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Synthesis of indole-fused scaffolds via [3+3] cyclization reaction of 2-indolylmethanols with quinone imines
Tetrahedron ( IF 2.1 ) Pub Date : 2020-11-28 , DOI: 10.1016/j.tet.2020.131742 Lu-Zhe Qin , Ya-Long Cheng , Xiaoan Wen , Qing-Long Xu , Le Zhen
中文翻译:
通过2-吲哚基甲醇与醌亚胺的[3 + 3]环化反应合成吲哚稠合的支架
更新日期:2020-12-16
Tetrahedron ( IF 2.1 ) Pub Date : 2020-11-28 , DOI: 10.1016/j.tet.2020.131742 Lu-Zhe Qin , Ya-Long Cheng , Xiaoan Wen , Qing-Long Xu , Le Zhen
A formal [3 + 3] cyclization reaction of 2-indolylmethanols with quinones was realized to furnish indole-fused scaffolds in moderate to excellent yields. This protocol was proceeded smoothly under acid condition, with high high yields and broad substrate scope.
中文翻译:
通过2-吲哚基甲醇与醌亚胺的[3 + 3]环化反应合成吲哚稠合的支架
实现了2-吲哚基甲醇与醌的正式[3 + 3]环化反应,以中等至优异的产率提供了吲哚融合的支架。该方案在酸性条件下顺利进行,具有高收率和广泛的底物范围。