Straightforward synthesis of enantiomerically pure 1,2,3-triazoles derived from amino esters†,Organic & Biomolecular Chemistry

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Straightforward synthesis of enantiomerically pure 1,2,3-triazoles derived from amino esters†
Organic & Biomolecular Chemistry ( IF 3.2 ) Pub Date : 2018-04-03 00:00:00 , DOI: 10.1039/c8ob00533h
Gastón Silveira-Dorta _{1,

2,

3,

4,

5} , Sampad Jana _{1,

2,

3,

4,

5} , Lucie Borkova _{6,

7,

8,

9,

10} , Joice Thomas _{1,

2,

3,

4,

5} , Wim Dehaen _{1,

2,

3,

4,

5}

Affiliation

A practical and straightforward approach that enables, for the first time, the synthesis of enantiomerically pure 1,4,5-trisubstituted, 1,5-disubstituted, and fused 1,2,3-triazole derivatives has been developed. The synthesis employs enantiomerically pure amino esters derived from amino acids and commercially available ketones under metal-free conditions.

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