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成果及论文

  1. Zhou, Y.; Lei, S. G.; Abudureheman, B.; Wang, L. S.; Yu, Z. C.; Xiang, J. C.; Wu, A. X. Transforming an Azaarene into the Spine of Fusedbicyclics via Cycloaddition-induced Scaffold Hopping of 5-Hydroxypyrazoles. Nat. Commun. 2024, 15, 10907.

  2.  Wang, L. S.; Song, Y. M.; Zhou, Y.; Tang, Y. X.; Wu, C. Y.; Yu, Z. C.; Zhou, H.; Zheng, K. L.; Wu, A. X. Iodine as Polarity-Reversal Catalyst: Synthesis of a Fused Heterocycle with Contiguous Stereocenters. Org. Lett. 2024, 27, 91-96. 

  3. Yang, D. S.; Xiang, J. C.; Wu, A. X. Recent Advances in the Synthesis of N-heterocycles from Α-amino Acids Mediated by Iodine. Chem. Commun. 2024, 60, 14318-14331. 

  4.  Du, Y. D.; Wang, J. G.; Liu, J. Y.; Wu, C. Y.; Hu, R. F.; Wu, A. X. I2–DMSO-mediated Formal [3 + 1 + 2] Synthesis of Pyrimido[1,2-b]indazole Using 1,4-dithiane-2,5-diol as a Surrogate of Ethylene. Tetrahedron Lett. 2025, 156, 155453. 

  5.  Yang, D. S.; Chen, X. L.; Wu, C. Y.; Zhou, Y.; Wang, L. S.; Wu, Y. D.; Wu, A. X. Intramolecular/Intermolecular Sequential Cyclization Accompanied by Double C–F Bond Cleavage: Access to Tricyclic Fluorine-Containing Pyrano[3,2-c]chromenes. J. Org. Chem. 2024, 89, 16553-16563. 

  6.  Du, Y. D.; Ma, L. L.; Wu, C. Y.; Wu, R. H.; Yu, Z. C.; Zhou, Y.; Yang, D. S.; Wu, Y. D.; Wang, J. G.; Wu, A. X. Synthesis of 6-oxa-Spiro [4.5]decane Derivatives by Merging Ring-Opening of Benzo[c]oxepines and Formal 1,2-Oxygen Migration. J. Org. Chem. 2024, 89, 15953-15963. 

  7. Wang, L. S.; Xiang, J. C.; Wu, A. X. Advances in the Self-organized Total Synthesis of Natural Products. Chem. Commun. 2024, 60, 12803-12815. 

  8.  Wu, C. Y.; Chen, X. L.; Yang, D. S.; Tang, Y. X.; Wang, L. S.; Du, Y. D.; Wu, Y. D.; Wu, A. X. Difluorocarbene-Enabled Trifluoromethylation and Cyclization for the Synthesis of 3-(Trifluoromethyl)-4H-pyrans. Org. Lett. 2024, 26, 8589-8593. 

  9. Yu, Z. C.; Zheng, K. L.; Shen, X.; Zhou, Y.; Chen, X. L.; Wang, L. S.; Wu, Y. D.; Wu, A. X. I2-Induced Umpolung: Synthesis of a 1,6-Dihydrofuro[3,2-b]pyrazolo[3,4-e][1,4]thiazine Skeleton via an Unconventional 1,4-Dithiane-2,5-diol Reaction Mode. Org. Lett. 2024, 26, 7891-7896. 

  10.  Tang, Y. X.; Wu, A. X. Research Progress of Self-organized Reaction Networks for Cascade Reactions. Tetrahedron 2024, 166, 134210. 

  11.  Wang, M.; Ren, H. Y.; Pu, X. Y.; Zhang, X. L.; Zhu, H. Y.; Wu, A. X.; Zhao, B. T. Rongalite/iodine-mediated C(sp3)–H Bond Oximation and Thiomethylation Reaction of Methyl Ketones Using Copper Nitrate as the [NO] Reagent: Synthesis of Thiohydroximic Acids. Org. Biomol. Chem. 2024, 22, 7623-7627. 

  12. Shen, X.; Yu, Z. C.; Zhou, Y.; Wu, Y. D.; Wu, A. X. Divergent Synthesis of Pyrrolidone Fused Pyrimido[1,2-b]indazole Through Selective Trapping of an Enone Intermediate by 1H-indazol-3-amine. Chem. Commun. 2024, 60, 9781-9784. 

