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N1-Arylation of 1,4-Benzodiazepine-2-ones with Diaryliodonium Salts
Synlett ( IF 2 ) Pub Date : 2017-09-25 , DOI: 10.1055/s-0036-1590920 Raysa Khan 1 , Robert Felix 2 , Paul Kemmitt 3 , Simon Coles 4 , Graham Tizzard 4 , John Spencer 1
Synlett ( IF 2 ) Pub Date : 2017-09-25 , DOI: 10.1055/s-0036-1590920 Raysa Khan 1 , Robert Felix 2 , Paul Kemmitt 3 , Simon Coles 4 , Graham Tizzard 4 , John Spencer 1
Affiliation
A library of N 1-arylated 5-phenyl-1,3-dihydro-2 H -1,4-benzodiazepin-2-ones has been synthesized starting with unsymmetrical diaryliodonium salts using aqueous ammonia as a base. This can also be applied to a similar 1,3,4-benzotriazepin-2-one derivative.
中文翻译:
1,4-苯并二氮杂-2-酮与二芳基碘盐的N1-芳基化
N 1-芳基化 5-苯基-1,3-dihydro-2 H -1,4-benzodiazepin-2-ones 库已合成开始使用不对称二芳基碘盐使用氨水作为碱。这也可以应用于类似的 1,3,4-benzotriazepin-2-one 衍生物。
更新日期:2017-09-25
中文翻译:
1,4-苯并二氮杂-2-酮与二芳基碘盐的N1-芳基化
N 1-芳基化 5-苯基-1,3-dihydro-2 H -1,4-benzodiazepin-2-ones 库已合成开始使用不对称二芳基碘盐使用氨水作为碱。这也可以应用于类似的 1,3,4-benzotriazepin-2-one 衍生物。