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Notoginsenoside R1 promotes Lgr5+ stem cell and epithelium renovation in colitis mice via activating Wnt/β-Catenin signaling Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-03-15 Zhi-lun Yu, Rui-yang Gao, Cheng Lv, Xiao-long Geng, Yi-jing Ren, Jing Zhang, Jun-yu Ren, Hao Wang, Fang-bin Ai, Zi-yi Wang, Bei-bei Zhang, Dong-hui Liu, Bei Yue, Zheng-tao Wang, Wei Dou
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Angiotensin II type-2 receptor signaling facilitates liver injury repair and regeneration via inactivation of Hippo pathway Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-03-15 Chang-yong Xu, Ji Jiang, Yue An, Peng-fei Ye, Cun-cun Zhang, Ning-ning Sun, Sai-nan Miao, Meng-qi Chai, Wen-min Liu, Mei Yang, Wei-hua Zhu, Jing-jing Yu, Man-man Yu, Wu-yi Sun, Huan Qiu, Shi-hao Zhang, Wei Wei
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Prenatal dexamethasone exposure impairs rat blood-testis barrier function and sperm quality in adult offspring via GR/KDM1B/FSTL3/TGFβ signaling Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-03-12 Yi Liu, Si-jia Chen, Can Ai, Peng-xia Yu, Man Fang, Hui Wang
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Clobetasol propionate, a Nrf-2 inhibitor, sensitizes human lung cancer cells to radiation-induced killing via mitochondrial ROS-dependent ferroptosis Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-03-13 Archita Rai, Raghavendra S. Patwardhan, Sundarraj Jayakumar, Pradnya Pachpatil, Dhruv Das, Girish Ch. Panigrahi, Vikram Gota, Sejal Patwardhan, Santosh K. Sandur
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zDHHC20-driven S-palmitoylation of CD80 is required for its costimulatory function Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-03-11 Bin Lu, Yi-yun Sun, Bo-ya Chen, Bo Yang, Qiao-jun He, Jun Li, Ji Cao
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HBB contributes to individualized aconitine-induced cardiotoxicity in mice via interfering with ABHD5/AMPK/HDAC4 axis Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-03-11 Ya-juan Guo, Jing-jing Yao, Zhen-zhen Guo, Ming Ding, Kun-lin Zhang, Qing-hong Shen, Yu Li, Shao-fang Yu, Ting Wan, Fu-ping Xu, Ying Wang, Xiao-xiao Qi, Jin-jun Wu, Jian-xin Chen, Zhong-qiu Liu, Lin-lin Lu
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Macrod1 suppresses diabetic cardiomyopathy via regulating PARP1-NAD+-SIRT3 pathway Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-03-08 Yu-ting Liu, Hong-liang Qiu, Hong-xia Xia, Yi-zhou Feng, Jiang-yang Deng, Yuan Yuan, Da Ke, Heng Zhou, Yan Che, Qi-zhu Tang
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A novel mouse model of familial combined hyperlipidemia and atherosclerosis Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-03-08 Mei-jie Chen, Yi-tong Xu, Lu Sun, Zhi-hua Wang, Peter J. Little, Li Wang, Xun-de Xian, Jian-ping Weng, Suo-wen Xu
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Intestinal epithelial Krüppel-like factor 4 alleviates endotoxemia and atherosclerosis through improving NF-κB/miR-34a-mediated intestinal permeability Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-03-04 He-zhong-rong Nie, Yi-wen Zhou, Xiao-hong Yu, Cong-guo Yin, Ling-fei Li, Hui-qin Hao, Tao Yuan, Yong Pan
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Discovery of a selective TRF2 inhibitor FKB04 induced telomere shortening and senescence in liver cancer cells Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-03-04 Yin-da Qiu, Qi Yan, Yi Wang, Yan-fei Ye, Yan Wang, Meng-ying Wang, Pei-pei Wang, Shu-yuan Zhang, Da-long Wang, Hao Yan, Jing Ruan, Yun-jie Zhao, Le-hao Huang, Namki Cho, Kun Wang, Xiao-hui Zheng, Zhi-guo Liu
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α4 nicotinic receptors on GABAergic neurons mediate a cholinergic analgesic circuit in the substantia nigra pars reticulata Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-03-04 Yu Han, Jia-qi Zhang, Ya-wei Ji, Yi-wen Luan, Shu-yi Li, Hui-zhen Geng, Ying Ji, Cui Yin, Su Liu, Chun-yi Zhou, Cheng Xiao