  13.  Song, Y. C.; Cao, W. H.; Wang, M. X.; Wang, R. Q.; Sun, Y. Y.; Wu, A. X.; Zhu, Y. P. One-Pot Total Synthesis of Natural Products Nitramarine, Nitraridine, and Analogues via a Cascade Oxidation/Pictet–Spengler Condensation/Annulation Process. J. Org. Chem. 2024, 89, 12832-12841. 

  14.  Shen, X.; Yu, Z.; Zhou, Y.; Wu, Y.; Wu, A. One‐Pot Synthesis of 3‐Hydroxy‐1H‐Pyrrolo[3,4‐b]quinolin‐1‐one via Enaminamides. Adv Synth Catal 2024, 366, 4399-4403. 

  15. Tang, Y. X.; Zhou, Y.; Wu, H. X.; Wang, L. S.; Wu, C. Y.; Zhuang, S. Y.; Wu, A. X. N-Benzylhydroxylamine as a Novel Synthetic Block in “C1N1” Embedding Reaction via Α-C(sp3)–H Activation Strategy. Chem. Commun. 2024, 60, 7180-7183. 

  16.  Wu, C. Y.; Chen, X. L.; Yang, D. S.; Tang, Y. X.; Wang, L. S.; Wu, Y. D.; Zhuang, S. Y.; Wu, A. X. Base-controlled Selective Cleavage of the C–F Bond of Difluorocarbene for the Divergent Assembly of Indolizines. Org. Chem. Front. 2024, 11, 4214-4218. 

  17.  Yang, D. S.; Chen, X. L.; Wu, C. Y.; Tang, B. C.; Xiao, Y. C.; Wu, Y. D.; Wu, A. X. Synthesis of Β,β-Dithioketones by Merging C–C and C–S Bond Cleavage in [1 + 1 + 1 + 1 + 1 + 1] Annulation. Org. Lett. 2024, 26, 4340-4345. 

  18.  Yu, Z.; Shen, X.; Zhou, Y.; Chen, X.; Wang, L.; Wu, Y.; Wu, A. I2–DMSO‐Mediated Multicomponent [2+1+1+1] Annulation Reaction via Ethyl Nitroacetate C—NO2 Bond Cleavage as a C1Synthon: A Route to Multisubstituted β‐Pyrrolidinones Derivatives with a Quaternary Center. Chin. J. Chem. 2024, 42, 2029-2034. 

  19.  Xiang, J. C.; Wang, Y. D.; Yuan, P.; Zhu, H. M.; Lei, T.; Wu, A. X.; Liao, Z. Diverting the Mannich Reaction to Access 2,2-disubstituted Indolin-3-ones by Merging 1,2-aryl Migration and Copper-catalyzed Aerobic Oxidation. Org. Chem. Front. 2024, 11, 3186-3195. 

  20.  Yang, D. S.; Chen, X. L.; Wu, A. X. Review of Application of the I2 and Dimethyl Sulfoxide Combined Reagent System to Aryl Methyl Ketones for Diverse Transformations. Org. Chem. Front. 2024, 11, 2665-2692. 

  21.  Zhou, Y.; Wang, L. S.; Lei, S. G.; Tang, B. C.; Yu, Z. C.; Li, X.; Wu, Y. D.; Zheng, K. L.; Wu, A. X. I2-DMSO Mediated Tetra-functionalization of Enaminones for the Construction of Novel Furo[2′,3′:4,5]pyrimido[1,2-b]indazole Skeletons via in Situ Capture of Ketenimine Cations. Chin. Chem. Lett. 2025, 36, 109799. 

  22. Cai, Q.; Si, M. J.; Shi, X. R.; Liao, M.; Liu, F. C.; Wang, M.; Li, K. X.; Chen, Y. T.; Wu, A. X. Copper-catalyzed Selective Construction of Vinyl Sulfones Employing TosMIC as a C1 Synthon and Sulfone Source. Org. Chem. Front. 2024, 11, 2528-2533. 

  23. Ma, L. L.; Zhou, Y.; Tang, Y. X.; Chen, T.; Wang, Z. H.; Wu, Y. D.; Wang, J. G.; Wu, A. X. I2-DMSO-Mediated Construction of 2,3- and 2,4-Disubstituted Pyrimido[1,2-b]indazole Skeletons. J. Org. Chem. 2024, 89, 3941-3953. 

