Both phosphinopeptides and phosphinodepsipeptides are important phosphorus analogues of naturally occurring peptides. They have been widely applied as biological active peptides, such as enzyme inhibitors, haptens for production of catalytic antibodies, and antibiotics. Synthetic methods of phosphinopeptides and phosphinodepsipeptides are reviewed and classified on the basis of the structural characteristics of aminoalkylphosphinic acids. This review focuses on the synthetic methods to phosphinopeptides and phosphinodepsipeptides, including α‐, β‐, and γ‐phosphinopeptides and α‐phosphinodepsipeptides.

中文翻译：

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磷脂肽和磷脂肽的合成

膦肽肽和膦二肽肽都是天然存在的肽的重要磷类似物。它们已被广泛用作生物活性肽，例如酶抑制剂，用于产生催化抗体的半抗原和抗生素。根据氨基烷基次膦酸的结构特征，对膦肽和膦二肽的合成方法进行了综述和分类。这篇综述着重于膦肽和膦肽肽的合成方法，包括α-，β-和γ-磷肽和α-膦肽二肽。