.     Qi, Hengzhen; Mo, Shanyan; Xu, Jiaxi. Highly stereoselective synthesis of trans-3-chloro-b-lactams from imines and mixed chloro- and nitroacetyl chlorides. Chem. Res. Chin. Univ. 2011, 27(6), 958–962.
50.     许家喜 取代牛磺酸的合成研究进展. 化学试剂 2011, 33(11), 961-965.
2012 (14篇, SCI 14篇) (SCI 共计189篇)
51.     Yang, Zhanhui; Xu, Jiaxi. Remarkable ketene substituent-dependent effect of photo irradiation on the diastereoselectivity in the Staudinger reaction. Tetrahedron Lett. 2012, 53(7), 786–789.
52.     Chen, Ning; Xu, Jiaxi. Facile synthesis of various substituted taurines, especially syn- and anti-1,2-disubstituted taurines, from nitroolefins. Tetrahedron 2012, 68(11), 2513–2522.
53.     周婵,许家喜 非对称环硫乙烷的区域选择性亲核开环反应. 化学进展, 2012, 24(2/3), 338–347.
54.     Liu, Guocheng; Xu, Jiaxi; Yu, Mingwu; Chen, Ning; Zhang, Si; Ding, Zhongren; Du, Hongguang. New approch to synthesize symmetric and unsymmetric 6-(N-alkyl(aryl)amino)- and 6-(N,N-dialkyl(aryl)amino)-2,4-bis(alkyl(aryl)thio)pyrimidines as antiplatelet agents. Phosphorus Sulfur Silicon Relat. Elem. 2012, 187(5), 650659.
55.     Liu, Guocheng; Xu, Jiaxi; Chen, Ning; Zhang, Si; Ding, Zhongren; Du, Hongguang. Synthesis of N6-alkyl(aryl)-2-alkyl(aryl)thioadenosines as antiplatelet agents. Eur. J. Med. Chem. 2012, 53, 114–123.
56.     Meng, Fanhua; He, Fengdan; Song, Xiuqing; Zhang, Leilei; Hu, Wenxiang; Liu, Gang; Xu, Jiaxi. Facile synthesis of hybrid sulfonophosphinodipeptides composing of taurines and 1-aminoalkylphosphinic acids. Amino Acids 2012, 43(1), 423–429.
57.     Ma, Yunhai; Xu, Jiaxi. Synthesis of homotaurine and 1-substituted homotaurines from a,b-unsaturated nitriles. Synthesis 2012, 44(14), 2225–2230.
58.     Mo, Shanyan; Xu, Jiaxi. Mechanistic investigation of the ring opening in the Staudinger cycloaddition involving ketenes with electron-withdrawing substituents. Helv. Chim. Acta. 2012, 95(7), 1079–1087.
59.     Lv, Xueguang; Xu, Jiaxi. Negative ion mass spectral fragmentation of N-alkoxycarbonyl-1-aminoarylmethylphosphonic monoesters under electrospray ionization conditions. Phosphorus Sulfur Silicon Relat. Elem. 2012, 187(10), 11511160.
60.     Zhou, Yang; Li, Xinyao; Hou, Shili, Xu, Jiaxi.* Facile synthesis of dihydrochalcones via the AlCl3-promoted tandem Friedel-Crafts acylation and alkylation of arenes and 2-alkenoyl chlorides. J. Mol. Catal. A: Chem. 2012, 365, 203–211.
61.     Xu, Jiaxi. Synthesis of b-lactams with p electron-withdrawing substituents. Tetrahedron 2012, 68(52), 10696–10747.
62.     Hou, Shili; Li, Xinyao, Xu, Jiaxi. Mechanistic insight into the formal [1,3]-migration in the thermal Claisen rearrangement. J. Org. Chem. 2012, 77(23), 10856–10869.
63.     Meng, Fanhua; Chen, Ning; Xu, Jiaxi. An efficient and facile synthesis of N-Cbz-b-aminoalkanesulfonamides. Sci China Chem. 2012, 55(12), 2548–2553.
64.     Li, C; Duan, S; Xu, J; Qiao, R; Xu, P; Zhao, Y. Modulation of ascorbic acid-induced DNA cleavage by polyamide: Cleavage manner, kinetics and mechanism. Curr. Med. Chem. 2012, 19(6), 921–926.
2013 (22篇, SCI 17篇) (SCI 共计206篇)
65.     Kakaei, Saeed; Chen, Ning; Xu, Jiaxi.* Expeditious synthesis of 1-substituted taurines with diverse functionalized side-chains. Tetrahedron 2013, 69(1), 302–309.
66.     Huang, Zhongyan; Xu, Jiaxi. Efficient synthesis of N-protected 1-substituted homotaurines from a xanthate and olefins. Tetrahedron 2013, 69(3), 1050–1056.
67.     Li, Xinyao; Xu, Jiaxi.* Annuloselectivity in cycloadditions of ketenes with imines: A DFT study. J. Org. Chem. 2013, 78(2), 347–355.
68.     Li, Xinyao; Yang, Zuoyin; Xu, Jiaxi.* Comprehensive theoretical investigation on regioselectivity in the nucleophilic ring opening of epoxides. Curr. Org. Synth. 2013, 10(1), 169177.
69.     Hou, Shili, Li, Xinyao; Xu, Jiaxi.* Theoretical studies on selectivities in the Staudinger reaction of vicinal diimines and ketenes. Sci China Chem. 2013, 56(3), 370–379.
70.     Li, Xinyao; Xu, Jiaxi.* DFT and experimental exploration of intramolecular [2+2+2] cycloaddition of oxanorbornadienedicarboxylates and anologs. J. Org. Chem. 2013, 78(7), 3039–3047.
71.     侯士立, 许家喜. 二烷基苯基不饱和羧酸钠盐双尾表面活性剂的合成及性能研究. 化学试剂, 2013, 35(4), 345–348.
72.     Meng, Fanhua; Xu, Jiaxi.* Synthesis of phosphinodepsipeptides via the pseudo-four-component condensation reaction. Tetrahedron 2013, 69(24), 4944–4952.
73.     Li, Xinyao; Xu, Jiaxi.* Theoretical insights into the [4 + 2]/retro [4 + 2] cycloaddition approach to synthesis of biaryls and polycyclic aromatics. Sci China Chem. 2013, 56(5), 633–640.
74.     Zhou, Chan; Xu, Jiaxi. Application of bisamide ligands in asymmetric catalysis. Curr. Org. Synth. 2013, 10(3), 394410.
75.     Yang, Zhanhui; Xu, Jiaxi.* Convenient and environment-friendly synthesis of sulfonyl chlorides from S-alkylisothiourea salts via the N-chlorosuccinimide chlorosulfonation. Synthesis 2013, 45(12), 1675–1682.
76.     许家喜. 芳基离子和芳基自由基与环己二烯离子和环己二烯自由基的区别. 大学化学, 2013, 28(3), 77–81.
77.     Nai, Youfeng; Xu, Jiaxi. Synthesis of substituted homotaurines from 2-alkenamides. Helv. Chim. Acta. 2013, 96(7), 1355–1365.
78.     许家喜. 膦酰肽和膦酰酯肽的汇聚式合成. 中国科学 化学, 2013, 43(8), 995-1004.
79.     Kakaei, Saeed; Xu, Jiaxi. Synthesis of (2-alkylthiothiazolin-5-yl)methyl dodecanoates via tandem radical reaction. Org. Biomol. Chem. 2013, 11(33), 5481–5490.
80.     Huang, Zhongyan; Xu, Jiaxi. One-pot synthesis of symmetric 1,7-dicarbonyl compounds via a tandem radical addition-elimination-addition reaction. RSC Adv. 2013, 3(35), 15114–15120.
81.     Kakaei, Saeed; Xu, Jiaxi. Efficient synthesis of protected sulfonopeptides from N-protected 2-aminoalkyl xanthates and thioacetates. Tetrahedron 2013, 69(43), 995–9075.
82.     Zhang, Jiantao; Xu, Jiaxi. Chemoselectivity in the reaction of 2-diazo-3-oxo-3-phenylpropanal with aldehydes and ketones. Helv. Chim. Acta. 2013, 96(9), 1733–1779.
83.     Yang, Zhanhui; Zheng, Yongpeng; Xu, Jiaxi. Simple synthesis of sulfonyl chlorides from thiol precursors and derivatives by NaClO2-mediated oxidative chlorosulfonation. Synlett 2013, 24(16), 2165–2169.
84.     Huang, Zhongyan; Xu, Jiaxi. Efficient synthesis of 5-substituted thiazolidin-2-ones from xanthates and tert-butyl N-allylcarbamates. Tetrahedron 2013, 69(48), 10272–10278.
85.     陈宁, 侯士立, 许家喜. 联苯胺重排在有机合成中的应用. 中国科技论文, 2013, 8(9), 851–855.
86.     许家喜. 联苯胺重排的反应机理. 大学化学, 2013, 28(5), 34–39.
2014 (18篇, SCI 18篇) (SCI 共计224篇)
87.     Yang, Zhanhui; Zhou, Bingnan; Xu, Jiaxi.* Clean and economic synthesis of alkanesulfonyl chlorides from S-alkyl isothiourea salts via Bleach oxidative chlorosulfonation. Synthesis 2014, 46(2), 225–229.
88.     Yang, Zhanhui; Xu, Jiaxi.* Preparation of alkanesulfonyl chlorides from S-alkyl isothiourea salts via N-chlorosuccinimide mediated oxidative chlorosulfonation. Org. Synth. 2014, 91, 116–124.
89.     Yang, Zhanhui; Xu, Jiaxi.* Synthesis of benzo-γ-sultams via the Rh-catalyzed aromatic C-H functionalization of diazosulfonamides. Chem. Commun. 2014, 50(27), 3616–3618.
90.     Kheira, Haiouani; Li, Pingfan; Xu, Jiaxi.* Synthesis of indenes via aluminum chloride-promoted tandem Friedel-Crafts alkylation of arenes and cinnamaldehydes. J. Mol. Catal. A: Chem. 2014, 391, 168–174.