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Brigatinib, a newly discovered AXL inhibitor, suppresses AXL-mediated acquired resistance to osimertinib in EGFR-mutated non-small cell lung cancer Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-03-04 Rui Han, Cong-hua Lu, Chen Hu, Yuan-yao Dou, Jun Kang, Cai-yu Lin, Di Wu, Wei-ling Jiang, Guo-qing Yin, Yong He
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PHPB ameliorates memory deficits and reduces oxidative injury in Alzheimer’s disease mouse model by activating Nrf2 signaling pathway Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-02-26 Nian-ying Shang, Long-jian Huang, Jia-qi Lan, Yu-ying Kang, Jing-shu Tang, Hong-yue Wang, Xin-nan Li, Zhuo Sun, Qiu-yu Chen, Meng-yao Liu, Zi-peng Wen, Xin-hong Feng, Lei Wu, Ying Peng
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Proteomics analysis of histone deacetylase inhibitor-resistant solid tumors reveals resistant signatures and potential drug combinations Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-02-21 Bing-bing Hao, Ke Ma, Jun-yu Xu, Ru-feng Fan, Wen-si Zhao, Xing-long Jia, Lin-hui Zhai, SangKyu Lee, Dong Xie, Min-jia Tan
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Inflammation-related molecular signatures involved in the anticancer activities of brigatinib as well as the prognosis of EML4-ALK lung adenocarcinoma patient Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-02-15 Fu-jing Ge, Xiao-yang Dai, Yao Qiu, Xiang-ning Liu, Chen-ming Zeng, Xiao-yuan Xu, Yi-dan Chen, Hong Zhu, Qiao-jun He, Ren-hua Gai, Sheng-lin Ma, Xue-qin Chen, Bo Yang
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Quantitative systems pharmacology modeling of HER2-positive metastatic breast cancer for translational efficacy evaluation and combination assessment across therapeutic modalities Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-02-15 Ya-ting Zhou, Jia-hui Chu, Shu-han Zhao, Ge-li Li, Zi-yi Fu, Su-jie Zhang, Xue-hu Gao, Wen Ma, Kai Shen, Yuan Gao, Wei Li, Yong-mei Yin, Chen Zhao
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Transforming growth factor-β receptors: versatile mechanisms of ligand activation Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-02-13 Zheng-Jie Chia, Ying-nan Cao, Peter J. Little, Danielle Kamato
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Glutamatergic neurons in ventral pallidum modulate heroin addiction via epithalamic innervation in rats Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-02-07 Ruo-song Chen, Jing Liu, Yu-jun Wang, Kuan Ning, Jing-gen Liu, Zhi-qiang Liu
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Discovery of a nitroaromatic nannocystin with potent in vivo anticancer activity against colorectal cancer by targeting AKT1 Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-02-07 Han Zhang, Fei Xie, Xiao-ya Yuan, Xin-tong Dai, Yun-feng Tian, Ming-ming Sun, Si-qi Yu, Jia-you Cai, Bin Sun, Wei-cheng Zhang, Chang-liang Shan
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GPCRs involved in metabolic diseases: pharmacotherapeutic development updates Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-02-07 Cheng Jin, Hui Chen, Li Xie, Yuan Zhou, Li-li Liu, Jian Wu
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tRF3-IleAAT reduced extracellular matrix synthesis in diabetic kidney disease mice by targeting ZNF281 and inhibiting ferroptosis Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-29 Yun-yang Qiao, Jia-ling Ji, Wei-ling Hou, Gao-ting Qu, Shan-wen Li, Xing-yue Li, Ran Jin, Yin-fang Li, Hui-min Shi, Ai-qing Zhang
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Desloratadine alleviates ALS-like pathology in hSOD1G93A mice via targeting 5HTR2A on activated spinal astrocytes Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-29 Jian Lu, An-xu He, Zhuo-ying Jin, Meng Zhang, Zhong-xin Li, Fan Zhou, Lin Ma, Hong-ming Jin, Jia-ying Wang, Xu Shen
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Macrophage-specific FGFR1 deletion alleviates high-fat-diet-induced liver inflammation by inhibiting the MAPKs/TNF pathways Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-26 Yan-ni Zhao, Zhou-di Liu, Tao Yan, Ting-xin Xu, Tian-yang Jin, Yong-sheng Jiang, Wei Zuo, Kwang Youl Lee, Li-jiang Huang, Yi Wang