  24. Chen, X.; Wu, C.; Yang, D.; Tang, B.; Wang, H.; Yu, Z.; Li, A.; Wu, Y.; Wu, A. Transition‐Metal‐Free Allylic Defluorination Cross‐Electrophile Coupling Employing Rongalite. Chin. J. Chem. 2024, 42, 1360-1366. 

  25.  Zhao, P.; Zhou, Y.; Wang, C.; Wu, A. X. Iodine-Promoted Thioylation and Dicarbonylation of Enaminone Α-C Sites: Synthesis of Fully Substituted Thiazoles via C═C Bond Cleavage. J. Org. Chem. 2024, 89, 2505-2515. 

  26.  Song, Y.; Wang, M.; Yi, Y.; Liu, Y.; Zhang, W.; Wang, Z.; Sun, Y.; Wu, A.; Zhu, Y. FeCl<sub>3</sub>/KI‐Catalyzed Tandem Oxidative Cyclization for Switchable Total Synthesis of Luotonin A, B and Derivatives. Adv Synth Catal 2024, 366, 1348-1355. 

  27.  Li, M.; Wan, Q. Y.; Lin, R. L.; Peng, Y. Q.; Shu, W. M.; Yu, W. C.; Wu, A. X. Azide-free Cyclization Reaction Access to 4-aryl-NH-1,2,3-triazoles: P-toluenesulfonyl Hydrazide and Sulfamic Acid as Nitrogen Sources. Org. Biomol. Chem. 2024, 22, 482-485. 

  28.  Yu, Z. C.; Shen, X.; Zhou, Y.; Chen, X. L.; Wang, L. S.; Wu, Y. D.; Zhang, H. K.; Zheng, K. L.; Wu, A. X. I2-promoted Formal [3 + 1 + 1 + 1] Cyclization to Construct 5-cyano-1H-pyrazolo[3,4-b]pyridine Using Malononitrile as a C1 Synthon. Org. Chem. Front. 2023, 10, 5958-5964. 

  29.  Wang, H. Y.; Chen, X. L.; Wu, C. Y.; Yang, D. S.; Chen, T.; Wu, A. X. Reductive N-Formylation of Nitroarenes Mediated by Rongalite. Org. Lett. 2023, 25, 7220-7224. 

  30. Lei, S. G.; Zhou, Y.; Wang, L. S.; Yu, Z. C.; Chen, T.; Wu, Y. D.; Gao, M.; Wu, A. X. I2-DMSO Mediated Dual Α,β-C(sp2)–H Functionalization/bicyclization of o-hydroxyphenyl Enaminones to Construct C2,C3-disubstituted Chromone Derivatives: Chromeno[2,3-b]pyrrol-4(1H)-ones. Org. Chem. Front. 2023, 10, 4843-4847. 

  31.  Liu, J. Y.; Zhuang, S. Y.; Tang, Y. X.; Chen, X. L.; Zhou, Y.; Wu, Y. D.; Zheng, K. L.; Wu, A. X. I2-DMSO-Mediated Transannulation of Benzo[d]isoxazol-3-amine: Direct Access to 2,4,5-Substituted Pyrimidine Derivatives. J. Org. Chem. 2023, 88, 12000-12012. 

  32.  Yuan, P.; Liu, R.; Zhu, H. M.; Liao, Z.; Xiang, J. C.; Wu, A. X. An I2–DMSO Catalytic Manifold Enabled Aromatization for C-ring Editing of Podophyllotoxone. Org. Biomol. Chem. 2023, 21, 6468-6473. 

  33.  Wang, L.; Zhou, Y.; Lei, S.; Tang, B.; Yu, Z.; Tang, Y.; Wu, Y.; Wu, A. Direct Introduction of −OCD3 into the Hantzsch Pyrrole Synthesis via Multicomponent Cascade Cyclization: Synthesis of Fully Substituted Pyrrole Derivatives. Adv Synth Catal 2023, 365, 2888-2893. 

  34. Lei, S. G.; Zhou, Y.; Wang, L. S.; Yu, Z. C.; Chen, T.; Wu, Y. D.; Gao, M.; Wu, A. X. One Stone, Three Birds: One-Pot Synthesis of Pyrido[3,2-a]phenoxazin-5-one Derivatives from o-Aminophenols with Triple Roles, Paraformaldehyde, and Enaminones via the Povarov Reaction. J. Org. Chem. 2023, 88, 11150-11160. 

