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化学制药工艺研究,尤其是绿色制药过程的开发 新药的研究与开发

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1. 黄文才,张丹,程度,张春红,陈文芝,雷华.一种三水合3-氨基丙基胺乙基硫代磷酸的合成方法. 中国发明专利,ZL201110152336.6,2014-02-26. 2. Junqiang Liu, Chenggen Mi, Xuemei Tang, Yuan Cao, Zicheng Li, Wencai Huang*. Facile microwave-assisted synthesis of substituted benzofuran derivatives. Res Chem Intermed, 2014, 40(5): 2083-2090. 3. 米成根, 唐雪梅, 刘俊强, 程度, 黄文才*.磷酸肌酸钠的合成.中国医药工业杂志. 2013,44(8):741-743. 4. 雷华,张春红,米成根,程度,黄文才*.氨磷汀的合成.中国医药工业杂志. 2012,43(8):649-650. 5. Li Yang, Hua Lei, Cheng-Gen Mi, Huan Liu, Tian Zhou, Ying-Lan Zhao, Xiao-Yun Lai, Zi-Cheng Li, Hang Song, Wen-Cai Huang*. Synthesis, antiproliferative activities and in vitro biological evaluation of novel benzofuransulfonamide derivatives. Bioorg Med Chem Lett, 2011, 21(18): 5389-5392. IF2.538 6. Sun Qiu, Luo Xin-feng, Yin Hai-bin, Huang Wen-cai*. Iron Trichloride-Assisted Selective Synthesis of 4-(2, 6-di-tert-butyl-4-(2-(3,5-di-tert-butyl-4-hydroxyphenylthio)propan-2-ylthio)phenoxy)-4-oxobutanoic acid. 化学研究与应用,2011, 23(5):559-563. 7. Xin-Feng Luo, Ling He, Hai-Bin Yin, Hu Zheng, Di Bei, Jin-Jin Deng, Wen-Cai Huang*. Efficient Acylation and One-Pot Synthesis of Dehydroandrographolide Succinate on a Large Scale Assisted with Microwave Radiation. Synth Commun, 2009, 39(19): 3444–3452.

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