91.     Abdellaoui, Hassane; Xu, Jiaxi. Versatile synthesis of 4-spiro-β-lactam-3-carbonitriles via the intramolecular nucleophilic cyclization of N-(p-hydroxyphenyl)cyanoacetamides. Tetrahedron 2014, 70(29), 4323–4330.
92.     Mo, Shanyan; Huang, Peipei; Xu, Jiaxi. Cascade nitrosation and addition-elimination of 2-nitroacetanilides for highly efficient synthesis of 1,4,2,5-dioxadiazine derivatives. Org. Biomol. Chem. 2014, 12(24), 4192–4200.
93.     Mo, Shanyan; Xu, Jiaxi. Chemospecific intramolecular Büchner reaction catalyzed by copper(II) acetylacetonate. ChemCatChem 2014, 6(6), 1679–1683.
94.     Mo, Shanyan; Yang, Zhanhui; Xu, Jiaxi. Aqueous copper nitrate catalyzed synthesis of 3-alkylideneoxindoles from α-diazo-β-ketoanilides. Eur. J. Org. Chem. 2014, (18), 3923–3929.
95.     Hou, Shili; Li, Xinyao; Xu, Jiaxi. N[1,3]-Sigmatropic shift in the benzidine rearrangement: Experimental and theoretical investigation. Org. Biomol. Chem. 2014, 12(27), 4952–4963.
96.     Zheng, Yongpeng; Xu, Jiaxi. Synthesis of enantiopure free and N-benzyloxycarbonyl-protected 3-substituted homotaurines from naturally occurring amino acids. Tetrahedron 2014, 70(34), 5197–5206.
97.     郑勇鹏, 许家喜. Thorpe-Ingold效应及其在有机成环反应中的应用. 化学进展, 2014, 26(9), 1471–1491.
98.     Mo, Shanyan; Li, Xinhao; Xu, Jiaxi. In situ generated iodonium ylides as safe carbene precursors for the chemoselective intramolecular Buchner reaction. J. Org. Chem. 2014, 79(19), 9186–9195.
99.     Yang, Zhanhui; Son, Kwon-Il; Li, Siqi; Zhou, Bingnan; Xu, Jiaxi. Specific 1,2-hydride shift in the boron trifluoride-catalyzed reactions of aromatic aldehydes with diazoacetonitrile: Simple synthesis of β-ketonitriles. Eur. J. Org. Chem. 2014, (29), 6380–6384.
100.  Zhou, Chan; Xu, Jiaxi. Synthesis of new C2-symmetric chiral bisamides from (S,S)-1,2-cyclohexanedicarboxylic acid. Helv. Chim. Acta. 2014, 97(10), 1396–1405.
101.  Yang, Zhanhui; Xu, Jiaxi.* Insights on β-sultam ring formation in the sulfa-Staudinger reactions. J. Org. Chem. 2014, 79(21), 10703–10708.
102.  Yang, Zhanhui; Li, Siqi; Zhang, Zhong; Xu, Jiaxi. Base-switched annuloselectivity in the reactions of ethyl malonyl chloride and imines. Org. Biomol. Chem. 2014, 12(48), 9822–9830.
103.  Hu, Gang; Xu, Jiaxi; Li, Pingfan. Sulfur mediated allylic C-H alkylation of tri- and disubstituted olefins. Org. Lett. 2014, 16(22), 6036–6039.
104.  Wang, Renchao; Xu, Jiaxi. Enantioselective sulfur-Michael addition of thioacetic acid to nitroalkenes catalyzed by bifunctional amine-thiourea catalysts. Helv. Chim. Acta. 2014, 97(12), 1700–1707.
2015 (11篇, SCI 11篇) (SCI 共计235篇)
105.  Chen, Ning; Du, Hongguang; Liu, Weidong; Wang, Shanshan; Li, Xinyao; Xu, Jiaxi. Synthesis and fungicidal activity of simple structural 1,3-thiazolidine-2-thione derivatives. Phosphorus Sulfur Silicon Relat. Elem. 2015, 190(1), 111.
106.  Wang, Renchao; Liu, Jing; Xu, Jiaxi. Organocatalytic enantioselective sulfur-Michael addition of thioacetic acid to arylmethylidenemalonates. Adv. Synth. Catal. 2015, 357(1), 159–167.
107.  Zhong, Xin; Chen, Ning; Li, Pingfan; Xu, Jiaxi. A mild radical method for the dimerization of dithiocarbamates. Eur. J. Org. Chem. 2015, (4), 802–809.
108.  Du, Hongguang; He, Qiwen; Chen, Ning; Xu, Jiaxi; Chen, Fei; Liu, Guochen. Proton NMR investigations of 6-alkylamino-2-alkylthioadenosine derivatives. Magn. Reson. Chem. 2015, 53(3), 218–222.
109.  Yang, Zhanhui; Chen, Ning; Xu, Jiaxi.* Substituent-controlled annuloselectivity and stereoselectivity in the sulfa-Staudinger cycloadditions. J. Org. Chem. 2015, 80(7), 3611–3620.
110.  Yang, Zhanhui; Xu, Jiaxi. Substituent effect on the diastereoselectivity in the sulfa-Staudinger cycloaddition. Tetrahedron 2015, 71(19), 2844–2852.
111.  Sun, Biyun; Xu, Jiaxi. Convenient and facile synthesis of hybrid sulfonophosphonodipeptides. Synthesis 2015, 47(10), 1479–1487.
112.  Wang, Jiandong; Chen, Ning; Xu, Jiaxi. Diastereoselectivity in the triethylamine-catalyzed sulfa-Michael addition of thiols to nitroalkenes: Kinetic and thermodynamic control. Tetrahedron 2015, 71(23), 4007–4014.
113.  Sun, Biyun; Xu, Jiaxi. Convenient synthesis of phosphonodipeptides containing C-terminal a-aminoalkylphosphonic acids. J. Pept. Sci. 2015, 21(7), 615–619.
114.  Li, Xinyao; Jin, Xin; Xu, Jiaxi.* Annuloselectivity in reactions of diacyl dichlorides and imines: Combined experimental and theoretical studies. J. Org. Chem. 2015, 80(14), 6976–6985.
115.  Yang, Zhanhui; Xu, Jiaxi. Annuloselectivity and stereochemistry in the sulfa-Staudinger cycloadditions of cyclic imines. RSC Adv. 2015, 5(96), 78396–78405.
2016 (19篇, SCI 17篇) (SCI 共计242篇)
116.  Xu, Wei; Xu, Jiaxi. Regioselectivity in the ring opening and expansion of unsymmetric thietanes. Curr. Org. Synth. 2016, 13(1), 73–81.
117.  Wang, Jiandong; Li, Pingfan; Yang, Zhanhui; Chen, Ning; Xu, Jiaxi. Insights into the diastereoselective control in the sulfa-Michael addition of thiols to nitroalkenes: Stereoelectronic effect in the cyclic chelated transition state. Tetrahedron 2016, 72(3), 370–378.
118.  Gao, Simiao; Zhang, Yu; Dong, Jun; Chen, Ning; Xu, Jiaxi. Synthesis of functionalized 5-substituted thiazolidine-2-thiones via adscititious xanthates-promoted radical cyclization of allyl(alkyl/aryl)dithiocarbamates. Org. Biomol. Chem. 2016, 14(3), 1002–1012.
119.  Yang, Zhanhui; Hou, Shili; He, Wei, Cheng, Baoxiang; Jiao, Peng; Xu, Jiaxi. Regioselectivity in ortho- and para-semidine and diphenyline rearrangements. Tetrahedron 2016, 72(17), 2186–2195.
120.  Yang, Zhanhui; Xu, Wei; Wu, Qiuyue; Xu, Jiaxi. Aminoxidation of thiols to N-chloro-N-sulfonyl sulfinamides. J. Org. Chem. 2016, 81(7), 3051–3057.
121.  Zhou, Bingnan; Xu, Jiaxi. Tertiary amine-catalyzed and direct synthesis of a-chloroalkanesulfonylhydrazines from azodicarboxylates and sulfonyl chlorides. Org. Biomol. Chem. 2016, 14(21), 4918–4926.
122.  Mo, Shanyan; Xu, Chuangchuang; Xu, Jiaxi. Expeditious and convenient synthesis of polycyclic difluoroboron complexes of 2-oxoindoline-3-carboxamides by tandem reaction. Adv. Synth. Catal. 2016, 358(11), 1767–1777.
123.  Yang, Zhanhui; He, Wei; Cheng, Baoxiang; Xu, Jiaxi. Stereochemistry and mechanistic insight in the [2k+2i+2i] annulations of ketenes and imines. J. Org. Chem. 2016, 81(11), 4506–4515.
124.  王建东, 许家喜. 含邻手性碳原子双键亲电加成反应的立体选择性模型. 化学进展 2016, 28(6), 784–800.
125.  Huang, Peipei; Jiaxi Xu. Synthesis of 2-oxophosphorindolines via the copper-catalyzed intramolecular aromatic C-H insertion of diazophosphonamidates. RSC Adv. 2016, 6(68), 63736–63748.
126.  Wu, Qiuyue; Yang, Zhanhui; Xu, Jiaxi. Temperature-dependent annuloselectivity and stereochemistry in the reactions of methanesulfonyl sulfene with imines. Org. Biomol. Chem. 2016, 14(30), 7258–7267.
127.  Li, Xinhao; Xu, Jiaxi. Determination on temperature gradient of different polar reactants in reaction mixture under microwave irradiation with molecular probe. Tetrahedron 2016, 72(35), 5515–5520.
128.  Wang, Jiandong; Son, Kwon-Il; Xu, Jiaxi. Thermal 1,3- and 1,5-sulfonyl migrations of N-arenesulfonylphenothiazines and N-arenesulfonylphenoxazines. Monatsh. Chem. 2016, 147(9), 1637–1649.