  35. Wang, M.; Jiang, S.; Lu, X. X.; Zhang, K.; Yuan, Z. Y.; Xu, R. L.; Zhao, B. T.; Wu, A. X. Synthesis of Primary Propargylic Alcohols from Terminal Alkynes Using Rongalite as the C1 Unit. Org. Biomol. Chem. 2023, 21, 5949-5952. 

  36.  Chen, T.; Ma, J. T.; Chen, X. L.; Zhou, Y.; Yu, Z. C.; Lei, S. G.; Wu, Y. D.; Xiang, J. C.; Wu, A. X. Modular and Selective Synthesis of Pyrazolo-azepino-centred Polycyclic Aromatic and Non-aromatic Architectures. Org. Chem. Front. 2023, 10, 4122-4130. 

  37. Tang, Y. X.; Zhuang, S. Y.; Liu, J. Y.; Zhou, Y.; Wang, L. S.; Wu, Y. D.; Wu, A. X. I2–DMSO Mediated Multicomponent Convergent Synthesis of Imidazo[2,1a]isoquinoline Derivatives via a Triple in Situ Cross-trapping Strategy. Org. Chem. Front. 2023, 10, 4080-4085. 

  38.  Wang, H.; Chen, X.; Wu, Y.; Wu, A. Rongalite as a Versatile Reagent in Organic Synthesis†. Chin. J. Chem. 2023, 41, 3388-3400. 

  39.  Yu, Z. C.; Shen, X.; Zhou, Y.; Ma, J. T.; Chen, X. L.; Wang, L. S.; Wu, Y. D.; Wu, A. X. Successive Promotion of Formal [3+2] Cycloaddition of Aryl Methyl Ketones by I2and Zn: Access to 2-Hydroxy-4-morpholin-2,5-diarylfuran-3(2H)-ones with a Quaternary Carbon Center. J. Org. Chem. 2023, 88, 9321-9331.

  40.  Wu, C. Y.; Chen, X. L.; Wang, H. Y.; Yang, D. S.; Zhuang, S. Y.; Zhou, Y.; Yu, Z. C.; Wu, Y. D.; Geng, X.; Wu, A. X. Dual Role of BrCF2CO2Et: Difluorocarbene-enabled Access to Α-trifluoromethyl Ketones from Sulfoxonium Ylides. Org. Chem. Front. 2023, 10, 3741-3745. 

  41.  Zhou, Y.; Lei, S. G.; Wang, L. S.; Ma, J. T.; Yu, Z. C.; Wu, Y. D.; Wu, A. X. I2-Promoted gem-Diarylethene Involved Aza-Diels–Alder Reaction and Wagner–Meerwein Rearrangement: Construction of 2,3,4-Trisubstituted Pyrimido[1,2-b]indazole Skeletons. Org. Lett. 2023, 25, 3386-3390. 

  42. Chen, X. L.; Yang, D. S.; Tang, B. C.; Wu, C. Y.; Wang, H. Y.; Ma, J. T.; Zhuang, S. Y.; Yu, Z. C.; Wu, Y. D.; Wu, A. X. Direct Hydrodefluorination of CF3-Alkenes via a Mild S<sub>N</sub>2′ Process Using Rongalite as a Masked Proton Reagent. Org. Lett. 2023, 25, 2294-2299. 

  43.  Ma, J. T.; Chen, T.; Tang, B. C.; Chen, X. L.; Yu, Z. C.; Zhou, Y.; Zhuang, S. Y.; Wu, Y. D.; Xiang, J. C.; Wu, A. X. A Pummerer Reaction-Enabled Modular Synthesis of Alkyl Quinoline-3-carboxylates and 3-Arylquinolines from Amino Acids. J. Org. Chem. 2023, 88, 3760-3771. 

  44. Ma, J. T.; Chen, T.; Chen, X. L.; Zhou, Y.; Yu, Z. C.; Zhuang, S. Y.; Wu, Y. D.; Xiang, J. C.; Wu, A. X. Aniline Assisted Dimerization of Phenylalanines: Convenient Synthesis of 2-aroyl-3-arylquinoline in an I2-DMSO System. Org. Biomol. Chem. 2023, 21, 2091-2095. 