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Pharmacologically significant constituents collectively responsible for anti-sepsis action of XueBiJing, a Chinese herb-based intravenous formulation Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-24 Chen Cheng, Chao Ren, Mu-zi Li, Yi-hui Liu, Ren-qi Yao, Yang Yu, Xuan Yu, Jian-li Wang, Li-xue Wang, Yu-chun Leng, Hui Zhang, Fei-fei Du, Ning Dong, Feng-qing Wang, Yao Wu, Fang Xu, Xiao-mei Zhu, Gui-ping Zhang, Kai Dong, Si Liu, Xiao-qing Yao, Chuan Li, Yong-ming Yao
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Endothelial cell Orai1 is essential for endothelium-dependent contraction of mouse carotid arteries in normotensive and hypertensive mice Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-26 Xiao Li, Zhen-chuan Lei, Chun Yin Lo, Tsz Yau Jan, Chi Wai Lau, Xiao-qiang Yao
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Mammalian integrated stress responses in stressed organelles and their functions Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-24 Hao-jun Lu, Nirmala Koju, Rui Sheng
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Chronic vascular pathogenesis results in the reduced serum Metrnl levels in ischemic stroke patients Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-22 Zhu-wei Miao, Nuo Wang, Wen-jun Hu, Si-li Zheng, Dong-sheng Wang, Fu-qiang Chang, Zhi Wang, Jia-sheng Tian, Xiao-hui Dong, Tao Wu, Chao-yu Miao
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The dual function of cGAS-STING signaling axis in liver diseases Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-17 Xiao-jiao-yang Li, Jiao-rong Qu, Yin-hao Zhang, Run-ping Liu
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Mangiferin alleviates diabetic pulmonary fibrosis in mice via inhibiting endothelial-mesenchymal transition through AMPK/FoxO3/SIRT3 axis Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-15 Ting-lv Fu, Guo-rui Li, Dong-hang Li, Ru-yuan He, Bo-hao Liu, Rui Xiong, Chen-zhen Xu, Zi-long Lu, Cong-kuan Song, Hong-liang Qiu, Wen-jie Wang, Shi-shi Zou, Ke Yi, Ning Li, Qing Geng
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Targeted inhibition of the HNF1A/SHH axis by triptolide overcomes paclitaxel resistance in non-small cell lung cancer Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-16 Ling-bing Li, Ling-xiao Yang, Lei Liu, Fan-rong Liu, Alex H. Li, Yi-lin Zhu, Hao Wen, Xia Xue, Zhong-xian Tian, Hong Sun, Pei-chao Li, Xiao-gang Zhao
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CCDC92 promotes podocyte injury by regulating PA28α/ABCA1/cholesterol efflux axis in type 2 diabetic mice Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-16 Fu-wen Zuo, Zhi-yong Liu, Ming-wei Wang, Jun-yao Du, Peng-zhong Ding, Hao-ran Zhang, Wei Tang, Yu Sun, Xiao-jie Wang, Yan Zhang, Yu-sheng Xie, Ji-chao Wu, Min Liu, Zi-ying Wang, Fan Yi
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Macrophages promote the transition from myocardial ischemia reperfusion injury to cardiac fibrosis in mice through GMCSF/CCL2/CCR2 and phenotype switching Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-15 Shi-chun Shen, Jie Xu, Cheng Cheng, Xin-jian Xiang, Bao-yu Hong, Meng Zhang, Chen Gong, Li-kun Ma
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Corynoxine promotes TFEB/TFE3-mediated autophagy and alleviates Aβ pathology in Alzheimer’s disease models Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-15 Xin-jie Guan, Zhi-qiang Deng, Jia Liu, Cheng-fu Su, Benjamin Chun-Kit Tong, Zhou Zhu, Sravan Gopalkrishnashetty Sreenivasmurthy, Yu-xuan Kan, Ke-jia Lu, Carol Pui-Kei Chu, Rong-biao Pi, King-ho Cheung, Ashok Iyaswamy, Ju-xian Song, Min Li
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DsbA-L ameliorates renal aging and renal fibrosis by maintaining mitochondrial homeostasis Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-10 Ming Yang, Yan Liu, Shi-lu Luo, Chong-bin Liu, Na Jiang, Chen-rui Li, Hao Zhao, Ya-chun Han, Wei Chen, Li Li, Lin Sun