129.  Zhong, Xin; Chen, Ning; Xu, Jiaxi. Mass spectral fragmentation of bis(1-arylimino-1-alkyl/arylthiomethyl) disulfides under positive electrospray ionization conditions. Phosphorus Sulfur Silicon Relat. Elem. 2016, 191(9), 1235–1239.
130.  Mo, Shanyan; Tu, Jianzhuo; Xu, Jiaxi. Chemospecific synthesis of 2-acetoxyindole-3-carbonitriles catalyzed by Cu(acac)2. Russ. Chem. Bull. 2016, 65(7), 1773–1778.
131.  许薇, 许家喜. 几种经典有机反应的分子轨道描述. 大学化学 2016, 31(8), 60–65.
132.  许薇, 张丽丹, 许家喜. 烷基异硫脲盐环保合成磺酰氯研究进展.化学试剂 2016, 31(10), 60–65.
133.  Zhang, Zhong; Du, Hongguang; Xu, Jiaxi; Li, Pingfan. Anti-Markovnikov rearrangement in sulfur mediated allylic C–H amination of olefins. Chem. Commun. 2016, 52(77), 11547–11550.
134.  李思琦, 许家喜. 非对称氧杂环丁烷的选择性开环. 化学进展 2016, 28(12), 1798–1810.
2017 (19篇, SCI 19篇) (SCI 共计261篇)
135.  Dong, Jun; Xu, Jiaxi. Facile synthesis of thietanes via ring expansion of thiiranes. Org. Biomol. Chem. 2017, 15(4), 836–844.
136.  Zhou, Bingnan; Yang, Xiao; Xu, Jiaxi. Synthesis of sulfonylhydrazine-1,2-dicarboxylates from thiols and dialkyl azodicarboxylates. Synthesis 2017, 49(7), 1632–1640.
137.  Chen, Xingpeng; Xu, Jiaxi. Synthesis of 3-acyl-5,6-dihydro-1,4-oxathiines through ring expansion of thiiranes. Tetrahedron Lett. 2017, 58(16), 1651–1654.
138.  Xu, Jiaxi. Diversity and chemoselectivity in the acid-catalyzed rearrangements of N,N’-diarylhydrazines. Curr. Org. Synth. 2017, 14(4), 511–530.
139.  陈兴鹏,许家喜. 非对称氮杂环丁烷的区域选择性开环反应. 化学进展 2017, 29(2/3), 181–197.
140.  Jiang, Jianhui; Xu, Jiaxi. Expeditious synthesis of dianionic-headed 4-sulfoalkanoic acid surfactants. Molecules 2017, 22(4), 640.
141.  Cheng, Baoxiang; Xu, Jiaxi. Mechanistic insight into the thermal 1,3-chlorine migrations of N-chloroacetanilides under neutral conditions. Phosphorus Sulfur Silicon Relat. Elem. 2017, 192(5), 518–525.
142.  Abdellaoui, Hassane; Chen, Xingpeng; Xu, Jiaxi. Efficient synthesis of N-benzyloxycarbonyl-2-aminoalkanesulfonyl chlorides with functionalized side-chains. Synthesis 2017, 49(10), 2250–2256.
143.  Yang, Zhanhui; Yang, Shiyi; Xu, Jiaxi. Sulfur-directed metal-free and regiospecific methyl C(sp3)-H imidation of thioanisoles. Tetrahedron 2017, 73(23), 3240–3248.
144.  Huang, Peipei; Yang, Zhanhui; Xu, Jiaxi. Specific intramolecular aromatic C-H insertion of diazosulfonamides. Tetrahedron 2017, 73(23), 3255–3265.
145.  Yang, Zhanhui; Abdellaoui, Hassane; Xu, Jiaxi. Ortho-nitro effect on the diastereoselective control in sulfa-Staudinger and Staudinger cycloadditions. Molecules 2017, 22(5), 784.
146.  Yang, Zhanhui; Yang, Shiyi; Haroone, Muhammad Sohail; He, Wei; Xu, Jiaxi. Sulfur-mediated C(sp2)-H imidation and 1,2-imidofluorination of vinyl sulfides. Tetrahedron 2017, 73(24), 3338–3346.
147.  Li, Xinhao; Xu, Jiaxi. Effects of the microwave power on the microwave assisted esterification. Curr. Microw. Chem. 2017, 4(2), 158–162.
148.  Tian, Miao; Yu, Mingwu; Shi, Tingting, Hu, Junbin; Li, Shunlai; Xu, Jiaxi; Chen, Ning; Du, Hongguang. Silver catalyzed direct C6-H arylation of purines and purine nucleosides with arylboronic acid. Eur. J. Org. Chem. 2017, (24), 3415–3420.
149.  He, Wei; Yang, Zhanhui; Xu, Jiaxi. Sterically controlled diastereoselectivity in the thio-Staudinger cycloaddition involving alkyl/alkenyl/aryl thioketenes. Org. Biomol. Chem. 2017, 15(26), 5541–5548.
150.  Liu, Jing; Tu, Jianzhuo; Yang, Zhanhui; Pak, Chol-Ung; Xu, Jiaxi. Improved Buchner reaction selectivity in the copper-catalyzed reactions of ethyl 3-arylmethylamino-2-diazo-3-oxopropanoates. Tetrahedron 2017, 73(31), 4616–4626.
151.  Xu, Chuangchuang; Xu, Jiaxi. An expeditious method to synthesize difluoroboron complexes of β-keto amides from β-ketonitriles and BF3.OEt2. Org. Biomol. Chem. 2017, 15(30), 6375–6383.
152.  He, Wei; Zhuang, Junpeng; Du, Hongguang; Yang, Zhanhui; Xu, Jiaxi. Stereochemistry and mechanistic insights in the [2t + 2i + 2i] annulations of thioketenes and imines. Org. Biomol. Chem. 2017, 15(44), 9424–9432.
153.  Li, Xinhao; Xu, Jiaxi. Identification of microwave selective heating effort in an intermolecular reaction with Hammett linear relationship as a molecular level probe. Curr. Microw. Chem. 2017, 4(4), 339–346.
2018 (16篇, SCI 16篇) (SCI 共计277篇)
154.  阙楚强, 陈宁, 许家喜. 氨基甲酸酯在C-H键活化中的应用, 化学进展, 2018, 30(2/3), 139–155.
155.  He, Wei; Ding, Yong; Tu, Jianzhuo; Que, Chuqiang; Yang, Zhanhui; Xu, Jiaxi. Thermal conversion of primary O-alkyl S-difluoroalkyl xanthates to disulfides: an extension to Chugaev elimination. Org. Biomol. Chem. 2018, 16(10), 1659–1666.
156.  Li, Siqi; Chen, Xingpeng; Xu, Jiaxi. Microwave-assisted copper-catalyzed stereoselective ring expansions of three-membered heterocycles with α-diazo-β-dicarbonyl compounds. Tetrahedron 2018, 74(14), 1613–1620.
157.  Xu, Wei; Fu, Zhicheng; Yang, Zhanhui; Zhang, Lidan; Xu, Jiaxi. Synthesis of 4-trifluoromethyl-β-sultams via sulfa-Staudinger cycloaddition. Phosphorus Sulfur Silicon Relat. Elem. 2018, 193(5), 335–344.
158.  Kheira, Haiouani; Chen, Xingpeng; Xu, Jiaxi. Expeditious preparation of N-[(9H-fluoren-9-ylmethoxy)carbonyl]-2-aminoethanesulfonyl chlorides with functionalized 1-substituents. Curr. Org. Synth. 2018, 15(2), 246–255.
159.  Liu, Jitian; Yang, Shiyi; Tang, Weiping; Yang, Zhanhui; Xu, Jiaxi. Iridium-catalyzed efficient reduction of ketones in water with formic acid as hydride donor at low catalyst loading. Green Chem. 2018, 20(9), 2118–2124.
160.  Dong, Jun; Xu, Jiaxi. NBS/DMSO-Mediated synthesis of (2,3-dihydrobenzo[b][1,4]oxathiin-3-yl)methanols from aryloxymethylthiiranes. New J. Chem. 2018, 42(11), 9037–9044.
161.  Dong, Jun; Xu, Jiaxi. Synthesis of alkenyl aryl sulfides and their sulfoxides from thiiranes and diaryliodoniums. Synthesis 2018, 50(12), 2407–2415.
162.  Gang Hu, Jiaxi Xu, Pingfan Li. Synthesis of N-alkylated 2-pyridones through Pummerer type reactions of activated sulfoxides and 2-fluoropyridine. Org. Biomol. Chem. 2018, 16(22), 4151–4158.
163.  Gang Hu, Jiaxi Xu, Pingfan Li. Sulfur mediated propargylic C−H alkylation of alkynes. Org. Chem. Front. 2018, 5(14), 2167–2170.
164.  Zhong, Xin; Chen, Ning; Xu, Jiaxi. A concise synthesis of cyclobrassinin and its analogues via thiyl radical aromatic substitution. New J. Chem. 2018, 42(16), 13549–13557.
165.  符志成,许家喜. 氮杂环丁烷的合成. 化学进展 2018, 30(8), 1047–1066.
166.  Yang, Shiyi; Tang, Weiping; Yang, Zhanhui; Xu, Jiaxi. Iridium-catalyzed highly efficient and site-selective deoxygenation of alcohols. ACS Catal20188(10), 9320–9326.
167.  Fu, Zhicheng; Yuan, Wenhao; Chen, Ning; Yang, Zhanhui; Xu, Jiaxi. Na2S2O8-mediated efficient synthesis of isothiocyanates from primary amines in water. Green Chem. 2018, 20(19), 4484–4491.
168.  Xu, Chuangchuang; Xu, Jiaxi. Oxygenophilic Lewis acid-promoted synthesis of 2-arylindoles from anilines and cyanoepoxides in alcohol. J. Org. Chem. 2018, 83(23), 14733–14742.
169.  Yang, Dongqiang; Xu, Jiaxi. Influence of the product polarity on temperature profiles in the microwave-assisted Claisen rearrangement. Curr. Microw. Chem. 2018, 5(2), 120–127.