  45.  Zhuang, S. Y.; Liu, J. Y.; Guo, H.; Tang, Y. X.; Chen, X. L.; Ma, J. T.; Wu, Y. D.; Wu, A. X.; Zheng, K. L. I2-DMSO Mediated Multicomponent [3+2] Annulation Reaction: An Approach to Pyrrolo[2,1-a]isoquinoline Derivatives with a Quaternary Center. Org. Lett. 2022, 24, 8573-8577. 

  46.  Xiang, J. C.; Wang, J. W.; Yuan, P.; Ma, J. T.; Wu, A. X.; Liao, Z. X. Switching Over of the Chemoselectivity: I2-DMSO-Enabled Α,α-Dichlorination of Functionalized Methyl Ketones. J. Org. Chem. 2022, 87, 15101-15113. 

  47. Hu, Y.; Wang, Z.; Xiang, J.; Ma, J.; Lin, R.; Wang, J.; Wu, A. Synthesis of Polysubstituted Phenols via [3+3] Condensation Reaction from Tricarbonyl Compounds and Readily Available Enaminones, Cinnamaldehydes or Arylformyl Trifluoroacetones. Tetrahedron 2022, 128, 133124. 

  48. Zhao, P.; Yu, Z. C.; Wang, L. F.; Zhou, Y.; Wu, Y. D.; Ma, Y.; Wu, A. X. I2-Promoted In Situ Cyclization–Rethiolation Reaction: Synthesis of 2-Aliphatic- or Aromatic-Substituted Indolizines. J. Org. Chem. 2022, 87, 15197-15209. 

  49.  Yu, Z. C.; Zhou, Y.; Chen, X. L.; Ma, J. T.; Wang, L. S.; Wu, Y. D.; Wu, A. X. One-Pot Synthesis of Diaryl 1,2-Diketones via Zn-Mediated Reductive Coupling. J. Org. Chem. 2022, 87, 14037-14044. 

  50.  Chen, X. L.; Wang, H. Y.; Wu, C. Y.; Tang, B. C.; Hu, Y. L.; Ma, J. T.; Zhuang, S. Y.; Yu, Z. C.; Wu, Y. D.; Wu, A. X. Synthesis of Tetrahydro-2H-thiopyran 1,1-Dioxides via [1+1+1+1+1+1] Annulation: An Unconventional Usage of a Tethered C–S Synthon. Org. Lett. 2022, 24, 7659-7664. 

  51. Tang, Y. X.; Zhuang, S. Y.; Liu, J. Y.; Chen, X. L.; Zhou, Y.; Wu, Y. D.; Wu, A. X. I2-DMSO Mediated N1/C5 Difunctionalization of Anthranils with Aryl Methyl Ketones: A Facile Access to Multicarbonyl Compounds. Tetrahedron 2022, 126, 133057. 

  52.  Zhu, Y. P.; Zhou, Y.; Li, W. J.; Liu, F. R.; Wang, W. C.; Hao, K. Y.; Chao, B. Y.; Shi, T. R.; Wu, A. X.; Sun, Y. Y. Iodine-Promoted Oxidative Cyclization of Methyl Azaarenes and Α-Amino Ketones for One-Pot Synthesis of 2-Azaaryl-5-aryl Oxazoles. J. Org. Chem. 2022, 87, 12460-12469. 

  53. Ma, J. T.; Chen, T.; Chen, X. L.; Zhou, Y.; Yu, Z. C.; Zhuang, S. Y.; Alimu, M.; Wu, Y. D.; Xiang, J. C.; Wu, A. X. One-step Synthesis of Azepino[3,4-b]indoles by Cooperative Aza-[4 + 3] Cycloaddition from Readily Available Feedstocks. Org. Chem. Front. 2022, 9, 4640-4648. 

  54.  Zhou, Y.; Wang, L. S.; Lei, S. G.; Gao, Y. X.; Ma, J. T.; Yu, Z. C.; Wu, Y. D.; Wu, A. X. I2-Promoted Site-selective C–C Bond Cleavage of Aryl Methyl Ketones as C1 Synthons for Constructing 5-acyl-1H-pyrazolo[3,4-b]pyridines. Org. Chem. Front. 2022, 9, 4416-4420. 

  55.  Wu, C. Y.; He, C.; Chen, X. L.; Tang, B. C.; Yu, Z. C.; Wang, H. Y.; Wu, Y. D.; Wu, A. X. Pd-Catalyzed Hydroxyl-Directed Cascade Hydroarylation/C–H Germylation of Nonterminal Alkenes and Aryl Iodides. J. Org. Chem. 2022, 87, 9184-9196. 

