Original articleAnticancer activity of THMPP: Downregulation of PI3K/ S6K1 in breast cancer cell line
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Keywords
Tetrahydroquinoline
Apoptosis
Gene expression
EGFR
Docking
ADME
QSAR
Abbreviations
THMPP
2-((1, 2, 3, 4-Tetrahydroquinolin-1-yl) (4 methoxyphenyl) methyl) phenol
IC50
The half maximal inhibitory concentration
FITC
Fluorescein isothiocyanate
AO/EtBr
Acridine orange/ethidium bromide
RTPCR
Reverse Transcriptase PCR
QSAR
Quantitative structure activity relationship
ADME-Absorption
Distribution, Metabolism, and Excretion
MCF-7
Michigan Cancer Foundation-7
SkBr3
Sloan–Kettering Cancer Center
EGFR
Epidermal Growth Factor Receptor
ER
Estrogen Receptor
PR
Progesterone Receptor
PI3K
Phosphoinositide 3-kinase
FACS
Fluorescence-activated cell sorting
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Peer review under responsibility of King Saud University.
© 2020 The Author(s). Published by Elsevier B.V. on behalf of King Saud University.