    1992 - 2007 北京大学 (published over 150 SCI papers


    1991 (1)

    1.         宋艳玲, 许家喜, 胡京诞, 金声*. N-(4-对氟苯基-4-芳胺基)-丁基-N’-二苯基哌嗪及其衍生物的合成. 北京大学学报(自然科学版) 1991, 27(6), 695699.

    1992 (1)

    2.         Xu, Jiaxi; Jin, Sheng*. New heterocyclic system synthesis IV: 4a,5,6,12-Tetrahydro-1H-1,3-oxazino[3,2-d][1,5]benzothiazepine-1-one. Chin. Chem. Lett. 1992, 3(3), 181182.

    1993 (3)

    3.         Xu, Jiaxi; Jin, Sheng*. The study on the water soluble peptides in Papaver Somniferum pollen: Extraction, purification, sequence determination and synthesis. Chin. Chem. Lett. 1993, 4(3), 213214.

    4.         Jin, Sheng*; Xu, Jiaxi; Miao, Ping. Studies on the peptides and polysaccharides in pollen. 有机化学(Youji Huaxue) 1993, 13, 202205.

    5.         贺晓然, 林孝元*, 何美玉, 俞振培, 许家喜. 噁嗪酮并苯并硫氮杂卓衍生物在质谱中的Retro Diels-Alder碎裂反应. 质谱学报 1993, 14(3), 2630.

    1994 (1)

    6.         Xu, Jiaxi; Jin, Sheng*. New heterocyclic system synthesis VI: The cycloaddition derivatives of benzothiazipine and benzodiazepine. Chin. Chem. Lett. 1994, 5(7), 557560.

    1995 (3, SCI 3)(SCI 共计3)

    7.         许家喜, 金声*. 罂粟花粉中水溶性肽的分离纯化、序列测定和合成的研究. 化学学报 1995, 53, 822827.

    8.         Xu, Jiaxi*; Qin, Zhihui; Yang, Jun; Cai, Mengshen. Design and synthesis of analogs of Schistosoma mansoni P28 antigenic peptide P141. Chin. Chem. Lett. 1995, 6(6), 465466.

    9.         Xu, Jiaxi*; Jin, Sheng; Cai, Mengshen. Design, synthesis and activities of some new analogs and segments of the papaver somniferum pollen peptide PSPP2. Chin. Chem. Lett. 1995, 6(11), 941942.

    1996 (5, SCI 3) (SCI 共计6)

    10.     许家喜*, 蔡孟深, 石佑恩. 曼氏血吸虫合成多肽抗原研究. 高等学校化学学报 1996, 17(3), 424426.

    11.     许家喜. 血吸虫疫苗研究进展. 生命的化学 1996, 16(2), 4244.

    12.     麻密, 周达峰, 许家喜, 匡廷云, 汤佩松, 林忠平*. 细胞分离素基因(T-cyt)在转基因烟草中的表达及其对生长发育的影响. 应用与环境生物学报 1996, 2(1), 17.

    13.     He, Meiyu*; Xu, Jiaxi; Chan, Tak-Wah, Dominic; Lau, L. C. Rebecca. Positive ion electronspray Fourier transform ion cyclotron resonance mass  spectra of polypeptides and proteins. Rapid Commun. Mass Spectrom. 1996, 10(8), 897902.

    14.     Lam, Fung; Xu, Jiaxi; Chan, Kin Shing*. Binucleating ligands: Synthesis of acyclic achiral and chiral Schiff base- pyridine  and Schiff base-phosphine ligands. J. Org. Chem. 1996, 61(24), 84148418.

    1997 (4, SCI 1) (SCI 共计7)

    15.     许家喜*, 麻远. 同步多重有机合成. 化学通报 1997, (3), 1-8.

    16.     林孝元*, 贺晓然, 俞振培, 许家喜. FABCI条件下的RDA碎裂反应的比较研究. 北京大学学报(自然科学版) 1997, 33(2), 158162.

    17.     许家喜*, 金声. 罂粟花粉十七肽类似物和片段的合成及其抗肿瘤活性研究. 高等学校化学学报 1997, 18(7), 10981102

    18.     许家喜. 血吸虫合成多肽疫苗. 中国寄生虫病防治杂志 1997, 10(3), 227–229.

    1998 (19, SCI 8) (SCI 共计15)

    19.     许家喜. 固相有机合成. 有机化学 1998, 18(1), 110.

    20.     许家喜*, 杨俊海. 糖肽的合成. 化学通报 1998, (3), 2229.

    21.     傅南雁, 许家喜*. 抗菌多肽研究进展. 生命的化学 1998, 18(2), 2528.

    22.     许家喜. 血吸虫抗原肽对某些肿瘤细胞的抑制作用. 生命科学 1998, 10(3), 150151.

    23.     Xu, Jiaxi*; Cai, Mengshen. Mapping the antigenic peptides of Sm26/2 in Glutathione S-transferases of Schistosoma Mansoni. Chin. Chem. Lett. 1998, 9(4), 377379.

    24.     Xu, Jiaxi; Jin, Sheng*; Zhang, Zeying; Mak, Thomas C. W. 7-Benzoyl-2,3,4a,6-tetraphenyl-4a,5,6,12-tetrahydro-1H,7H-1,3-oxazino[3,2-d][1,5]benzodiazepine. Acta Cryst. 1998, C54, 666668.

    25.     许家喜, 金声*, 张泽莹, 麦松威. 1,3,3a,5-四苯基-3a,4,5,11-四氢-3H,6H-1,2,4-三唑并[4,3-d][1,5]苯并二氮杂卓的合成和晶体结构. 高等学校化学学报 1998, 19(7), 10701073.

    26.     许家喜, 金声*. 1,3,3a-三苯基-5-(2-溴苯基)-3a,4,5,11-四氢-3H-1,2,4-三唑并[4,3-d][1,5]苯并硫氮杂卓的合成和晶体结构. 北京大学学报(自然科学版) 1998, 34(4), 442446.

    27.     Xu, Jiaxi*; He, Meiyu; Jin, Sheng. Mass spectrometeric studies of tetrasubstituted 3a,4,5,11-tetrahydro-3H-1,2,4-triazolo[4,3-d][1,5]benzothiazepines. Rapid Commun. Mass Spectrom. 1998, 12(16), 11151117.

    28.     许家喜*, 杨俊海. 糖肽的固相合成. 合成化学 1998, 6(3), 248254.

    29.     Xu, Jiaxi; Lan, Ruoxi; Jin, Sheng*. Crystal structure of 3-(4-methoxyphenyl)-1-methyl-pyrrolo[2,1-b]benzothiazole. Jiegou Huaxue (Chin. J. Struct. Chem.) 1998, 17(5), 345348.

    30.     Xu, Jiaxi; Lan, Ruoxi; Jin, Sheng. Crystal structure of 1,1-dichloro-1a,3-diphenyl-1,1a,2,3-tetrahydro-azirino[2,1-d][1,5]benzothiazepine (C22H17Cl2NS). Jiegou Huaxue (Chin. J. Struct. Chem.) 1998, 17(5), 349352.

    31.     Xu, Jiaxi; Jin, Sheng*; Zhang, Zeying; Mak, Thomas C. W. Structure of 6-(4-chlorophenyl)-3-methyl-2,4a-diphenyl-4a,5,6,12-tetrahydro-1H-1,3-oxazino[3,2-d][1,5]benzothiazepine. Acta Cryst. 1998, C54(10), 15251527.

    32.     许家喜, 兰若曦, 金声*. 1a,3-二苯基-1,1,4,4-四氯-1a,2,3,4-四氢-1H-口丫丙啶并[2,1-e][1,6]苯并硫氮辛因的合成及晶体结构. 高等学校化学学报 1998, 19(11), 17741776.

    33.     许家喜, 金声*. 2,6-二甲基-3-苯基-4a-对甲苯基-7-苯甲酰基-4a,5,6,12-四氢-1H,7H-1,3-噁嗪并[3,2-d][1,5]苯并二氮杂卓-1-酮的合成及晶体结构. 结构化学 1998, 17(6), 454458.

    34.     许家喜*, 金声. 血吸虫抗原肽对某些肿瘤细胞的抑制作用. 北京大学学报(自然科学版) 1998, 34(6), 836840.

    35.     许家喜, 蔡孟深. 曼氏血吸虫谷胱甘肽S-转移酶Sm26/2的抗原肽研究. 高等学校化学学报 1998, 19(12), 19751978.

    36.     许家喜. 含手性碳原子的[3,3]s 迁移反应的立体化学过程. 大学化学 1998, 13(6), 1619.

