The Rh(III)-catalyzed directed CH activation/carbenoid coupling reactions for the synthesis of NH-3-aryloxindoles is described. This mild, highly efficient and time-economical coupling reaction displays excellent functional group compatibility and regioselectivity. This methodology provided the straightforward way for the synthesis of NH-3-aryloxindoles, which might be of considerable bioactivities.

中文翻译：

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一种在室温下通过Rh（III）催化的C H活化合成NH -3-芳基吲哚的简便方法

描述了用于合成NH -3-芳基吲哚的Rh（III）催化的定向C H活化/类胡萝卜素偶联反应。这种温和，高效和省时的偶联反应显示出出色的官能团相容性和区域选择性。该方法学为合成NH -3-芳基吲哚提供了直接的方法，该方法可能具有相当大的生物活性。