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SIBP-03, a novel anti-HER3 antibody, exerts antitumor effects and synergizes with EGFR- and HER2-targeted drugs Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-10 Wen-jing Li, Cheng-ying Xie, Xi Zhu, Jiao Tang, Lei Wang, Li-guang Lou
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New horizons for the role of RNA N6-methyladenosine modification in hepatocellular carcinoma Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-09 Yu-jia Li, Yang-ling Qiu, Meng-ran Li, Min Shen, Feng Zhang, Jiang-juan Shao, Xue-fen Xu, Zi-li Zhang, Shi-zhong Zheng
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Inhibition of PPP1R15A alleviates osteoporosis via suppressing RANKL-induced osteoclastogenesis Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-08 Zong-bao Ding, Yan Chen, Yu-rong Zheng, Yi-yuan Wang, Wen-de Deng, Jie-huang Zheng, Qin Yang, Zi-ye Chen, Li-hong Li, Hui Jiang, Xiao-juan Li
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Structural and functional insights into the epigenetic regulator MRG15 Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-08 Nan Jiang, Yong-bo Li, Jia-yu Jin, Jie-yu Guo, Qiu-rong Ding, Dan Meng, Xiu-ling Zhi
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O-GlcNAcylation mediates H2O2-induced apoptosis through regulation of STAT3 and FOXO1 Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-08 Chen-chun Zhang, Yuan Li, Chang-you Jiang, Qiu-min Le, Xing Liu, Lan Ma, Fei-fei Wang
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Second messenger 2'3'-cyclic GMP-AMP (2'3'-cGAMP): the cell autonomous and non-autonomous roles in cancer progression Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-04 Xiao-yu Ma, Man-man Chen, Ling-hua Meng
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Empagliflozin ameliorates vascular calcification in diabetic mice through inhibiting Bhlhe40-dependent NLRP3 inflammasome activation Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-03 Xiao-xue Li, Zheng-dong Chen, Xue-jiao Sun, Yi-qing Yang, Hong Jin, Nai-feng Liu
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Britannin as a novel NLRP3 inhibitor, suppresses inflammasome activation in macrophages and alleviates NLRP3-related diseases in mice Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2024-01-03 Jing-jing Shao, Wei-feng Li, Jin-feng Sun, Zai-shou Zhuang, Ju-lian Min, Xiao-hong Long, Gao-jun Wu, Hao-wen Xu, Guang Liang
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Epigenetic-based combination therapy and liposomal codelivery overcomes osimertinib-resistant NSCLC via repolarizing tumor-associated macrophages Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-12-19 Ting-ting Lin, Wei Xiong, Gui-hua Chen, Yang He, Li Long, Xin-fu Gao, Jia-lin Zhou, Wen-wen Lv, Yong-zhuo Huang
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OTUD1 promotes hypertensive kidney fibrosis and injury by deubiquitinating CDK9 in renal epithelial cells Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-12-18 Meng-yang Wang, Tian-xiang Yu, Qin-yan Wang, Xue Han, Xiang Hu, Shi-ju Ye, Xiao-hong Long, Yi Wang, Hong Zhu, Wu Luo, Guang Liang
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Nucleic acid and protein methylation modification in renal diseases Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-12-15 Juan Jin, Xue-mei Liu, Wei Shao, Xiao-ming Meng
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Autoimmune diseases: targets, biology, and drug discovery Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-12-14 Shu-jie Li, Yan-li Wu, Juan-hua Chen, Shi-yi Shen, Jia Duan, H. Eric Xu
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Zonisamide attenuates pressure overload-induced myocardial hypertrophy in mice through proteasome inhibition Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-12-14 Qian Wu, Wan-jie Liu, Xin-yu Ma, Ji-shuo Chang, Xiao-ya Zhao, Ying-hua Liu, Xi-yong Yu
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Sigma-1 receptor activation mediates the sustained antidepressant effect of ketamine in mice via increasing BDNF levels Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-12-14 Hui Ma, Jin-feng Li, Xin Qiao, Yue Zhang, Xiao-juan Hou, Hai-xia Chang, Hong-lei Chen, Yong Zhang, Yun-feng Li
