25230
当前位置: 首页   >  成果及论文
成果及论文

论文

第一作者及通讯作者

30 An efficient synthesis of Indolo[3,2-c]coumarins by Pd-catalyzed intramolecular Csingle bondH carbonylation

Hai-Bing Long, Xue-Hua Huang, Da-Xian You, Ye Liang, Jin-Bao Peng, Jia-Lei Yan*, Ai-Jun Ma*

      Tetrahedron Lett.2025, 168, 155716.


29 Synthesis of Tetracyclic Indole Skeleton Via Palladium-catalyzed Intramolecular Heck/Amino-carbonylation Cascade Reaction

BAI Ruiyi(白瑞异), DU Xiao, YAN Jialei, MA Aijun*  

      Chin. J. Syn. Chem.2025DOI: 10.15952/j.cnki.cjsc.1005-1511.20250023.


28 Chelation-Controlled Stereospecific Ring-Opening Arylation of α-Aminoaryl-Tethered Alkylidenecyclopropanes: Stereoselective Synthesis of Polysubstituted Conjugated Dienes

Miao-Miao Ji, Ying Tang, Wen-Mei Luo, Yong-Yu He, Ai-Jun Ma* and Jin-Bao Peng*  


25 De novo synthesis of atropisomeric benzofurans via Cu/SPDO complex catalyzed asymmetric formal [3 + 2] annulation

Fan-Xiao Meng(孟凡晓), Xing-Yu Wang, Ka Lu, Ju-Song Yang, Fu-Min Zhang,* Ai-Jun Ma,* Bao Du, Yong-Qiang Tu*

Sci. China Chem. 2025, 68, 174-180.

23 Copper-Catalyzed Sequential C(sp2)−H/C(sp3)−H Annulation of Indoles with Propargylic Alcohols to Access Hydrobenzo[b]carbazoles

Yi-Rui ZhangZong-Wang QiuZhao-Jie FuShao-Shuai ChenHan-Peng PanBao Qiong LiAi-Jun Ma*Xiang-Zhi Zhang*

Advanced Synthesis & Catalysis2024336, 1320-1324.


22 Cooperative Cu/Pd-Catalyzed 1,5-Boroacylation of Cyclopropyl-Substituted Alkylidenecyclopropanes

Hui-Hui Zeng, Yu-Qing Wang, Yong-Yu He, Xiao-Ling Zhong, Hongguang Li, Ai-Jun Ma*, and Jin-Bao Peng*

J. Org. Chem. 2024 89, 2637–2648.


    21 Acid-Promoted Cyclization of α-Azidobenzyl Ketones through C═N Bond Formation: Synthesis of 6-Substituted Quinoline Derivatives

    Jing-Yun Zheng(郑景云)Ying LuoTing-Ting OuXin-Jie ZhangYong-Qiang LaoNa FengJin-Bao PengXiang-Zhi ZhangXiaojun Yao, and Ai-Jun Ma*

    Org. Lett. 202426586-590.



    20  Ruthenium-Catalyzed Carbonylation of α-Aminoaryl-Tethered Alkylidenecyclopropanes: Synthesis of Eight-Membered Benzolactams  

    Miao-Miao Ji, Peng-Rui Liu, Jun-Dong Yan, Yong-Yu He, Hongguang Li, Ai-Jun Ma*, and Jin-Bao Peng*

    Org. Lett. 202426, 231-235.


    19 Direct syntheses of N-alkyl-2-pyridones using 2-halogenated pyridines

    Xia Chen(陈霞), Jianyi Shi, Yuqun Lin, Yibiao Li, Shaohua Jiang, Tianxiang Chen, Zhongzhi Zhu*, Ai-Jun Ma*

    Eur. J. Org. Chem. 2024, 27, e202301184.


    18 Synthesis of Benzo[6,6]-Spiroketal Compounds

    LIN Siwu(林思武), ZHAO Lili, SHEN Zhonghui, MA Ai-Jun*

    Chin. J. Syn. Chem.202331, 252-256.