    37.     Xu, Jiaxi; Jin, Sheng*; Xing, Qiyi. Cycloaddition reaction of benzoheteroazepine: Synthesis of 4a,5,6,12-tetrahydro-1H-1,3-oxazino[3,2-d][1,5]benzothiazepin-1-ones and 1H,7H-1,3-oxazino[3,2-d][1,5]benzodiazepin-1-ones. Phosphorus Sulfur Silicon Relat. Elem. 1998, 141, 5770.

    1999 (31, SCI 25) (SCI 共计40)

    38.     Xu, Jiaxi*; Jin, Sheng. Thermal cycloaddition reaction of symmetrical and unsymmetrical a-diazo-b-diketones with 4-aryl-2-methyl-2,3-dihydro-1,5-benzothia/diazepines. Heteroat. Chem. 1999, 10(1), 3540.

    39.     Xu, Jiaxi*; Wu, Haitao; Jin, Sheng. Cycloaddition reaction of benzoheteroazepine II: Reactions and conformations of cycloadducts on 1,5-benzothiazepines and 1,5-benzodiazepines with nitrile imine and nitrile oxides. Chin. J. Chem. 1999, 17(1), 8491.

    40.     Xu, Jiaxi*; Cai, Mengshen. Prediction, synthesis and antigenicity of the antigenic peptides of 26kDa glutathione S-transferase of Schistosoma japonicum (Sj26). Chin. Chem. Lett. 1999, 10(1), 2728.

    41.     Xu, Jiaxi*; Jin, Sheng. Synthesis, structure and antitumor activities of tridecapeptide PSPP3 from Papaver Somniferum pollen. Chin. Chem. Lett. 1999, 10(2), 115116.

    42.     Xu, Jiaxi; Zhang Xinyu; Jin, Sheng*. Crystal structure of 1,1-dichloro-3-dichloromethyl-1a,3-diphenyl-1a,2,3,4-tetrahydro-1H-azirino[1,2-a][1,5]benzodiazepine (C23H18Cl4N2). Jiegou Huaxue (Chin. J. Struct. Chem.) 1999, 18(2), 154158.

    43.     许家喜*, 秦致辉, 易有云, 蔡孟深. 曼氏血吸虫28kD谷胱甘肽S-转移酶的有效抗原肽P141结构与活性研究. 北京大学学报(自然科学版) 1999, 35(2), 162166.

    44.     许家喜, 缪平, 宋艳玲, 金声*. 几种花粉多肽和多糖的研究. 北京大学学报(自然科学版) 1999, 35(2), 178182.

    45.     许家喜*, 秦致辉, 蔡孟深, 庄辉. 戊型肝炎病毒(HEV)蛋白抗原肽的化学合成及其在血清学诊断的应用. 药学学报 1999, 34(4), 286289.

    46.     许家喜*, 麻密, 麻远, 林忠平. 一种简单有效的检测基因表达产物的方法. 科学通报 1999, 44(9), 947951.

    47.     许家喜*, 金声. 罂粟花粉十三肽类似物的合成及其结构与抗肿瘤活性关系研究. 高等学校化学学报 1999, 20(5), 722726.

    48.     Xu, Jiaxi*; Wu, Haitao; Jin, Sheng. Fast-atom bombardment mass spectrometric studies of trisubstituted 3a,4,5,11-tetrahydro-1,2,4-oxadiazolo[5,4-d][1,5]benzothiazepines. Rapid Commun. Mass Spectrom. 1999, 13(10), 908911.

    49.     Xu, Jiaxi*; Wu, Haitao; Jin, Sheng. Fast-atom bombardment mass spectrometric studies of trisubstituted 3a,4,5,11-tetrahydro-6H-1,2,4-oxadiazolo[5,4-a][1,5]benzodiazepines. Rapid Commun. Mass Spectrom. 1999, 13(10), 963965.

    50.     Xu, Jiaxi; Li, Xiaoyu; Wang, Zhemin; Yang, Qingchuan; Yan, Chunhua. Methyl (2S)-2-[(5R)-3,5-diphenyl-4,5-dihydro-1,2,4-oxadiazol-4-yl]-3-phenylpropanoate. Acta Cryst. 1999, C55, 650652.

    51.     许家喜*, 于力. 氨基膦酸及其酯的合成. 合成化学 1999, 7(2), 153158.

    52.     许家喜*, 王述恒, 易有云, 蔡孟深. 日本血吸虫26ku谷胱甘肽S-转移酶Sj26合成多肽抗原研究. 应用化学 1999, 16(3), 3740.

    53.     Wang, Hongzhong; Xu, Jiaxi; Mi, Baoyu; Jin, Sheng*. Crystal structure of triethyl 6-benzoyl-3a-(4-fluorophenyl)-2,3,3a,4,5,6-hexahydro-5-methyl-1H-pyrro[1,2-a][1,5]benzodiazepine-1,2,3-tricarboxylate. Jiegou Huaxue (Chin. J. Struct. Chem.) 1999, 18(4), 254258.

    54.     Wang, Hongzhong; Xu, Jiaxi; Mi, Baoyu; Jin, Sheng*. Crystal structure of ethyl 4-benzoyl-1a,2,3,4-tetrahydro-3-methyl-1a-(4-methylphenyl)-1H-azirino[1,2-a][1,5]benzodiazepine-1-carboxylate (C28H28N2O3). Jiegou Huaxue (Chin. J. Struct. Chem.) 1999, 18(4), 263266.

    55.     Xu, Jiaxi; Zhang Xinyu; Jin, Sheng*. Crystal structure of 1,1-dichloro-4-formyl-3-methyl-1a-phenyl-1a,2,3,4-tetrahydro-1H-azirino[1,2-a][1,5]benzodiazepine (C18H16Cl2N2O). Jiegou Huaxue (Chin. J. Struct. Chem.) 1999, 18(4), 267270.

    56.     Xu, Jiaxi*; Zhang, Zeying. Synthesis and crystal structure of 4,6-di-tert-butyl-2-hydroxy-3-(N-1-phenylethyliminomethyl)phenyl bis(triphenylphosphine)palladium bromide. Jiegou Huaxue (Chin. J. Struct. Chem.) 1999, 18(4), 290295.

    57.     Xu, Jiaxi*; Jiao, Peng; Wang, Zhemin. Synthesis and crystal structure of triethyl 1,2,2-triphenylpyrrolidine-3,4,5-tricarboxylate, a proline derivative. Jiegou Huaxue (Chin. J. Struct. Chem.) 1999, 18(4), 310314.

    58.     王鼎, 许家喜*. 肿瘤坏死因子(TNF)及其抑制剂. 生命的化学 1999, 19(4), 189192.

    59.     Xu, Jiaxi*; Zhang, Xinyu; Jin, Sheng. The mass spectral fragmentation of cis- and trans-1a,3-disubstituted-1,1-dichloro-1a,2,3,4-tetrahydro-1H-azirino[1,2-a][1,5]benzodiazepines. Rapid Commun. Mass Spectrom. 1999, 13(14), 14441447.

    60.     Xu, Jiaxi; Lan, Ruoxi; Jin, Sheng*. Mass spectral fragmentation patterns of 1a,3-diaryl-1,1,4,4-tetrachloro-1a,2,3,4-tetrahydro-1H-azirino[2,1-e][1,6]benzothiazocines. Rapid Commun. Mass Spectrom. 1999, 13(14), 15061510.

    61.     Xu, Jiaxi; Lan, Ruoxi; Jin, Sheng*. Electron impact mass spectra of 1a,3-disubstituted-1,1-dichloro-1,1a,2,3-tetrahydro-azirino[2,1-d][1,5]benzothiazepines. Rapid Commun. Mass Spectrom. 1999, 13(14), 15111514.

    62.     Zhang Xinyu; Xu, Jiaxi; Jin, Sheng*. Cycloaddition of benzoheteroazepine III: Reaction of 2,3-dihydro-1H-1,5-benzodiazepines with dichlorocarbene and stereo-structures of products. Chin. J. Chem. 1999, 17(4), 404410.

    63.     Wang, Hongzhong; Yao, Dan; Lan, Ruoxi; Xu, Jiaxi; Jin, Sheng*. A new rearrangement reaction of 2-phenyl substituted benzothiazepine with ethoxycarbonyl carbene: Mechanism of the reaction and structure of the product. Chin. Chem. Lett. 1999, 10(8), 625628.

    64.     Xu, Jiaxi; Jin, Sheng*. 1,3a,5-Triphenyl-3a,4,5,6-tetrahydro-1,2,4-oxadiazolo[4,5-a][1,5]benzodiazepine. Acta Cryst. 1999, C55, 15791581.

    65.     Xu, Jiaxi; Liang, Bo; Jin, Sheng*. Synthesis of 1,5-benzothiazepine-1-oxide/-1,1-dioxide derivatives and 1,2-oxazirino[2,3-a][1,5]benzodiazepine. Phosphorus Sulfur Silicon Relat. Elem. 1999, 152, 18.

    66.     Xu, Jiaxi*; Xia, Chengfeng; Yu, Li; Zhou, Qingzhong. Synthesis of phosphonopeptides containing 1-aminoalkylphosphonic acid. Phosphorus Sulfur Silicon Relat. Elem. 1999, 152, 3544.

    67.     许家喜, 兰若曦, 金声*. 3-甲基-1a-(4-甲氧基苯基)-1,1-二氯-1,1a,2,3-四氢-口丫丙啶并[2,1-a][1,5]苯并硫氮杂卓的合成和晶体结构. 化学学报 1999, 57(12), 13591363.

    68.     Xu, Jiaxi*; Chen, Liangbi. The mass spectral fragmentation of 1a,3-disubstituted 4-benzoyl-1a,2,3,4-tetrahydro-oxazirino[2,3-a][1,5]benzodiazepines. Rapid Commun. Mass Spectrom. 1999, 13(23), 24242427.