  56.  Wang, L. S.; Zhou, Y.; Lei, S. G.; Yu, X. X.; Huang, C.; Wu, Y. D.; Wu, A. X. Iodine-Mediated Multicomponent Cascade Cyclization and Sulfenylation/Selenation: Synthesis of Imidazo[2,1-a]isoquinoline Derivatives. Org. Lett. 2022, 24, 4449-4453. 

  57.  Zhuang, S. Y.; Tang, Y. X.; Liu, J. Y.; Chen, X. L.; Ma, J. T.; Wu, Y. D.; Zheng, K. L.; Wu, A. X. I2-DMSO-Mediated N–H/α-C(sp3)–H Difunctionalization of Tetrahydroisoquinoline: Formal [2 + 2 + 1] Annulation for the Construction of Pyrrolo[2,1-a]isoquinoline Derivatives. Org. Lett. 2022, 24, 2858-2862. 

  58.  Zhang, X. K.; Miao, X. Y.; Zhou, Y.; Wang, Y. M.; Song, Y. C.; Liu, H.; Xiong, Y. L.; Li, L. Y.; Wu, A. X.; Zhu, Y. P. Iodine-catalyzed Oxidative Annulation: Facile Synthesis of Pyrazolooxepinopyrazolones via Methyl Azaarene Sp3 C–H Functionalization. Org. Biomol. Chem. 2022, 20, 1236-1242. 

  59.  Zhang, X. K.; Miao, X. Y.; Zhou, Y.; Wang, Y. M.; Song, Y. C.; Liu, H.; Xiong, Y. L.; Li, L. Y.; Wu, A. X.; Zhu, Y. P. Iodine-catalyzed Oxidative Annulation: Facile Synthesis of Pyrazolooxepinopyrazolones via Methyl Azaarene Sp3 C–H Functionalization. Org. Biomol. Chem. 2022, 20, 1236-1242. 

  60.  Huang, C.; Zhou, Y.; Yu, X. X.; Wang, L. S.; Wu, Y. D.; Wu, A. X. I2/CuCl2-Copromoted Formal [4 + 1 + 1] Cyclization of Methyl Ketones, 2-Aminobenzonitriles, and Ammonium Acetate: Direct Access to 2-Acyl-4-aminoquinazolines. J. Org. Chem. 2021, 86, 16916-16925.

  61.  Zhuang, S. Y.; Tang, Y. X.; Chen, X. L.; Wu, Y. D.; Wu, A. X. Copper-Catalyzed Oxidative C(sp3)–H/C(sp3)–H Cross-Coupling Reaction of 3-Methylbenzo[c]isoxazoles with Methyl Ketones: Access to Indigoid Analogues. J. Org. Chem. 2021, 86, 17101-17109. 

  62.  Huang, C.; Geng, X.; Zhao, P.; Zhou, Y.; Yu, X. X.; Wang, L. S.; Wu, Y. D.; Wu, A. X. Direct Synthesis of 4-Aryl-1,2,3-triazoles via I<sub>2</sub>-Promoted Cyclization Under Metal- and Azide-Free Conditions. J. Org. Chem. 2021, 86, 13664-13672. 

  63.  Yu, X. X.; Zhao, P.; Zhou, Y.; Huang, C.; Wang, L. S.; Wu, Y. D.; Wu, A. X. Iodine-Promoted Formal [3+2] Cycloaddition of Enaminone: Access to 2-Hydroxy-1,2-dihydro-pyrrol-3-ones with Quaternary Carbon Center. J. Org. Chem. 2021, 86, 12141-12147. 

  64. Zhou, Y.; Zhao, P.; Wang, L. S.; Yu, X. X.; Huang, C.; Wu, Y. D.; Wu, A. X. Direct C–C Bond Cleavage of 1,3-Dicarbonyl Compounds as a Single-Carbon Synthon: Synthesis of 2-Aryl-4-quinolinecarboxylates. Org. Lett. 2021, 23, 6461-6465. 

  65.  Yu, X. X.; Zhao, P.; Zhou, Y.; Huang, C.; Wang, L. S.; Wu, Y. D.; Wu, A. X. Employing Arylacetylene as a Diene Precursor and Dienophile: Synthesis of Quinoline via the Povarov Reaction. J. Org. Chem. 2021, 86, 8381-8388. 