    17 Total Synthesis of (+)-Peniciketal B

     Shan-Shan Li(李汕珊), Li-Li Zhao(赵丽丽), Min Pan, Na Feng, Bao-Qiong Li, Xiang-Zhi Zhang, Jin-Bao Peng*, and Ai-Jun Ma*

    Org. Lett. 2023, 25, 8501–8505.


    16 Palladium-Catalyzed Intramolecular Heck/Aminocarbonylation of Alkene-Tethered Iodobenzenes with Nitro Compounds: Synthesis of Carbamoyl-Substituted Benzoheterocycles

    Yun Kang, Jin-Liang Lu, Zhi ZhangYing-Kang LiangAi-Jun Ma*, and Jin-Bao Peng*

    J. Org. Chem. 2023, 88, 5097–5107.


    15 Ring-Opening-Recombination Strategy Based on 2-Methylbenzothiazole Salts: Syntheses of Thiazinopyrrole Fused-Ring Derivatives

    Shengting Xu, Zhongzhi Zhu, Zhendong Yang, Zuyu Mai, Tianxiang Chen, Ai-Jun Ma*,  Xiuwen Chen* 

      Advanced Synthesis & Catalysis, 2023365, 3819-3823.




    14 K2CO3-Promoted oxy-Michael Addition/Cyclization of α,β-Unsaturated Carbonyl Compounds with Naphthols: Synthesis of Naphthopyrans

     Shan-Shan Li(李汕珊), Li-Li Zhao(赵丽丽), Min Pan, Na Feng, Jin-Bao Peng, and Ai-Jun Ma*

    Molecules, 2023, 28, 5502.



    13 Synthesis and Antioxidant Activities of Novel Melatonin Derivatives

    HE Li(贺利), CHEN Mengting, ZHOU Junjie, LUO Lu, FENG Na*, MA Ai-Jun*

    Chinese Journal of Synthetic Chemistry, 2022, 30, 893-901.


    12 Total synthesis of bi-magnolignan

    Si-Yuan Lu(卢思远), Hong-Mei Wang, Na Feng* and Ai-Jun Ma*

    RSC Adv., 2023, 13, 8844-8846. 



    11 Studies toward synthesis of the core skeleton of spiroaspertrione A

    Zhong-Hui Shen(沈中辉), Si-Yuan Lu, Jing-Yun Zheng, Xiang-Zhi Zhang, Jin-Bao Peng, Ai-Jun Ma*

    Frontiers in Chemistry2022, doi:10.3389/fchem.2022.1022533


    10 Synthesis of melatonin derivatives and the neuroprotective effects in Parkinson's disease models of Caenorhabditis elegans

    Li He(贺利), Jing-Jing Du, Meng-Ting Chen, Jun-Jie Zhou, Lu Luo, Baoqiong Li, Xiang-Zhi Zhang, Wen-Zhe Ma, Ai-Jun Ma*, Na Feng*

    Frontiers in Chemistry, 2022, doi:10.3389/fchem.2022.918116.


    9 Intramolecular Aerobic Ring Expansion of Cyclic Ketone: A Mild Method for the Synthesis of Medium-Sized Lactones and Macrolactones

    Qi-Ming Liang(梁绮明),Jing-Yun Zheng, Si-Yuan Lu, Hong-Mei Wang, Lu Luo, Xiang-Zhi Zhang, Jin-Bao Peng, Na Feng, Ai-Jun Ma*

    Advanced Synthesis & Catalysis, 2022364, 2152-2156.  (Featured in Org. Chem. Highlights)


    8 Synthesis of disubstituted γ-butyrolactones and spirocyclopropanes via a multicomponent reaction of aldehydes, Meldrum’s acid and sulfoxonium ylides

    Shan-Shan Li(李汕珊), Qi Qin, Zhuang Qi, Li-Miao Yang, Yun Kang, Xiang-Zhi Zhang, Ai-Jun Ma* and Jin-Bao Peng *

    Org. Chem. Front., 2021, 8, 3069-3075.