    2000 (15, SCI 10) (SCI 共计50)

    69.     许家喜*, 杨俊海. 正交保护赖氨酸的合成. 化学通报 2000, 63(1), 2629.

    70.     Xu, Jiaxi*; Chen, Liangbi. Synthesis of oxazirino[2,3-a][1,5]benzodiazepines by oxidation of 1H-1,5-benzodiazepines with m-chloroperbenzoic acid (MCPBA). Heteroat. Chem. 2000, 11(2), 158162.

    71.     Xu, Jiaxi; Zhang, Xinyu; Jin, Sheng*. Mass spectral fragmentation of cis- and trans-1a,3-disubstituted-1,1-dichloro-4-formyl-1a,2,3,4-tetrahydro-1H-azirino[1,2-a][1,5]benzodiazepines. Chin. J. Chem. 2000, 18(3), 368372.

    72.     Xu, Jiaxi*; Zuo, Gang; Jiao, Peng; Wang, Hongzhong; Jin, Sheng; Chan, Albert S. C. Electron impact mass spectral fragmentation patternsof 2a,4-disubstituted 5-benzoyl-2-chloro-2a,3,4,5-tetrahydro-azeto[1,2-a][1,5]benzodiazepin-1(2H)-ones. Rapid Commun. Mass Spectrom. 2000, 14(8), 633636.

    73.     Xu, Jiaxi*; Jiao, Peng; Zuo, Gang; Jin, Sheng. Electron impact mass spectral fragmentation of 2a,4-disubstituted 2-chloro/2,2-dichloro-2,2a,3,4-tetrahydro-1H-azeto[2,1-d][1,5]benzothiazepin-1-ones. Rapid Commun. Mass Spectrom. 2000, 14(8), 637640.

    74.     陈良壁; 许家喜*. 通过a-重氮-b-二酮与醛酮的环加成反应合成4H-1,3-二噁环己-5--4-酮衍生物. 合成化学 2000, 8(3), 231233.

    75.     许家喜*; 焦鹏. 固相载体上的环加成反应及其应用. 化学进展 2000, 12(2), 131140.

    76.     Xu, Jiaxi*; Fu, Nanyan. A facile synthesis of N-protected 1-aminoalkylphosphonamidate derivatives. Synth. Commun. 2000, 30(22), 41374145.

    77.     Xu, Jiaxi*; Wang, Ding; Zhang, Qihan; Huang, Aijin. Regioselective synthesis and electron impact mass spectral fragmentation differentiation of 2- or 3-isopropylthio/phenylthiosuccinic acid 4-methyl/isopropyl esters. Rapid Commun. Mass Spectrom. 2000, 14(19), 17461750.

    78.     Xu, Jiaxi*; Ma, Yuan, Duan, Lifang. A novel synthetic route to N-protected 1-aminoalkylphosphonates. Heteroat. Chem. 2000, 11(6), 417421.

    79.     许家喜*, 夏成峰. 芳核手性树状化合物的合成. 合成化学 2000, 8(5), 410412, 418.

    80.     Xu, Hao; Xu, Jiaxi; Liu, Xuehui; Jin, Sheng, Cui, Yuxin*. 1H NMR study on the stereochemistry of 1,3-oxazino[3,2-d][1,5]benzodiazepin-1-ones. 波谱学杂志 2000, 17(5), 363367.

    81.     许家喜. 合成多肽疫苗研究进展. 高等学校化学学报 2000, 21(11), 16881693.

    82.     Xu, Jiaxi*; Zhang, Qihan; Wang, Chengbo. Electron impact mass spectral fragmentation of 3a,5-disubstituted 1,3-diphenyl-3a,4,5,6-tetrahydro-3H-1,2,4-triazolo[4,3-a][1,5]benzodiazepines. Rapid Commun. Mass Spectrom. 2000, 14(24), 23392342.

    83.     Xu, Jiaxi*; Zuo, Gang. Electron impact mass spectral studies of 2a,4-disubstituted 2-phthalimido-2,2a,3,4-tetrahydro-1H-azeto[2,1-d][1,5]benzothiazepin-1-ones. Rapid Commun. Mass Spectrom. 2000, 14(24), 23732376.

    2001 (13, SCI 13) (SCI 共计63)

    84.     陈良壁, 张奇涵, 许家喜*. a-重氮-b-二羰基化合物在有机合成中的应用. 有机化学 2001, 21(2), 8996.

    85.     Zhang, Qihan; Xu, Jiaxi*. A novel conversion of 2,4-diaryl-2,3-dihydro-1H-1,5-benzodiazepines into 2,4-diaryl-3H-1,5-benzodiazepines. Chin. J. Chem. 2001, 19(4), 378380.

    86.     Xu, Jiaxi*; Fu, Nanyan. A novel and convenient method for synthesizing unsymmetrical N-benzyloxycarbonyl-protected 1-amino-1-aryl-alkylphosphonate mixed diesters. J. Chem. Soc. Perkin. Trans. 1 2001, 12231226.

    87.     Tian, Hongqi; She, Xuegong; Xu, Jiaxi; Shi, Yian*. Enantioselective epoxidation of terminal olefins by chiral dioxirane. Org. Lett. 2001, 3(12), 19291931.

    88.     Xu, Jiaxi*; Wei, Ming. A convenient method for the synthesis of N-protected 1-aminoalkyl-phosphonate mixed monothioesters and dithioesters. Synth. Commun. 2001, 31(10), 14891497.

    89.     Xu, Jiaxi*; Zhang, Qihan; Chen, Liangbi; Chen, Hui. Chemoselectivity in reactions of an a-diazo-b-diketone with some conjugative double bond systems. J. Chem. Soc. Perkin. Trans. 1 2001, (18), 22662268.

    90.     He, Meiyu*; Xu, Jiaxi; He, Xiaoran; Chan, Tak Wah Dominic; Lau, Rebecca, L. C. Sequence analysis of peptides with biological activities using electrospray-Fourier transform ion cyclotron resonance mass spectrometry. Chin. Sci. Bull. 2001, 46(15), 12811285.

    91.     Xu, Jiaxi*; Wang, Chenbo; Zhang, Qihan. Synthesis of 1,3,3a,5-tetraaryl-3a,4,5,6-tetrahydro-3H-1,2,4-triazolo[4,3-a][1,5]benzodiazepines. Heteroat. Chem. 2001, 12(6), 557559.

    92.     Wang, Hongzhong*; Zhou, Xin; Xu, Jiaxi; Jin, Sheng; Li, Yueming; Chan, Albert S. C. On the mechanism and stereochemistry of the formation of b-lactam derivatives of 2,4-disubstituted-2,3-dihydrobenzo[1,4]diazepines. J. Heterocycl. Chem. 2001, 38 (5), 10311034.

    93.     Xu, Jiaxi*; Zhang, Qihan. Synthesis of 4H-1,3-oxathiin-4-ones by reaction of a-diazo-b-diketone with thiones. Heteroat. Chem. 2001, 12(7), 630632.

    94.     Xu, Jiaxi*; Zuo, Gang; Chan, Wing-lai. Reaction of 2,3-dihydro-1H-1,5-benzodiazepines and chloroacetyl chlorides: Synthesis of 2a,3,4,5-tetrahydro-azeto[1,2-a][1,5]benzodiazepin-1(2H)-ones. Heteroat. Chem. 2001, 12(7), 636640.

    95.     Tam, James P*; Xu, Jiaxi; Eom, Khee Dong. Methods and strategies of peptide ligation. Biopolymers (Pept. Sci.) 2001, 60(3), 194205.

    96.     Jiao, Peng; Xu, Jiaxi*; Zhang, Qihan; Choi, Michael C. K.; Chan, Albert S. C. Synthesis of novel C2-symmetric and enantiomerically pure bisbenzoxazoles and bisbenzothiazoles derived from L- and D-tartaric acids. Tetrahedron: Asymmetry 2001, 12(22), 30813088.

    2002 (8, SCI 7) (SCI 共计70)

    97.     许家喜*; 麻远. 液相组合化学. 化学通报 2002, (3), 145152.

    98.     Xu, Jiaxi*; Chen, Liangbi. Reactions of unsymmetrical a-diazo-b-diketones with imines: syntheses of 4H-1,3-oxazin-4-ones. Heteroat. Chem. 2002, 13(2), 165168.

    99.     Xu, Jiaxi*; Zuo, Gang; Zhang, Qihan; Chan, Wing Lai. Stereospecific synthesis of 2-phthalimido-2a,3,4,5-tetrahydro-1H-azeto[2,1-d][1,5]benzothiazepin-1-ones. Heteroat. Chem. 2002, 13(3), 276279.

    100.  Xu, Jiaxi*; Jiao, Peng; Deng, Dayi; Zhang, Qihan; Tsang, Chun Wai; Chan, Albert S. C. Electron impact mass spectral fragmentation of chiral bisbenzoxazole, bisbenzothiazole and biscarbamide derivatives of 2,2-dimethyl-1,3-dioxolane. Rapid Commun. Mass Spectrom. 2002, 16(12), 11741179.

    101.  杨俊海; 许家喜*. 曼氏和日本血吸虫副肌球蛋白的抗原肽研究. 有机化学 2002, 22(6), 423427.

    102.  Xu, Jiaxi*; Jiao, Peng. Direct NH-aziridination of a,b-unsaturated ketones. J. Chem. Soc. Perkin. Trans. 1 2002, (12), 14911493.

    103.  苏贤斌, 张奇涵, 武永庆, 许家喜. 用α-苯乙胺拆分制备高光学活性的线性二级醇. 有机化学 2002, 22(7), 496-500.