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Chemokine CCL2 promotes cardiac regeneration and repair in myocardial infarction mice via activation of the JNK/STAT3 axis Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-12-12 Wei Wang, Xiao-kang Chen, Lu Zhou, Feng Wang, Yan-ji He, Bing-jun Lu, Ze-gang Hu, Zhu-xin Li, Xue-wei Xia, Wei Eric Wang, Chun-yu Zeng, Liang-peng Li
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Lonicerin promotes wound healing in diabetic rats by enhancing blood vessel regeneration through Sirt1-mediated autophagy Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-12-08 Zhen Lin, Lu-yao Li, Lu Chen, Chen Jin, Yue Li, Lan Yang, Chang-zhou Li, Cai-yu Qi, Yu-yang Gan, Jia-rui Zhang, Piao Wang, Li-bin Ni, Gao-feng Wang
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SMAD4 endows TGF-β1-induced highly invasive tumor cells with ferroptosis vulnerability in pancreatic cancer Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-12-06 Hai-di Chen, Zeng Ye, Hai-feng Hu, Gui-xiong Fan, Yu-heng Hu, Zheng Li, Bo-rui Li, Shun-rong Ji, Chen-jie Zhou, Xiao-wu Xu, Xian-jun Yu, Yi Qin
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E3 ubiquitin ligase NEDD4L inhibits epithelial-mesenchymal transition by suppressing the β-catenin/HIF-1α positive feedback loop in chronic rhinosinusitis with nasal polyps Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-12-05 Si-yuan Chen, Pei-qiang Liu, Dan-xue Qin, Hao Lv, Hui-qin Zhou, Yu Xu
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From bench to bedside: current development and emerging trend of KRAS-targeted therapy Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-12-04 Yi Chen, Qiu-pei Liu, Hua Xie, Jian Ding
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Colon-targeted S100A8/A9-specific peptide systems ameliorate colitis and colitis-associated colorectal cancer in mouse models Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-12-01 Euni Cho, Seok-Jun Mun, Hyo Keun Kim, Yu Seong Ham, Woo Jin Gil, Chul-Su Yang
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A novel human single-domain antibody-drug conjugate targeting CEACAM5 exhibits potent in vitro and in vivo antitumor activity Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-11-29 Xiao-yi Zhu, Quan-xiao Li, Yu Kong, Ke-ke Huang, Gang Wang, Yun-ji Wang, Jun Lu, Guo-qiang Hua, Yan-ling Wu, Tian-lei Ying
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Schisandrin B, a dual positive allosteric modulator of GABAA and glycine receptors, alleviates seizures in multiple mouse models Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-11-28 Jun Wu, Miao Zhao, Yu-chen Jin, Min Li, Ke-xin Yu, Hai-bo Yu
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Combination of eriocalyxin B and homoharringtonine exerts synergistic anti-tumor effects against t(8;21) AML Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-11-28 Yi-chen Lei, Xin-jie Chen, Yu-ting Dai, Bing Dai, Ji-yue Wang, Miao-hui Li, Ping Liu, Han Liu, Kan-kan Wang, Lu Jiang, Bing Chen
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Amuc_1100 pretreatment alleviates acute pancreatitis in a mouse model through regulating gut microbiota and inhibiting inflammatory infiltration Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-11-27 Li-juan Wang, Yuan-ling Jin, Wen-long Pei, Jia-cong Li, Rui-lin Zhang, Jia-ju Wang, Wei Lin
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Baicalein attenuates rotenone-induced SH-SY5Y cell apoptosis through binding to SUR1 and activating ATP-sensitive potassium channels Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-11-22 De-wen Kong, Li-da Du, Run-zhe Liu, Tian-yi Yuan, Shou-bao Wang, Yue-hua Wang, Yang Lu, Lian-hua Fang, Guan-hua Du
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Lipid droplets in pathogen infection and host immunity Acta Pharmacol. Sin. (IF 8.2) Pub Date : 2023-11-22 Yan-jie Tan, Yi Jin, Jun Zhou, Yun-fan Yang