     

    7 Synthesis of Cinnamic Acid Ester Derivatives of Chrysin

    CHEN Han-qia(陈汉洽), YANG Meng-yuan, WEI Dong-mei, HE Li, ZHENG Jing-yun, LI Jie-fang, ZHONG Hao-liang, FENG Na, MA Ai-jun*, ZHANG Shu-yu*, ZHANG Kun*

    Chin. J. Syn. Chem. 2020, 28, 848-854.

     

    6 Recent Progress in Synthesis of Polysubstituted Pyrazoles

    Wang, Shaohua, Zhang, Banghong, Chen, Jie, Zheng, Yingying, Feng, Na, Ma, Aijun*, Xu, Xuetao*, Abdullah, M. Asirid

    Chin. J. Org. Chem. 2020, 40, 15-27.

     

    5 Synthesis and biological evaluation of coumarin derivatives as aglucosidase inhibitors

    Xue-Tao Xu, Xu-Yang Deng, Jie Chen, Qi-Ming Liang, Kun Zhang, Dong-Li Li, Pan-Pan Wu, Xi Zheng, Ren-Ping Zhou, Zheng-Yun Jiang, Ai-Jun Ma*, Wen-Hua Chen*, Shao-Hua Wang*

    Eur. J. Med. Chem. 2020, 189, 112013.

     

    4 Synthetic Studies on the Kigamicins

    Ai-Jun Ma and Joseph M. Ready*

    Org. Lett. 2019, 21, 11481151.

     

    Before 2018

    3 Synthesis and Biological Evaluation of Kibdelone C and Its Simplified Derivatives

    Janjira Rujirawanich, Soyeon Kim, Ai-Jun Ma, John R. Butler, Yizhong Wang, Chao Wang, Michael Rosen, Bruce Posner, Deepak Nijhawanc, and Joseph M. Ready*

    J. Am. Chem. Soc. 2016, 138, 10561-10570.

     

    2 Total Synthesis of the Nominal Didemnaketal A

    Fu-Min Zhang, Lei Peng, Hui Li, Ai-Jun Ma, Jin-Bao Peng, Jing-Jing Guo, Dengtao Yang, Si-Hua Hou, Yong-Qiang Tu*, and William Kitching

    Angew. Chem. Int. Ed. 2012, 51, 10846-10850.

     

    1 Total Synthesis of (-)-FR901483

    Ai-Jun Ma, Yong-Qiang Tu*, Jin-Bao Peng, Qing-Yun Dou, Si-Hua Hou, Fu-Min Zhang, and Shao-Hua Wang

    Org. Lett. 2012, 14, 3604–3607.


    其他合作论文

            34 Discovery of Bi-magnolignan as a novel BRD4 inhibitor inducing apoptosis and DNA damage for cancer therapy

            Zifeng Huang, Tong Chu, Aijun Ma, Wanjun Lin, Yan Gao, Na Zhang, Meina Shi, Xuening Zhang, Yanchao Yang, Wenzhe Ma

            Biochemical Pharmacology, 2025, 235, 116843. 


          33 Synthesis of The Key Heptapeptide Fragment for Marine Cyclotide Portobelamide A

          HE Wangjin, CHEN Yuanying, HUANG Lifeng, MA Aijun, YAN Jialei*

          Chin. J. Syn. Chem., 2025, 33, 254.


        32 Remote Stereocontrol in C6-Functionalization of Indoles via Synergistic Ion-Pair Catalysis

        Zhi-Qiang Zhu, Han-Peng Pan, Liang Long, Ze-Yu Su, Ai-Jun Ma, Jin-Bao Peng, Hao Gao, Guo-Dong Chen*, Yong-Heng Wang*, Xiang-Zhi Zhang*

        ACS Catalysis2025, 10.1021/acscatal.5c00780.