    104.  Xu, Jiaxi. A new and expeditious asymmetric synthesis of (R)- and (S)-2-aminoalkanesulfonic acids from chiral amino alcohols. Tetrahedron: Asymmetry 2002, 13(11), 11291134.

    2003 (6, SCI 6) (SCI 共计76)

    105.  许家喜. 羟基磺酸、氨基磺酸和磺酰肽的合成. 有机化学 2003, 23(1), 19.

    106.  Zuo, Gang; Zhang, Qihan; Xu, Jiaxi*. Diastereospecific synthesis of (S,S)-2-substituted-4,4-diphenyl-3,1-oxazabicyclo[3.3.0]octanes. Heteroat. Chem. 2003, 14(1), 4245.

    107.  Xu, Jiaxi*, Zuo, Gang. Mass spectral fragmentation of (S,S)-2-substituted-4,4-diphenyl-3,1-oxazabicyclo[3.3.0]octanes: Ring contraction of pyrrolidine and 1,3-oxazolidine in mass spectrometry. Rapid Commun. Mass Spectrom. 2003, 17(14), 16511656.

    108.  Xu, Jiaxi*; Su, Xianbin; Zhang, Qihan. Preparation of high optically pure linear secondary alcohols via asymmetric reduction of prochiral ketones by borane. Tetrahedron: Asymmetry 2003, 14(13), 17811786.

    109.  Huang, Xu; Xu, Jiaxi*. Specific synthesis of azeto[1,2-d][1,5]benzothiazepin/diazepin-1-ones. Heteroat. Chem. 2003, 14(6), 564569.

    110.  Xu, Jiaxi*; Wei, Tiezheng; Zhang, Qihan. Effect of temperature on the enantioselectivity in the oxazaborolidine-catalyzed asymmetric reduction of ketones. non-catalytic borane reduction, a non-neglectable factor in reduction system. J. Org. Chem. 2003, 68(26), 1014610151.

    2004 (12, SCI 11) (SCI 共计87)

    111.  Xu, Jiaxi*; Xu Shu. A general route to synthesis of N-protected 1-substituted and 1,2-disubstituted taurines. Synthesis 2004, (2), 276282.

    112.  Gao, Yuanhe; Zhang, Qihan; Xu, Jiaxi*. A convenient and effective method for synthesizing b-amino-a,b-unsaturated esters and ketones. Synth. Commun. 2004, 34(5), 909916.

    113.  马琳鸽, 许家喜*. 非对称氮杂环丙烷的亲核开环反应及其区域选择性. 化学进展 2004, 16(2), 220235.

    114.  Xu, Jiaxi*; Huang, Xu. Mass spectrometric fragmentation of 2a,4-disubstituted 2,2a,3,4-tetrahydro-2-phenoxyl-1H-azeto[2,1-d][1,5]benzothiazepin-1-ones under electron impact ionization conditions. Rapid Commun. Mass Spectrom. 2004, 18(8), 859862.

    115.  Xu, Jiaxi*; Jiao, Peng; He, Zheng; Zhang, Qihan; Yan, Chunhua. Intermolecular phenolic hydroxy methylation occurring between chiral N,N-bis(2-hydroxyphenyl)-2,2-dimethyl-1,3-dioxolane-4,5-dicarbamide and co-crystallized methanol under electron impact ionization conditions. Chin. J. Chem. 2004, 22(5), 455459.

    116.  Xu, Jiaxi*; Wei, Tiezheng; Xia, Jiakun; Zhang, Qihan; Wu, Hesong. Preparation of highly optically pure homochiral sulfide-containing alcohols via oxazaborolidine-catalyzed asymmetric borane reduction of ketones. Chirality 2004, 16(6), 341346.

    117.  Xu, Jiaxi*; Ma, Linge; Jiao, Peng. Asymmetric aziridination of chalcones catalyzed by a novel backbone 1,8-bisoxazolinylanthracene (AnBOX)-bopper bomplex. Chem. Commun. 2004, (14), 1616-1617.

    118.  张奇涵 林晨翔 张珊珊 许家喜*. 光学活性反式1-(4-烷基环己基)醇的制备. 有机化学 2004, 24(9),  10691074.

    119.  Xu, Jiaxi*; Wang, Chao; Zhang, Qihan. Reaction of 2,3-dihydro-1,5-benzothiazepines and phenylacetyl chloride in the presence of triethylamine: a new aspect on the formation mechanism of dihydro-1,3-oxazin-4-one derivatives. Chin. J. Chem. 2004, 22(9), 10121018.

    120.  Xu, Jiaxi*; Wei, Tiezheng; Zhang, Qihan. Influences of electronic effects and anions on the enantioselectivity in the oxazaborolidine-catalyzed asymmetric borane reduction of ketones. J. Org. Chem. 2004, 69(20), 68606866.

    121.  许家喜. 花粉多肽与花粉过敏. 大学化学 2004, 19(5), 2426, 30.

    122.  Lu, Shao-Feng; Du, Da-Ming*; Zhang, Shi-Wei; Xu, Jiaxi*. Facile synthesis of C2-symmetric tridentate bis(thiazoline) and bis(oxazoline) ligands and their application in the enantioselective Henry reaction. Tetrahedron: Asymmetry 2004, 15(21), 34333441.

    2005 (20, SCI 19) (SCI 共计106)

    123.  Liang, Yong; Jiao, Lei; Zhang, Shiwei; Xu, Jiaxi*. Microwave and photoirradiation-induced Staudinger reactions of cyclic imines and ketenes generated from α-diazoketones. A further investigation into the Stereochemical process. J. Org. Chem. 2005, 70(1), 334337.

    124.  Wei, Tiezheng; Lan, Yu; Xu, Jiaxi*. Mildly and highly selective reductive deoxygenation of para-di- and monoalkylaminophenyl ketones by borane. Heteroat. Chem. 2005, 16(1), 25.

    125.  Xu, Jiaxi*; Wei, Tiezheng; Lin, Shrong-Shi; Zhang, Qihan. Rationale on abnormal effect of temperature on the enantioselectivity in the asymmetric borane reduction of ketones catalyzed by prolinol. Helv. Chim. Acta 2005, 88(1), 180186.

    126.  Jiao, Lei; Liang, Yong; Wu, Chunzan; Huang, Xu; Xu, Jiaxi*. Reaction of imidates with phenoxyacetyl chloride. Chem. Res. Chin. Univ. 2005, 21(1), 5964.

    127.  Wang, Zhanyue; Du, Daming*; Xu, Jiaxi. Synthesis of novel chiral semicrown ether-like bis(oxazoline) ligands and application in enantioselective cycloaddition of styrene. Synth. Commun. 2005, 35(2), 299313.

    128.  Xu, Jiaxi. A structurally diverse heterocyclic library: A benzothiazepine-fused b-lactam library derived from reaction of 2,3-dihydro-1,5-benzothiazepines and acyl chlorides: synthesis and stereochemistry. Molecular Diversity 2005, 9(1-3), 4549.

    129.  Du, Da-Ming*; Lu, Shao-Feng; Fang, Tao; Xu, Jiaxi*. Asymmetric Henry reaction catalyzed by C2-symmetric tridentate bis(oxazoline) and bis(thiazoline) complexes: Metal-controlled reversal of enantioselectivity. J. Org. Chem. 2005, 70(9), 37123715.

    130.  Du, Da-Ming*; Fang, Tao; Lu, Shao-Feng; Xu, Jiaxi*. C3-Symmetric tris(b-hydroxy amide)-titanium complex catalyzed enantioselective addition of phenylacetylene to aldehydes. Org. Lett. 2005, 7(11), 20812084.

    131.  Chen, Hui; Xu, Jiaxi; Xin, Bin; He, Meiyu*. Sequence analysis on biological active peptides using electrospray ionization-Fourier transform ion cyclotron resonance mass spectrometer. Chin. Sci. Bull. 2005, 50(9), 853857.

    132.  Xu, Jiaxi*; Ma, Yuan; Xu, Shu; Zhao, Yufen. Negative ion electrospray ionization mass spectrometry of N-benzyloxycarbonyl protected 1-substituted and cyclic taurines. Rapid Commun. Mass Spectrom. 2005, 19(13), 18351838.

    133.  Xu, Jiaxi*; Zuo, Gang; Liang, Bo. Differentiation of constitutional isomer of 2,2a,3,4-tetrahydro-4-methyl-2a-phenyl-2-(thiophen-2-yl)-1H-azeto[2,1-d][1,5]benzothiazepin-1-one-5-oxide and fragmentations of 2,3-dihydro- 2,4-diphenyl-1,5-benzothiazepine-1-oxide/-1,1-dioxide. Chem. Res. Chin. Univ. 2005, 21(3), 274279.

    134.  Huang, Jiaxing; Wang, Fei; Du, Daming; Xu, Jiaxi*. An expeditious synthesis of 1-substituted and cyclic taurines. Synthesis 2005, (13), 21222128.

    135.  Xu, Jiaxi*; Huang, Xu. Mass spectrometry of 2a,4-disubstituted 5-benzoyl-2a,3,4,5-tetrahydro-2-phenoxy-azeto[1,2-a][1,5]benzodiazepin-1(2H)-ones under electron impact ionization conditions. Chem. Res. Chin. Univ. 2005, 21(4), 452456.

    136.  Xu, Jiaxi*; Xia, Jiakun; Lan, Yu. Convenient and efficient synthesis of 1,1-bis-(4-alkylthiophenyl)-1-alkenes via tandem Friedel-Crafts acylation and alkylation of sulfides and acyl chlorides. Synth. Commun. 2005, 35(17),  23472353.

    137.  Xu, Jiaxi*; Xu, Shu; Zhang, Qihan. The first synthesis of optically active 1-substituted taurines. Heteroat. Chem. 2005, 16(6), 466471.