  66.  He, C.; Chen, X.; Zhuang, S.; Wu, Y.; Tang, B.; Wu, A. Palladium‐Catalyzed Heck/Insertion/Decarboxylation Domino Sequence: Synthesis of Dihydrocyclohepta[de]naphthalenes. Adv Synth Catal 2021, 363, 3476-3480. 

  67. Ma, J. T.; Wang, L. S.; Chai, Z.; Chen, X. F.; Tang, B. C.; Chen, X. L.; He, C.; Wu, Y. D.; Wu, A. X. Access to 2-arylquinazolines via Catabolism/reconstruction of Amino Acids with the Insertion of Dimethyl Sulfoxide. Chem. Commun. 2021, 57, 5414-5417. 

  68. Zhuang, S. Y.; Tang, Y. X.; Chen, X. L.; Wu, Y. D.; Wu, A. X. I2-DMSO Mediated Oxidative Amidation of Methyl Ketones with Anthranils for the Synthesis of α-ketoamides. Org. Biomol. Chem. 2021, 19, 4258-4262. 

  69. Xu, C.; Yin, G.; Jia, F. C.; Wu, Y. D.; Wu, A. X. Merging Annulation with Ring Deconstruction: Synthesis of (E)-3-(2-Acyl-1H-benzo[d]imidazol-4-yl)acrylaldehyde Derivatives via I2/FeCl3-Promoted Dual C(sp3)–H Amination/C–N Bond Cleavage. Org. Lett. 2021, 23, 2559-2564. 

  70. Zhuang, S.; Tang, Y.; He, C.; Chen, X.; Xue, W.; Wu, Y.; Wu, A. Copper‐catalyzed Reaction of Anthranils with Methyl Ketones: Site‐Selective C5‐Dicarbonylation of Anthranils. Adv Synth Catal 2020, 363, 1137-1141. 

  71.  Tang, B. C.; He, C.; Chen, X. L.; Ma, J. T.; Wang, M.; Wu, Y. D.; Wu, A. X. Palladium Catalyzed Annulation of 2-iodobiphenyl with a Non-terminal Alkene Enabled by Neighboring Group Assistance. Chem. Commun. 2021, 57, 121-124. 

  72. Tang, B. C.; Lin, W. X.; Chen, X. L.; He, C.; Ma, J. T.; Wu, Y. D.; Lan, Y.; Wu, A. X. Quadruple C-H Activation Coupled to Hydrofunctionalization and C-H Silylation/borylation Enabled by Weakly Coordinated Palladium Catalyst. Nat. Commun. 2020, 11，5662.

  73.  Zhou, Y.; Zhao, P.; Yu, X. X.; Geng, X.; Wang, C.; Huang, C.; Yang, H.; Zhao, Z. Y.; Wu, A. X. Radical Tandem Bicyclization Triggered by the Α-Position of Α,β-Unsaturated Ketones Bearing Nonterminal 1,6-Enynes: Synthesis of the 5H-Benzo[a]fluoren-5-one Skeleton. Org. Lett. 2020, 22, 8359-8364. 

  74.  Zhao, P.; Zhou, Y.; Yu, X. X.; Huang, C.; Wu, Y. D.; Yin, G.; Wu, A. X. Iodine-Promoted Multicomponent Synthesis of 2,4-Diamino-1,3,5-triazines. Org. Lett. 2020, 22, 8528-8532. 

  75.  Zhao, P.; Yu, X. X.; Zhou, Y.; Huang, C.; Wu, Y. D.; Zhu, Y. P.; Wu, A. X. Arylacetylenes as Two-carbon Synthons: Synthesis of Eight-membered Rings via CC Bond Cleavage. Chem. Commun. 2020, 56, 12554-12557. 

  76.  Chen, X. L.; Tang, B. C.; He, C.; Ma, J. T.; Zhuang, S. Y.; Wu, Y. D.; Wu, A. X. Rongalite as a Sulfone Source: a Novel Copper-catalyzed Sulfur Dioxide Anion Incorporation Process. Chem. Commun. 2020, 56, 13653-13656. 

  77.  Zhao, P.; Yu, X. X.; Zhou, Y.; Geng, X.; Wang, C.; Huang, C.; Wu, Y. D.; Zhu, Y. P.; Wu, A. X. Splitting Methyl Ketones into Two Parts: Synthesis of 4(3H)-Quinazolinones via Consecutive Cyclization/Ring-Opening Reaction. Org. Lett. 2020, 22, 7103-7107. 

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