      31 Discovery of Bi-magnolignan as a novel BRD4 inhibitor inducing apoptosis and DNA damage for cancer therapy

      Zifeng Huang, Tong Chu, Aijun Ma, Wanjun Lin, Yan Gao, Na Zhang, Meina Shi, Xuening Zhang, Yanchao Yang, Wenzhe Ma*

      Biochemical Pharmacology2025, 116843


                    30 Lewis-Acid-Catalyzed (3+2) Annulation of 2-Indolylmethanols with Propargylic Alcohols to Access Cyclopenta[b]indoles

                    Teng-Fei Wu, Zhao-Jie Fu, Yi-Rui Zhang, Zong-Wang Qiu, Bao Qiong Li*, Shao-Shuai Chen, Han-Peng Pan, Ai-Jun Ma and Xiang-Zhi Zhang* 

                    Molecules, 2024, 29, 1251. 

                           

                    29 Melatonin derivative 6a protects Caenorhabditis elegans from formaldehyde neurotoxicity via ADH5         
                    Meng-Ting Chen, Jun-Jie Zhou, Rui-Ting Han, Qing-Wei Ma, Zi-Jie Wu, Peng Fu,                                          Ai-Jun Ma                                         , Na Feng*              
                    Free Radical Biology and Medicine                                         ,                                         2024                                         ,                                         223                                         , 57–368.  
                      28 Ni-Catalyzed Enantioselective Reductive Cross- and Homo-Coupling of Aryl Electrophiles: Synthesis of Axially Chiral Diaryl Dicarboxylates        
                      Ye Zhang, Yun-Zhou Gu, Ka Lu, Yun-Peng Wang, Ai-Fang Wang, Shuang-Hu Wang, Shi-Qiang Wei, Fu-Min Zhang, Xiao-Ming Zhang, Ai-Jun Ma, Jin-Bao Peng & Yong-Qiang Tu*        
                      CCS Chem.,                                          2024                                         7, 1067–1077. 
                      27 Enantioselective synthesis of α,α-diarylketones by sequential visible light photoactivation and phosphoric acid catalysis        

                Hong-Fu Liu, Liang Long, Zhi-Qiang Zhu, Teng-Fei Wu, Yi-Rui Zhang, Han-Peng Pan,Ai-Jun Ma, Jin-Bao Peng, Yong-Heng Wang, Hao Gao*, Xiang-Zhi Zhang*

                Sci. Adv., 20239, eadg7754.


              26 Photoinduced reductive Reformatsky reaction of a-haloesters and aldehydes or ketones by cooperative dual-metal catalysis

              Qi-Long Chen, Le Mao, Yi-Fan Pan, Heng Cai, Xiao-Ming Zhang,* Fu-Min Zhang,  Ai-Jun Ma,  Jin-Bao Peng  and Yong-Qiang Tu 

              Chem. Commun., 2023, 59, 14427–14430.


              25 Catalytic Asymmetric Syntheses of 2,5-Diketopiperazine (DKP) Frameworks

              Ju-Song Yang, Fu-Min Zhang,* Ai-Jun Ma, Jin-Bao Peng, Kun Zhang, Xiao-Ming Zhang,* and Yong-Qiang Tu*

              Asian J. Org. Chem., 2023, 12, e202300177.


              24 Molybdenum-Mediated Reductive Hydroamination of Vinylcyclopropanes with Nitroarenes: Synthesis of Homoallylamines

              Jin-Liang Lu, Zhi Zhang, Jing-Tong Deng, Ai-Jun Ma, and Jin-Bao Peng*

              Org. Lett., 2023, 25, 2991–2995.


              23 Bismuth(III)-Catalyzed 1,8-Addition/Cyclization/Rearrangement of Propargylic para-Quinone Methides with 2Vinylphenol: Synthesis of Indeno[2,1c]chromenes

              Zhi-Qiang Zhu, Teng-Fei Wu, Han-Peng Pan, Jin-Bao Peng, Ai-Jun Ma, and Xiang-Zhi Zhang*

              Org. Lett.,2023, 25, 1299–1304.


            22 Base-promoted [4 + 2] annulation of pyrrole-2- carbaldehyde derivatives with β,γ-unsaturated α-ketoesters: syntheses of 5,6-dihydroindolizines

            You-Ya Zhang, Lin Li, Ai-Jun Ma, Wei-Feng Wang* and Jin-Bao Peng* 

            Org. Biomol. Chem., 202220, 8633.


