Pd-catalyzed C–H arylation of benzothioamides with boronic acids using thioamides as directing groups,Organic Chemistry Frontiers

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Pd-catalyzed C–H arylation of benzothioamides with boronic acids using thioamides as directing groups
Organic Chemistry Frontiers ( IF 5.4 ) Pub Date : 2017-08-04 00:00:00 , DOI: 10.1039/c7qo00532f
Kai-Xiang Tang _{1,

2,

3,

4,

5} , Chun-Meng Wang _{1,

2,

3,

4,

5} , Tian-Hong Gao _{1,

2,

3,

4,

5} , Cong Pan _{1,

2,

3,

4,

5} , Li-Ping Sun _{1,

2,

3,

4,

5}

Affiliation

The Pd(II)-catalyzed C–H arylation of benzothioamides with boronic acids using thioamides as directing groups, prevalent organic motifs found in vital biological and pharmaceutical molecules, has been achieved for the first time. The reactions proceed with high functional group tolerance in yields of 21–84%.

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