    138.  Xu, Jiaxi*; Lan, Yu; Wei, Tiezheng; Zhang, Qihan. Chiral oxazaborolidine-catalyzed asymmetric borane reduction of alkyl 1-(4-dialkylaminophenyl) ketones. Chin. J. Chem. 2005, 23(10),14571461.

    139.  Ma, Linge; Du, Daming; Xu, Jiaxi*. Rational tuning chelate size of bis-oxazoline ligands to improve enantioselectivity in the asymmetric aziridination of chalcones. J. Org. Chem. 2005, 70 (24),  1015510158.

    140.  Ma, Linge; Jiao, Peng; Zhang, Qihan; Xu, Jiaxi*. Rigid backbone 1,8-anthracene-linked bis-oxazolines (AnBOXes): design, synthesis, application and characteristics in catalytic asymmetric aziridination. Tetrahedron: Asymmetry 2005, 16(22), 37183734.

    141.  Xu, Jiaxi*; Wang, Chao. Mass spectrometric fragmentation of 2a,4-disubstituted 2,2a,3,4-tetrahydro-2-phenyl-1H-azeto[2,1-d][1,5]benzothiazepin-1-ones under electron impact ionization conditions and comparison with their 2-heteroatom substituted analogues. Phosphorus Sulfur Silicon Relat. Elem. 2005, 180(12), 27792785.

    142.  Liu, H.; Xu, J. X*. Synthesis of 1-(N-ethoxycarbonylamino)alkylphosphonic monoesters. Amino Acids 2005, 29(3), 241243.

    2006 (30, SCI 27) (SCI 共计133)

    143.  Huang, Jiaxing; Du, Da-Ming; Xu, Jiaxi* Facile synthesis of 1,1-disubstituted taurines. Synthesis 2006, (2), 315319.

    144.  Jiao, Lei; Zhang,Qianfeng; Liang, Yong; Zhang, Shiwei; Xu, Jiaxi*. A versatile method for the synthesis of 3-alkoxycarbonyl b-lactam derivatives. J. Org. Chem. 2006, 71(2), 815818.

    145.  Wu, Chunzan; Huang, Jiaxing; Zhang, Qihan; Xu, Jiaxi*. Further investigation on the rearrangement mechanism in the reaction of 1,5-benzothiazepines and ethoxycarbonylcarbene. Chem. Res. Chin. Univ. 2006, 22(1), 3639.

    146.  Liu, Han.; Xu, Jiaxi*. (S)-2-Aryl-4,4-diphenyl-3,1,2-oxazaboro[3.3.0]octanes: Efficient catalysts for the asymmetric borane reduction of electron-deficient ketones. J. Mol. Cat. A: Chem. 2006, 244(1-2), 6872.

    147.  Jiao, Lei; Liang, Yong; Zhang, Qianfeng; Zhang, Shiwei; Xu, Jiaxi*. Catalyst-free, high-yield, and stereospecific synthesis of 3-phenylthio b-lactam derivatives. Synthesis 2006, (4), 659665.

    148.  Xu, Jiaxi*; Gao, Yuanhe, Straightforward synthesis of depsiphosphonopeptides via Mannich-type multiple component condensation. Synthesis 2006, (5), 783788.

    149.  Fu, Nanyan; Zhang, Qihan; Duan, Lifang; Xu, Jiaxi*. Facile synthesis of phosphonamidate and phosphonate-linked phosphonopeptides. J. Peptide Sci. 2006, 12(4), 303309.

    150.  Du, Da-Ming*; Fang, Tao; Xu, Jiaxi; Zhang, Shiwei. Structure well defined, recoverable C3-symmetric tris(b-hydroxy phosphoramide) catalyzed enantioselective borane reduction of ketones. Org. Lett. 2006, 8(7), 1327–1330.

    151.  王鼎, 张奇涵, 许家喜* 新型含硫肿瘤坏死因子类肽抑制剂的合成与活性, 高等学校化学学报 2006, 27(4), 669671.

    152.  马琳鸽,杜大明,许家喜*. 在不对称氮杂环丙烷化中双噁唑啉配位空间大小对对映选择性的影响.有机化学 2006, 26(4),  568572.

    153.  Liu, Han; Cai, Shuzong, Xu, Jiaxi*. Asymmetric synthesis of N-protected chiral 1-aminoalkylphosphonic acids and synthesis of side-chain functionalized depsiphosphonopeptides. J. Peptide Sci. 2006, 12(5), 337340.

    154.  Lu, Shao-Feng; Du, Da-Ming*; Xu, Jiaxi*. Enantioselective Friedel-Crafts alkylation of indoles with nitroalkenes catalyzed by bifunctional tridentate bis(oxazoline)-Zn(II) complex. Org. Lett. 2006, 8(10), 21152118.

    155.  Jiao, Lei; Liang, Yong; Xu, Jiaxi*. Origin of the relative stereoselectivity of the b-lactam formation in the Staudinger reaction. J. Am. Chem. Soc. 2006, 128(18), 60606069.

    156.  Yin, Wei; Ma, Yuan; Xu, Jiaxi; Zhao, Yufen. Microwave-assisted one-pot synthesis of 1-indanones from arenes and a,b-unsaturated acyl chlorides. J. Org. Chem. 2006, 71(11), 43124315.

    157.  Zhang, Qihan; Su, Xianbin; Xu, Jiaxi*. Comparative study on mass spectrometric fragmentation of linear chiral secondary alcohols (R)-1-(4-alkylphenyl) and (R)-1-(4-alkoxyl/thiophenyl) alcohols. Chem. Res. Chin. Univ. 2006, 22(3), 347350.

    158.  Liu, Han; Du, Daming; Xu, Jiaxi*. Effect of the secondary reduction on the enantioselectivity and function of additives in the chiral oxazaborolidine-catalyzed asymmetric borane reduction of ketones. Helv. Chim. Acta 2006, 89(5), 10671074.

    159.  Lu, Shao-Feng; Du, Da-Ming*; Xu, Jiaxi; Zhang, Shi-Wei. Asymmetric Michael addition of nitroalkanes to nitroalkenes catalyzed by C2-symmetric tridentate bis(oxazoline) and bis(thiazoline) zinc complexes. J. Am. Chem. Soc. 2006, 128(23), 74187419.

    160.  Fang, Tao; Xu, Jiaxi; Du, Da-Ming*. Highly enantioselective borane reduction of prochiral ketones catalyzed by C3-symmetric tripodal b-hydroxyl amines. Synlett 2006, (10), 15591563.

    161.  Ma, Linge; Du, Daming; Xu, Jiaxi*. Asymmetric aziridination of 1,3-dienes catalyzed by bisoxazoline-copper complexes. Chirality 2006, 18(8), 575580.

    162.  许家喜. 多烯化合物的Cope重排反应: [5,5]s迁移、串联[3,3]s迁移与自由基重排机理.大学化学 2006, 21(3), 2833.

    163.  Wang, Xiao; Wang, Yikai; Du, Daming; Xu, Jiaxi*. Solvent-free, AlCl3-promoted tandem Friedel-Crafts reaction of arenes and aldehydes. J. Mol. Cat. A: Chem. 2006, 255(1-2), 3135.

    164.  Xu, Shu; Xu, Jiaxi*. Mass spectrometric fragmentation of 1-(benzyloxycarbonyl)amino-2-alkyl/cycloalkyl thioacetates: A thioester pyrolysis-type rearrangement under electron impact ionization. Chin. Chem. Lett. 2006, 17(8), 10691072.

    165.  Wang, Yikai; Liang, Yong; Jiao, Lei; Du, Da-Ming; Xu, Jiaxi*. Do reaction conditions affect the stereoselectivity in the Staudinger reaction? J. Org. Chem. 2006, 71(18), 69836990.

    166.  许家喜. [3,3]s迁移反应过渡态立体化学过程的新观点.大学化学 2006, 21(4), 4044.

    167.  Fang, Tao; Xu, Jiaxi; Du, Da-Ming*. Facile synthesis of C3-symmetric tripodal β-hydroxy amide ligands and their Ti (IV) complex-catalyzed asymmetric addition of diethylzinc to aldehydes. Lett. Org. Chem. 2006, 3(10), 780786.

    168.  王一恺, 杜大明, 许家喜*. 微波对烯酮和亚胺形成b-内酰胺顺反选择性的影响. 辽宁石油化工大学学报 2006, 26(4), 9495.

    169.  Jiao, Peng; Ma, Linge; Zhang, Qihan; Xu Jiaxi*. Mass spectral fragmentation of 1,8-bis[4-substituted (oxazolin-2-yl)]anthracenes: ring-contraction rearrangement of oxazoline ring under electron impact ionization conditions. Chem. Res. Chin. Univ. 2006, 22(6), 753755.

    170.  Jiao, Peng; Zhang, Qihan; Xu Jiaxi*. Mass spectral fragmentation and cyclization of (S,S)-N,N’-bis[1-(hydroxymethyl)alkyl]anthracene/ naphthalene-1,8-dicarboxamides  under electron impact ionization conditions. Chem. Res. Chin. Univ. 2006, 22(6), 756759.

    171.  Liang, Yong; Jiao, Lei; Wang, Yuanyuan; Chen, Yuanyuan; Ma, Linge; Xu, Jiaxi; Zhang, Shiwei; Yu, Zhiqiang*. Nitrene equivalent mediated metal-free ring expansions of alkylidenecyclopropane and an alkylidenecyclobutane. Org. Lett. 2006, 8(25), 58775879.

    172.  Shen, Yu-Mei; Zhao, Mei-Xin; Xu, Jiaxi; Shi, Yian*. An amine promoted aziridination of chalcones. Anew. Chem. Int. Ed. 2006, 45(47), 80058008.