            21 Mitochondrial toxicity evaluation of traditional Chinese medicine injections with a dual in vitroapproach

            Yunfu Shen, Kaiqiang Guo, Ai-Jun Ma, Zhe Huang1, Jingjing Du, Junhe Chen, Qianyu Lin, Chengming Wei, Zi Wang, Fuming Zhang, Juan Zhang, Wanjun Lin, Na Feng* and Wenzhe Ma*

            Front. Pharmacol., 2022, 13, 1039235.


            20 Palladium-Catalyzed Nucleophilic Reaction of Alkylidenecyclopropanes with β,γ-Unsaturated α‑Ketoesters: Ligand-Controlled Divergent Synthesis

            Xin-Lian Liu, You-Ya Zhang, Lin Li, Lu-Qi Tan, Yin-Ai Huang, Ai-Jun Ma, and Jin-Bao Peng*

            Org. Lett., 2022, 24, 6692−6696.


            19 Palladium Catalyzed Dicarbonylation of α‑Iodo-Substituted Alkylidenecyclopropanes: Synthesis of Carbamoyl Substituted Indenones

            Lin Li, Xin-Lian Liu, Jin-Yan Liang, Yong-Yu He, Ai-Jun Ma, Wei-Feng Wang,* and Jin-Bao Peng*

            Org. Lett., 2022, 24, 5624−5628.


            18 Palladium-Catalyzed Carbonylative Sonogashira/Annulation Reaction: Synthesis of Indolo[1,2‑b]isoquinolines

            Lin Li, Xin-Lian Liu, Zhuang Qi, Ai-Hua Yang, Ai-Jun Ma, and Jin-Bao Peng*

            Org. Lett., 2022, 24, 1201−1206.


            17 Asymmetric Three-Component Reaction to Assemble the Acyclic All Carbon Quaternary Stereocenter via Visible Light and Phosphoric Acid Catalysis

            Zong-Wang Qiu, Liang Long, Zhi-Qiang Zhu, Hong-Fu Liu, Han-Peng Pan, Ai-Jun Ma, Jin-Bao Peng, Yong-Heng Wang, Hao Gao,* and Xiang-Zhi Zhang*

            ACS Catal., 2022, 12, 13282−13291.


            16 Visible-Light-Induced Carbonylation of Indoles with Phenols under Metal-Free Conditions: Synthesis of Indole-3-carboxylates

            Zhuang Qi, Lin Li, Ying-Kang Liang, Ai-Jun Ma, Xiang-Zhi Zhang, and Jin-Bao Peng*

            Org. Lett.2021, 23, 4769−4773.


            15 Remote asymmetric conjugate addition catalyzed by a bifunctional spiro-pyrrolidine-derived thiourea catalyst

            Ming-Hui Xu, Yong-Hai Yuan, Dong-Dong Liang, Xiao-Ming Zhang,* Fu-Min Zhang, Yong-Qiang Tu,* Ai-Jun Ma, Kun Zhang and Jin-Bao Peng

            Org. Chem. Front., 2021, 8, 3292–3297.


            14 Brønsted Acid-Catalyzed Formal (3+3)-Annulation of Propargylic (Aza)-para-Quinone Methides with 4‑Hydroxycoumarins and 1,3- Dicarbonyl Compounds

            Zong-Wang Qiu, Xue-Tao Xu, Han-Peng Pan, Zhen-Sheng Jia, Ai-Jun Ma, Jin-Bao Peng, Ji-Yuan Du, Na Feng, Bao Qiong Li, and Xiang-Zhi Zhang*

            J. Org. Chem., 2021, 86, 6075−6089.


            13 Formal (3 + 4)-Annulation of Propargylic pQuinone Methides with 2Indolylmethanols: Synthesis of Polysubstituted Indole-Fused Oxepines

            Zong-Wang Qiu, Bao Qiong Li, Hong-Fu Liu, Zhi-Qiang Zhu, Han-Peng Pan, Na Feng, Ai-Jun Ma, Jin-Bao Peng, and Xiang-Zhi Zhang*

            J. Org. Chem., 2021, 86, 74907499.


          12 Development and validation of ultra-high performance supercritical fluid chromatography method for quantitative determination of six compounds in Guizhi Fuling capsule and tablet samples

          Bao Qiong Li, Xin Kang Li, Yuan Lin, Ze Ying Li, Xiang-Zhi Zhang, Na Feng, Ai-Jun Ma, Chao Yang, Chen Lin, Fan Tan

          J. Sep. Sci.2021, 44, 3199–3207.


            11 Palladium Catalyzed Cascade Azidation/Carbonylation of Aryl Halides with Sodium Azide for the Synthesis of Amides 

            Zhuang Qi, Shan-Shan Li, Lin Li, Qi Qin, Li-Miao Yang, Ying-Kang Liang, Yun Kang, Xiang-Zhi Zhang, Ai-Jun Ma, and Jin-Bao Peng*

            Chem Asian J.2021, 16, 503 –506.


            10 Unprecedented Multicomponent Reaction of Indoles, CS2 and Nitroarenes: Stereoselective Synthesis of (Z)-3-((Arylamino) methylene)indoline-2-thiones

            Qi Qin, Xin-Lian Liu, Ai-Jun Ma, Xiang-Zhi Zhang,* and Jin-Bao Peng*

            Chem Asian J.2021, 16, 3890–3894.


            9 Oxidative [3+2] Annulation of Pyridinium Salts with gemDifluoroalkenes: Synthesis of 2-Fluoroindolizines

            Li–Miao Yang, You-Ya Zhang, Jing-Tong Deng, Ai-Jun Ma, Xiang-Zhi Zhang, Shu-Yu Zhang,* and Jin-Bao Peng*

            Asian J. Org. Chem., 2021, 10, 1679-1682.


            8 Palladium Catalyzed Aminocarbonylation of Benzylic Ammonium Triflates with Nitroarenes: Synthesis of Phenylacetamides

            Li-Miao Yang, Shan-Shan Li, You-Ya Zhang, Jin-Liang Lu, Jing-Tong Deng, Ai-Jun Ma, Xiang-Zhi Zhang, Shu-Yu Zhang,* and Jin-Bao Peng,*

            Adv. Synth. Catal., 2021, 363, 2061– 2065.


        7 Synthesis of Pyrrolo[1,2-a]indoles via (3+2)-Annulations of (Aza)-para-Quinone Methides with Indoles

        Xiang-Zhi Zhang*, Zong-Wang Qiu, Gui-Hua Wen, Ai-Jun Ma, Peng-Jin Bao, Ji-Yuan Du, Xue-Tao Xu, Na Feng, Bao Qiong Li*

        Synthesis, 2020, 52, 3640-3649.


        Diastereoselective Synthesis of Cycloheptannelated Indoles via Lewis-Acid-Catalyzed (4 + 3)-Cyclization of DonorAcceptor Cyclopropanes

        Bao Qiong Li, Zong-Wang Qiu, Ai-Jun Ma, Jin-Bao Peng, Na Feng, Ji-Yuan Du, Han-Peng Pan, Xiang-Zhi Zhang,* and Xue-Tao Xu*

        Org. Lett., 2020, 22, 1903–1907.


      5 A dienamine-mediated deconjugative addition/ cyclization cascade of γ,γ-disubstituted enals with carboxylic acid-activated enones: a rapid access to highly functionalized γ-lactones

      Wei Jiang, Jia Zhou, Ai-Jun Ma, Dongli Li,  Yan-Yan Ma, Deng-Gao Zhao, Si-Hua Hou, Jun-Bing Lin*, Shu-Yu Zhang*

      Org. Chem. Front., 2020, 7, 571.


      4 Facile access to diverse all-carbon quaternary center containing spirobicycles by exploring a tandem CastroStephens coupling/acyloxy shift/ cyclization/semipinacol rearrangement sequence

      Ye Zhang, Tian-Lu Zheng, Fu Cheng, Kun-Long Dai, Kun Zhang, Ai-Jun MaFu-Min Zhang, Xiao-Ming Zhang,  Shao-Hua Wang*band Yong-Qiang Tu*

      Chem. Sci., 2020, 11, 3878.


      3 N-way partial least squares combined with new self-construction strategy—A promising approach of using near infrared spectral data for quantitative determination of multiple compounds

      Xiang-Zhi Zhang, Ai-Jun Ma, Na Feng and Bao Qiong Li*

      Journal of Near Infrared Spectroscopy, 2019, 28, 113 - 121.


      2 A catalytic asymmetric one-pot [3+2] cyclization/semipinacol rearrangement sequence: an efficient construction of a multi-substituted 3H-spiro[benzofuran-2,10-cyclopentane] skeleton

      Lin Liu, Lin-Sheng Lei, Zong-Song Zhan, Si-Zhan Liu, Yu-Xiao Wang,Yong-Qiang Tu,* Fu-Min Zhang,  Xiao-Ming Zhang, Ai-Jun Ma and Shao-Hua Wang*

      Chem. Commun., 201955, 3789.


        1 Cascade Oxidative Dearomatization/Semipinacol Rearrangement: An Approach to 2-Spirocyclo-3-oxindole Derivatives

        Jin-Bao Peng, Yue Qi, Ai-Jun Ma, Yong-Qiang Tu,* Fu-Min Zhang, Shao-Hua Wang, and Shu-Yu Zhang*

        Chem. Asian J., 2013, 8, 883 – 887.


      【授权发明专利

      11 马爱军;郑景云;罗颖;冯娜 “一种喹啉衍生物及其制备方法”,2025.07.11(授权),中国,ZL202310195220.3

      10 冯娜马爱军;卢思远 “一种联二厚朴脂素的制备方法”,2025.06.13(授权),中国,ZL202310342265.1

      马爱军;刘振伟;白瑞异;冯娜 “一种四环内酰胺类化合物及其制备方法”,2025.05.30(授权),中国,ZL202310532300.3

      马爱军;林思武;赵丽丽;李汕珊;冯娜 “一种苯并[6,6]-螺环缩酮化合物的制备方法”,2025.05.27(授权),中国,ZL202310075818.5

      马爱军;王红梅;梁绮明;冯娜 “一种羧酸类化合物及其制备方法与应用”,2024.09.24(授权),中国,ZL202310103680.9

      陈霞马爱军;师建毅;陈修文;朱忠智 “一种金鸡纳碱衍生物及其制备方法和应用”,2024.03.26(授权),中国,ZL202211233912.4

      马爱军;李汕珊;赵丽丽;潘敏;冯娜;陈春灵;游松涛 “一种苯并吡喃类化合物及其制备方法”,2024.01.12(授权),中国,ZL202210881947.2 

      马爱军;贺利;朱瑞焘;周俊杰;陈梦婷;文慧心;罗路;冯娜 “一种褪黑激素肉桂酸衍生物及其制备方法”,2023.07.04(授权),中国,ZL202210518275.9 

      冯娜;贺利;杨梦圆;韦冬梅;马爱军 一种白杨素肉桂酸酯或其衍生物及其制备方法”,2023.02.17(授权),中国,ZL 202010891873.1

      马爱军;梁绮明;欧婷婷;郑景云;李凤萍;卢思远;冯娜;陈春灵;游松涛 “2-乙基-3,4-二氢-1(2H)-异喹啉酮的制备方法”,2022.6.21(授权),中国,ZL202110688971.X

      涂永强马爱军 “一种免疫抑制剂FR901483中间体及其合成方法2015.2.18(授权),中国,CN102643276B



      教学

      中国大学慕课《药物化学》

      《药物化学》是一门发现与发明新药、合成化学药物、阐明药物化学性质、研究药物分子与机体细胞(生物大分子)之间相互作用规律的综合性学科,是药学领域中重要的带头学科。本课程由大湾区九所高校十名老师共同倾力打造!采九校之石可以攻玉,纳十师之长可以厚己。一起学习《药物化学》,走近新药梦开始的地方。 —— 课程团队